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Acetylcholine receptor; alpha1/beta1/delta/gamma Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
NicotineIC501000.0 [1]
NicotineKi1480.0 [1], 5500.0 [2], 6270.0 [3]
BupropionIC507.9 [1], 7900.0 [2]
VareniclineIC501000.0 [1]
VareniclineKi8200.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseAcetylcholine receptor; alpha1/beta1/delta/gamma Inhibitors (IC50, Ki)." AAT Bioquest, Inc.4 Dec2025https://www.aatbio.com/data-sets/acetylcholine-receptor-alpha1-beta1-delta-gamma-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 4). Quest DatabaseAcetylcholine receptor; alpha1/beta1/delta/gamma Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/acetylcholine-receptor-alpha1-beta1-delta-gamma-inhibitors-ic50-ki.
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