Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| CID 46215815 | IC50 | 10.0 [1] | |
| Urea, (2,3-dihydro-2-oxo-3-(1-(1H-pyrrol-2-yl)ethylidene)-1H-indol-5-yl)- | IC50 | 5.0 [1], 6.0 [2], 9.0 [3], 100.0 [4] | |
| N-[3-[[5-Bromo-4-[3-(thiophene-2-carbonylamino)propylamino]pyrimidin-2-yl]amino]phenyl]pyrrolidine-1-carboxamide | IC50 | 2.3 [1], 9.5 [2], 11.0 [3], 26.0 [4] | |
| 1-[(2R,3R)-3-[[6-(4-Amino-7-propan-2-ylpyrrolo[2,3-d]pyrimidine-5-carbonyl)pyrazin-2-yl]amino]-2-phenylpyrrolidin-1-yl]ethanone | IC50 | 200.0 [1], 300.0 [2], 320.0 [3] | |
| 1-[(2R,3R)-3-[[6-(4-Amino-7-propan-2-ylpyrrolo[2,3-d]pyrimidine-5-carbonyl)pyrazin-2-yl]amino]-2-phenylpyrrolidin-1-yl]ethanone | Ki | 1.4 [1] | |
MLA | "Quest Database™ 3-phosphoinositide dependent protein kinase-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 11 Dec. 2025, https://www.aatbio.com/data-sets/3-phosphoinositide-dependent-protein-kinase-1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 11). Quest Database™ 3-phosphoinositide dependent protein kinase-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/3-phosphoinositide-dependent-protein-kinase-1-inhibitors-ic50-ki. | |
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