1-acylglycerol-3-phosphate O-acyltransferase beta Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	6-(5-Chloro-2-ethoxyphenyl)-4-N-(4-chlorophenyl)pyrimidine-2,4-diamine	IC50	17.0 [1]
	6-(5-Chloro-2-methoxyphenyl)-4-N-(4-chlorophenyl)pyrimidine-2,4-diamine	IC50	54.0 [1]
	6-(5-Chloro-2-methoxyphenyl)-2-N-(4-chlorophenyl)pyrimidine-2,4-diamine	IC50	2050.0 [1], 7000.0 [2]
	2-(5-Chloro-2-methoxyphenyl)-4-N-(4-chlorophenyl)pyrimidine-4,6-diamine	IC50	7000.0 [1]
	4-(1,3-Benzothiazol-2-yl)-2-methylaniline	IC50	40000.0 [1]
	Unii-5TT4A4mblr	IC50	60.0 [1]
	N-[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-propionamide	IC50	1500.0 [1]
	2,4-Pyrimidinediamine, 6-(5-chloro-2-methylphenyl)-N4-(4-(trifluoromethyl)phenyl)-	IC50	140.0 [1]
	6-(5-Chloro-2-ethoxy-phenyl)-N-(4-chloro-phenyl)-[1,3,5]triazine-2,4-diamine	IC50	260.0 [1]
	(4-Chloro-3-(1,5-dimethyl-1H-benzoimidazol-2-yl)-phenyl)-carbamic Acid Methyl Ester	IC50	11000.0 [1]
	N-[4-Chloro-3-(5-chloro-benzooxazol-2-yl)-phenyl]-2-cyano-acetamide	IC50	27.0 [1]
	[4-Chloro-3-(5-trifluoromethyl-benzooxazol-2-yl)-phenyl]-carbamic acid prop-2-ynyl ester	IC50	140.0 [1]
	(4-Chloro-3-(5-trifluoromethyl-benzothiazol-2-yl)-phenyl)-carbamic Acid Prop-2-ynyl Ester	IC50	15.0 [1]
	[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	1000.0 [1]
	(4-Chloro-3-(5-chloro-benzooxazol-2-yl)-phenyl)-carbamic Acid Prop-2-ynyl Ester	IC50	35.0 [1]
	2-Azido-N-[4-chloro-3-(5-chloro-benzooxazol-2-yl)-phenyl]-acetamide	IC50	170.0 [1]
	6-(5-Chloro-2-methoxy-phenyl)-N-(4-chloro-phenyl)-[1,3,5]triazine-2,4-diamine	IC50	45.0 [1]
	(4-Chloro-3-(5-trifluoromethyl-benzothiazol-2-yl)-phenyl)-carbamic Acid Methyl Ester	IC50	200.0 [1]
	[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid prop-2-ynyl ester	IC50	190.0 [1]
	[4-Chloro-3-(5-chloro-1-methyl-1H-benzoimidazol-2-yl)-phenyl]-carbamic acid prop-2-ynyl ester	IC50	60.0 [1]
	Benzenemethanol, 4-((2-amino-6-(5-chloro-2-ethoxyphenyl)-4-pyrimidinyl)amino)-	IC50	75.0 [1]
	6-(5-Chloro-2-ethoxyphenyl)-4-N-(4-nitrophenyl)pyrimidine-2,4-diamine	IC50	10.0 [1]
	4-(5-Chloro-2-methoxy-phenyl)-N-p-tolyl-pyridine-2,6-diamine	IC50	240.0 [1]
	6-(5-Chloro-2-methoxyphenyl)-2-N-(4-chlorophenyl)pyridine-2,4-diamine	IC50	6500.0 [1]
	6-(5-Chloro-2-methoxyphenyl)-4-N-(1H-indazol-6-yl)pyrimidine-2,4-diamine	IC50	80.0 [1]
	4-N-(4-Bromophenyl)-6-(5-chloro-2-methylphenyl)pyrimidine-2,4-diamine	IC50	34.0 [1]
	4-[6-Amino-4-(5-chloro-2-ethoxy-phenyl)-pyridin-2-ylamino]-benzaldehyde	IC50	50.0 [1]
	4-(5-Chloro-2-ethoxy-phenyl)-N-(4-chloro-phenyl)-pyridine-2,6-diamine	IC50	50.0 [1]
	4-(5-Chloro-2-ethoxy-phenyl)-N-p-tolyl-pyridine-2,6-diamine	IC50	490.0 [1]
	4-[6-Amino-4-(5-chloro-2-methoxy-phenyl)-pyridin-2-ylamino]-benzaldehyde	IC50	260.0 [1]
	4-N-(4-Bromophenyl)-6-(5-chloro-2-methoxyphenyl)pyrimidine-2,4-diamine	IC50	28.0 [1]
	6-(5-Chloro-2-methylphenyl)-4-N-(4-chlorophenyl)pyrimidine-2,4-diamine	IC50	22.0 [1]
	6-(5-Chloro-2-methoxyphenyl)-4-N-(4-chlorophenyl)pyridine-2,4-diamine	IC50	18000.0 [1]
	6-(5-Chloro-2-ethoxyphenyl)-4-N-(1H-indazol-6-yl)pyrimidine-2,4-diamine	IC50	24.0 [1]
	{4-[6-Amino-4-(5-chloro-2-ethoxy-phenyl)-pyridin-2-ylamino]-phenyl}-methanol	IC50	99.0 [1]
	N-(4-Bromo-phenyl)-2-(5-chloro-2-methoxy-phenyl)-pyrimidine-4,6-diamine	IC50	8000.0 [1]
	6-(5-Bromo-2-methylphenyl)-4-N-(4-bromophenyl)pyrimidine-2,4-diamine	IC50	18.0 [1]
	4-(5-Chloro-2-methoxy-phenyl)-N-(4-chloro-phenyl)-pyridine-2,6-diamine	IC50	40.0 [1]
	6-(5-Bromo-2-methylphenyl)-4-N-(4-chlorophenyl)pyrimidine-2,4-diamine	IC50	31.0 [1]
	2-{4-[2-Amino-6-(5-chloro-2-ethoxy-phenyl)-pyrimidin-4-ylamino]-phenyl}-ethanol	IC50	28.0 [1]
	6-(5-Chloro-2-methoxyphenyl)-4-N-(4-methylphenyl)pyridine-2,4-diamine	IC50	40000.0 [1]
	4-N-(4-Chlorophenyl)-6-(2,5-dichlorophenyl)pyrimidine-2,4-diamine	IC50	20.0 [1]
	2-(5-Chloro-2-methoxy-phenyl)-N-(1H-indazol-6-yl)-pyrimidine-4,6-diamine	IC50	2100.0 [1]
	3-{4-[2-Amino-6-(5-chloro-2-ethoxy-phenyl)-pyrimidin-4-ylamino]-phenyl}-propan-1-ol	IC50	230.0 [1]
	6-(5-Chloro-2-methoxyphenyl)-2-N-(4-methylphenyl)pyridine-2,4-diamine	IC50	29000.0 [1]
	6-(5-Chloro-2-methoxyphenyl)-2-N-(1H-indazol-6-yl)pyrimidine-2,4-diamine	IC50	800.0 [1]
	N*4*-(4-Chloro-phenyl)-6-phenyl-pyrimidine-2,4-diamine	IC50	1100.0 [1]
	2-[2-Amino-6-(4-chloro-phenylamino)-pyrimidin-4-yl]-4-bromo-phenol	IC50	450.0 [1]
	2-[2-Amino-6-(4-chloro-phenylamino)-pyrimidin-4-yl]-4-chloro-phenol	IC50	10000.0 [1]
	N-[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-butyramide	IC50	2500.0 [1]
	N-[4-Chloro-3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]acetamide	IC50	2500.0 [1]
	1-{4-[2-Amino-6-(5-bromo-2-ethoxyphenyl)pyrimidin-4-ylamino]phenyl}ethanone	IC50	34.0 [1]
	(NZ)-N-[1-[4-[[2-amino-6-(5-bromo-2-ethoxyphenyl)pyrimidin-4-yl]amino]phenyl]ethylidene]hydroxylamine	IC50	84.0 [1]
	4-[2-Amino-6-(5-bromo-2-ethoxy-phenyl)-pyrimidin-4-ylamino]-phenyl-boronic acid	IC50	91.0 [1]
	4-[2-Amino-6-(5-bromo-2-ethoxy-phenyl)-pyrimidin-4-ylamino]-N-hydroxy-benzamide	IC50	88.0 [1]
	4-[2-Amino-6-(5-bromo-2-ethoxy-phenyl)-pyrimidin-4-ylamino]-benzamide	IC50	750.0 [1]
	But-2-ynyl N-[4-chloro-3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]carbamate	IC50	75.0 [1]
	But-3-ynyl N-[4-chloro-3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]carbamate	IC50	75.0 [1]
	[3-(5-Chloro-benzooxazol-2-yl)-4-methyl-phenyl]-carbamic acid methyl ester	IC50	550.0 [1]
	4-[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenylamino]-butyronitrile	IC50	5000.0 [1]
	Methyl N-[4-chloro-3-(5-chloro-1-methylbenzimidazol-2-yl)phenyl]carbamate	IC50	650.0 [1]
	Prop-2-ynyl N-[4-chloro-3-[1-methyl-5-(trifluoromethyl)benzimidazol-2-yl]phenyl]carbamate	IC50	120.0 [1]
	Prop-2-ynyl N-[4-chloro-3-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]phenyl]carbamate	IC50	5200.0 [1]
	[4-Chloro-3-(6-methyl-benzothiazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	64000.0 [1]
	[4-Chloro-3-(4-methyl-benzothiazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	9000.0 [1]
	2-(2-Chloro-5-methoxycarbonylamino-phenyl)-benzooxazole-5-carboxylic acid	IC50	20000.0 [1]
	N-(3-Benzothiazol-2-yl-4-methyl-phenyl)-2-cyano-acetamide	IC50	70.0 [1]
	N-[4-Chloro-3-(5-trifluoromethyl-benzothiazol-2-yl)-phenyl]-2-cyano-acetamide	IC50	50.0 [1]
	1-[4-Chloro-3-(5-chloro-benzooxazol-2-yl)-phenyl]-3-methyl-urea	IC50	950.0 [1]
	1-[4-Chloro-3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-3-prop-2-ynylurea	IC50	100.0 [1]
	[4-Chloro-3-(5-hydroxy-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	20000.0 [1]
	N-[4-Chloro-3-(5-chloro-benzooxazol-2-yl)-phenyl]-2-methylamino-acetamide	IC50	5000.0 [1]
	2-Azido-N-[4-chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-acetamide	IC50	600.0 [1]
	N-[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-benzamide	IC50	40000.0 [1]
	N-[4-Chloro-3-(5-chloro-benzooxazol-2-yl)-phenyl]-2-dimethylamino-acetamide	IC50	5000.0 [1]
	Prop-2-ynyl N-[3-(5-chloro-1,3-benzoxazol-2-yl)-4-methylphenyl]carbamate	IC50	100.0 [1]
	Prop-2-ynyl N-[4-chloro-3-(5-hydroxy-1,3-benzoxazol-2-yl)phenyl]carbamate	IC50	2000.0 [1]
	[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid isopropyl ester	IC50	16000.0 [1]
	[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid propyl ester	IC50	12000.0 [1]
	[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid allyl ester	IC50	1400.0 [1]
	N-[4-Chloro-3-(5-chloro-1-methylbenzimidazol-2-yl)phenyl]-2-cyanoacetamide	IC50	300.0 [1]
	[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid ethyl ester	IC50	1500.0 [1]
	[3-(5-Chloro-benzothiazol-2-yl)-4-methyl-phenyl]-carbamic acid prop-2-ynyl ester	IC50	15.0 [1]
	Methyl N-[4-chloro-3-(1,6-dimethylbenzimidazol-2-yl)phenyl]carbamate	IC50	20000.0 [1]
	[4-Chloro-3-(4-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	500.0 [1]
	N-[4-Chloro-3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]pent-4-ynamide	IC50	500.0 [1]
	N-[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-formamide	IC50	5000.0 [1]
	N-[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-2-cyano-acetamide	IC50	100.0 [1]
	N-[4-Chloro-3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]pent-4-ynamide	IC50	100.0 [1]
	[4-Fluoro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	64000.0 [1]
	[3-(5-Methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	64000.0 [1]
	[4-Methoxy-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	64000.0 [1]
	[4-Chloro-3-(5-phenyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	64000.0 [1]
	[4-Chloro-3-(5-trifluoromethyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	800.0 [1]
	[4-Chloro-3-(6-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester	IC50	400.0 [1]
	N-[4-Chloro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-2-hydroxy-acetamide	IC50	31000.0 [1]
	N-[4-Chloro-3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]but-2-ynamide	IC50	20000.0 [1]
	N-[4-Chloro-3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]but-2-ynamide	IC50	20000.0 [1]
	2-N-(4-Bromophenyl)-6-(5-chloro-2-methoxyphenyl)pyrimidine-2,4-diamine	IC50	2300.0 [1]
	4-N-(4-Chlorophenyl)-6-(5-fluoro-2-methylphenyl)pyrimidine-2,4-diamine	IC50	150.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ 1-acylglycerol-3-phosphate O-acyltransferase beta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/1-acylglycerol-3-phosphate-o-acyltransferase-beta-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ 1-acylglycerol-3-phosphate O-acyltransferase beta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/1-acylglycerol-3-phosphate-o-acyltransferase-beta-inhibitors-ic50-ki.
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