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40S ribosomal protein S27 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
TC Mps1 12IC506.4 [1], 131.0 [2]
4-[(4-Amino-5-Cyano-6-Ethoxypyridin-2-Yl)amino]benzamideIC5037.0 [1], 1800.0 [2]
4-Amino-5-cyano-6-ethoxy-N-[(4-methylsulfonylphenyl)methyl]pyridine-2-carboxamideIC50568.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-phenylacetamideIC504200.0 [1]
4-Amino-N-benzyl-5-cyano-6-ethoxypyridine-2-carboxamideIC50529.0 [1]
3-[[5-(1,3-Benzodioxol-5-yl)-[1,2,4]triazolo[1,5-c]quinazolin-8-yl]amino]propan-1-olIC5010000.0 [1]
1-Methyl-2-[2-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]pyrimidin-4-yl]-6,7-dihydro-5H-pyrrolo[3,2-c]pyridin-4-oneIC5010000.0 [1]
2-{[2-Amino-5-(1,3-Benzodioxol-5-Ylmethyl)[1,2,4]triazolo[1,5-C]quinazolin-8-Yl]amino}ethanolIC5010000.0 [1]
5-(1,3-Benzodioxol-5-ylmethyl)-[1,2,4]triazolo[1,5-c]quinazoline-2,8-diamineIC5010000.0 [1]
5-(1,3-Benzodioxol-5-Ylmethyl)-10-Fluoro[1,2,4]triazolo[1,5-C]quinazolin-2-AmineIC5010000.0 [1]
5-(1,3-Benzodioxol-5-ylmethyl)-10-fluoro-8-(4-methylpiperazin-1-yl)-[1,2,4]triazolo[1,5-c]quinazolin-2-amineIC5010000.0 [1]
1-Methyl-5-[2-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]pyrimidin-4-yl]pyrrole-3-carboxamideIC5010000.0 [1]
4-Amino-2-ethoxy-6-(2-phenylethylamino)pyridine-3-carbonitrileIC503970.0 [1]
4-Amino-6-anilino-2-ethoxypyridine-3-carbonitrileIC50228.0 [1]
2-[(4S)-7-(3-Chlorophenyl)-1-oxo-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-4-yl]-N-[(1S)-1-cyclohexyl-2-(4-methylpiperazin-1-yl)ethyl]acetamideIC5010000.0 [1]
N-(2,2-Dimethylpropyl)-2-(1-oxo-7-thiophen-3-yl-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-4-yl)acetamideIC5010000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ 40S ribosomal protein S27 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.8 May2024https://www.aatbio.com/data-sets/40s-ribosomal-protein-s27-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 8). Quest Database™ 40S ribosomal protein S27 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/40s-ribosomal-protein-s27-inhibitors-ic50-ki.
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