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Adenosine kinase Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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5-IodotubercidinIC5026.0 [1]
5-IodotubercidinKi30.0 [1]
5-(3-Bromophenyl)-7-[6-(morpholin-4-yl)pyridin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC502.0 [1]
7-(5-Deoxy-beta-D-Ribofuranosyl)-5-Iodo-7h-Pyrrolo[2,3-D]pyrimidin-4-AmineIC509.0 [1]
ToyocamycinIC50310.0 [1], 3228494122.0 [2], 3235936569.0 [3]
SangivamycinIC50470.0 [1], 2127649080.0 [2], 2137962090.0 [3]
5-BromotubercidinIC50120.0 [1], 8317637711.0 [2], 8336811846.0 [3]
ClitocineIC5026000.0 [1]
ClitocineKi300.0 [1], 2500.0 [2], 3000.0 [3]
5-ChlorotubercidinIC50210.0 [1], 4764309868.0 [2], 4786300923.0 [3]
2-(4-Chloro-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diolIC5024.0 [1], 41667745222.0 [2], 41686938347.0 [3]
2-Methyl-5-(5-phenyl-4-phenylamino-pyrrolo[2,3-d]pyrimidin-7-yl)-tetrahydro-furan-3,4-diolIC500.5 [1]
2-Hydroxymethyl-5-(5-iodo-4-methylamino-pyrrolo[2,3-d]pyrimidin-7-yl)-tetrahydro-furan-3,4-diolIC501200.0 [1], 831763771.1 [2], 833297348.6 [3]
(2R,3R,4S,5R)-2-[4-(4-Fluoroanilino)-5-phenylpyrrolo[2,3-d]pyrimidin-7-yl]-5-methyloxolane-3,4-diolIC501.5 [1], 5.0 [2], 134.0 [3]
2-(4-Amino-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-aminomethyl-tetrahydro-furan-3,4-diolIC500.6 [1], 1659590000000.0 [2], 1666480000000.0 [3]
2-(4-Amino-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-vinyl-tetrahydro-furan-3,4-diolIC50100.0 [1], 10000000000.0 [2]
2-(4-Amino-5-bromo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC5040.0 [1], 24997697022.0 [2], 25118864315.0 [3]
7-[4-(Dimethylamino)phenyl]pyrido[2,3-d]pyrimidine-4-amineIC50773.0 [1], 10000.0 [2]
4-Pteridinamine, 7-(4-(dimethylamino)phenyl)-IC50440.0 [1], 3600.0 [2]
5-(3-Bromophenyl)-7-[6-[4-(oxan-4-yloxyimino)piperidin-1-yl]pyridin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC508.0 [1], 10.0 [2], 70.9 [3], 71.0 [4]
5'-Amino-5'-deoxyadenosineIC50170.0 [1], 6330.0 [2]
5'-DeoxytoyocamycinIC50310.0 [1], 3228494122.0 [2]
2-(4-Chloro-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methoxymethyl-tetrahydro-furan-3,4-diolIC50450.0 [1], 2238721139.0 [2]
2-(4-Amino-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methoxymethyl-tetrahydro-furan-3,4-diolIC501200.0 [1], 831763771.1 [2]
5-[4-(Dimethylamino)phenyl]-6-[(6-Morpholin-4-Ylpyridin-3-Yl)ethynyl]pyrimidin-4-AmineIC502.0 [1], 68.0 [2]
2-(4-Amino-5-bromo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-aminomethyl-tetrahydro-furan-3,4-diolIC500.2 [1], 5000350000000.0 [2]
2-Aminomethyl-5-(4-chloro-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-tetrahydro-furan-3,4-diolIC500.1 [1], 10000000000000.0 [2]
2-(5-Iodo-4-methylsulfanyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC5045.0 [1], 22222862543.0 [2]
2-(4-Chloro-5-methyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC50535.0 [1], 1868959972.0 [2]
2-Azidomethyl-5-(5-bromo-4-chloro-pyrrolo[2,3-d]pyrimidin-7-yl)-tetrahydro-furan-3,4-diolIC50100.0 [1], 10000000000.0 [2]
2-(4-Chloro-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC503.0 [1], 333350000000.0 [2]
2-(5-Bromo-4-chloro-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC5050.0 [1], 19998618696.0 [2]
2-(4-Amino-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-ethyl-tetrahydro-furan-3,4-diolIC5060.0 [1], 16664795936.0 [2]
2-(4-Amino-5-bromo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-ethyl-tetrahydro-furan-3,4-diolIC50500.0 [1], 1999861870.0 [2]
2-(4-Amino-5-bromo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-azidomethyl-tetrahydro-furan-3,4-diolIC5063.0 [1], 15874497983.0 [2]
2-(4-Chloro-5-methylsulfanyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC5070.0 [1], 14285649814.0 [2]
2-Azidomethyl-5-(4-chloro-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-tetrahydro-furan-3,4-diolIC509.0 [1], 111122000000.0 [2]
2-(4-Amino-5-methylsulfanyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC501350.0 [1], 740798339.2 [2]
2-(4-Amino-5-methyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC5016500.0 [1], 60603820.05 [2]
2-(4-Amino-5-iodo-pyrrolo[2,3-d]pyrimidin-7-yl)-5-azidomethyl-tetrahydro-furan-3,4-diolIC5035.0 [1], 28569326346.0 [2]
Ethyl 4-amino-7-[(2R,3R,4S,5R)-3,4-dihydroxy-5-methyloxolan-2-yl]pyrrolo[2,3-d]pyrimidine-5-carboxylateIC501000.0 [1], 1000000000.0 [2]
4-Amino-7-[(2R,3R,4S,5R)-3,4-dihydroxy-5-methyloxolan-2-yl]pyrrolo[2,3-d]pyrimidine-5-carboxamideIC50460.0 [1], 2172701179.0 [2]
6-(4-Methoxyphenyl)-7-[4-(dimethylamino)phenyl]pyrido[2,3-d]pyrimidine-4-amineIC5092.0 [1], 567.0 [2]
6-{2-[4-(Dimethylamino)phenyl]ethynyl}-5-phenylpyrimidin-4-amineIC5020.0 [1], 1000.0 [2]
5-(2H-1,3-Benzodioxol-5-yl)-6-{2-[4-(dimethylamino)phenyl]ethynyl}pyrimidin-4-amineIC509.0 [1], 250.0 [2]
7-(4-Dimethylamino-phenyl)-6-phenyl-pyrido[2,3-d]pyrimidin-4-ylamineIC50350.0 [1], 1500.0 [2]
(2R,3R,4S,5R)-2-[4-Amino-5-(furan-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC502000.0 [1], 5000.0 [2]
(2R,3R,4S,5R)-2-(4-Amino-5-thiophen-2-ylpyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)oxolane-3,4-diolIC505000.0 [1]
6-Ethyl-6-[4-(phenylsulfanylmethyl)phenyl]pyrrolo[2,1-d][1,5]benzoxazepin-7-oneIC501200.0 [1]
2-(5-Iodo-4-mercapto-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC506500.0 [1]
5-Phenyl-7-[4-(dimethylamino)phenyl]pyrido[2,3-d]pyrimidine-4-amineIC50467.0 [1]
(2R,3R,4S,5R)-2-(4-Amino-5-phenylpyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)oxolane-3,4-diolIC505000.0 [1]
(2R,3R,4S,5R)-2-[4-Amino-5-(furan-3-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC505000.0 [1]
(2R,3R,4S,5R)-2-(4-Amino-5-thiophen-3-ylpyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)oxolane-3,4-diolIC505000.0 [1]
(2R,3R,4S,5S)-2-(4-Anilino-5-phenylpyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)oxolane-3,4-diolIC500.47 [1]
7-(2-Morpholinopyridine-5-yl)-5-[[(1H-indole-3-yl)methyl]amino]pyrido[2,3-d]pyrimidine-4-amineIC5010.0 [1]
2-(4-Cyclohexylamino-5-phenyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC50250.0 [1], 1200.0 [2]
2-(6-Bromo-5-phenyl-4-phenylamino-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC501.0 [1]
2-Hydroxymethyl-5-(5-phenyl-4-phenylamino-pyrrolo[2,3-d]pyrimidin-7-yl)-tetrahydro-furan-3,4-diolIC500.8 [1]
2-(4-Amino-5-phenyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-methyl-tetrahydro-furan-3,4-diolIC50320.0 [1]
(2R,3R,4S,5S)-2-(4-Amino-5-iodopyrrolo[2,3-d]pyrimidin-7-yl)-5-methyloxolane-3,4-diolIC50400.0 [1]
6-{2-[4-(Dimethylamino)phenyl]ethynyl}-2-methyl-5-phenylpyrimidin-4-amineIC501000.0 [1]
(2R,3R,4S,5R)-2-[4-Amino-5-(4-methoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC502000.0 [1], 5000.0 [2]
(2R,3R,4S,5R)-2-[4-Amino-5-(4-methylsulfanylphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC5010000.0 [1]
(2R,3R,4S,5R)-2-(4-Amino-5-naphthalen-1-ylpyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)oxolane-3,4-diolIC5010000.0 [1]
(2R,3R,4S,5R)-2-(4-Amino-5-naphthalen-2-ylpyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)oxolane-3,4-diolIC505000.0 [1]
(2R,3R,4S,5R)-2-[4-Amino-5-(1-benzofuran-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC5010000.0 [1]
(2R,3R,4S,5R)-2-[4-Amino-5-(1H-pyrrol-3-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC504500.0 [1], 5000.0 [2]
(2R,3R,4S,5R)-2-[4-Amino-5-(1H-pyrazol-5-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC5010000.0 [1]
5-Ethynyl-7-(beta-D-Ribofuranosyl)-7h-Pyrrolo[2,3-D]pyrimidin-4-AmineIC50200.0 [1]
(2R,3R,4S,5R)-2-[4-Amino-5-(1H-imidazol-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC505000.0 [1], 20000.0 [2]
(2R,3R,4S,5R)-2-[4-Amino-5-(1H-pyrazol-4-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC5050.0 [1], 10000.0 [2]
(2R,3R,4S,5R)-2-[4-Amino-5-(1H-imidazol-5-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolIC5010000.0 [1], 13000.0 [2]
(2R,3R,4S,5S)-2-(4-Amino-5-iodopyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)oxolane-3,4-diolIC5068.0 [1]
(2R,3R,4S,5S)-2-(4-Anilino-5-phenylpyrrolo[2,3-d]pyrimidin-7-yl)-5-methyloxolane-3,4-diolIC500.8 [1]
7-(4-Dimethylamino-phenyl)-6-pentyl-pyrido[2,3-d]pyrimidin-4-ylamineIC5030.0 [1], 700.0 [2]
6-(4-Dimethylamino-phenyl)-7-pyridin-4-yl-pyrido[2,3-d]pyrimidin-4-ylamineIC50467.0 [1], 4170.0 [2]
6-[(3-Bromophenyl)methyl]-7-thiophen-2-ylpyrido[2,3-d]pyrimidin-4-amineIC503.8 [1], 650.0 [2]
6-(3-Bromo-phenyl)-7-(4-dimethylamino-phenyl)-pyrido[2,3-d]pyrimidin-4-ylamineIC5070.0 [1], 1000.0 [2]
6,7-Bis[4-(dimethylamino)phenyl]pyrido[2,3-d]pyrimidin-4-amineIC50183.0 [1], 367.0 [2]
6-Benzyl-7-(4-dimethylamino-phenyl)-pyrido[2,3-d]pyrimidin-4-ylamineIC50114.0 [1], 650.0 [2]
5-(3-Bromophenyl)-7-[6-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)pyridin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC501.4 [1], 28.3 [2]
6-(3-Bromo-4-methoxy-phenyl)-7-(4-dimethylamino-phenyl)-pyrido[2,3-d]pyrimidin-4-ylamineIC5033.0 [1], 225.0 [2]
6-(3-Bromo-4-methoxy-phenyl)-7-thiophen-2-yl-pyrido[2,3-d]pyrimidin-4-ylamineIC508.0 [1], 375.0 [2]
5-(3-Bromo-phenyl)-7-(6-pyrrolidin-1-yl-pyridin-3-yl)-pyrido[2,3-d]pyrimidin-4-ylamineIC503.4 [1], 45.0 [2]
5-(3-Bromophenyl)-7-[6-[(2R)-2-methoxypyrrolidin-1-yl]pyridin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC504.12 [1], 37.7 [2]
5-(3-Bromophenyl)-7-[6-[methyl(3-pyridinylmethyl)amino]-3-pyridinyl]pyrido[2,3-d]pyrimidine-4-amineIC504.1 [1], 42.3 [2]
5-(3-Bromophenyl)-7-(6-thiomorpholino-3-pyridinyl)pyrido[2,3-d]pyrimidine-4-amineIC501.3 [1], 42.5 [2]
5-(3-Bromophenyl)-7-[6-(4-hydroxypiperidino)-3-pyridinyl]pyrido[2,3-d]pyrimidine-4-amineIC501.8 [1], 33.0 [2]
5-(3-Bromophenyl)-7-[6-[4-(2-methoxyethoxy)piperidin-1-yl]pyridazin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC5015.1 [1], 81.9 [2]
5-(3-Bromophenyl)-7-[6-[4-[2-(oxan-4-yloxy)ethyl]piperidin-1-yl]pyridazin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC5022.8 [1], 89.5 [2]
[(2S)-1-[6-[4-Amino-5-(3-bromophenyl)pyrido[2,3-d]pyrimidin-7-yl]pyridazin-3-yl]pyrrolidin-2-yl]methanolIC5016.2 [1], 153.8 [2]
(3R,4S)-1-[5-[4-Amino-5-(3-bromophenyl)pyrido[2,3-d]pyrimidin-7-yl]pyridin-2-yl]-4-hydroxypyrrolidine-3-carbonitrileIC507.5 [1], 495.6 [2]
(3S,4R)-1-[5-[4-Amino-5-(3-bromophenyl)pyrido[2,3-d]pyrimidin-7-yl]pyridin-2-yl]pyrrolidine-3,4-diolIC506.5 [1], 130.1 [2]
1-[5-[4-Amino-5-(3-bromophenyl)pyrido[2,3-d]pyrimidin-7-yl]pyridin-2-yl]-4-[(Z)-C-methyl-N-(oxan-4-yloxy)carbonimidoyl]piperidin-4-olIC5031.7 [1], 43.7 [2]
5-(3-Bromophenyl)-7-[6-(2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)pyridin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC507.5 [1], 19.5 [2]
5-(3-Bromophenyl)-7-[6-(4-ethoxypiperidin-1-yl)pyridazin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC5010.4 [1], 51.7 [2]
5-(3-Bromophenyl)-7-[6-[4-(oxan-4-yloxymethyl)piperidin-1-yl]pyridazin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC502.8 [1], 17.3 [2]
5-(3-Bromophenyl)-7-[6-(1,3-dioxa-8-azaspiro[4.5]decan-8-yl)pyridin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC508.3 [1], 378.1 [2]
5-(3-Bromophenyl)-7-[6-(4-methoxyiminopiperidin-1-yl)pyridazin-3-yl]pyrido[2,3-d]pyrimidin-4-amineIC5018.8 [1], 74.4 [2]
Items per page: 1 - 10 of 100
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References

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MLA

"Quest Database™ Adenosine kinase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/adenosine-kinase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Adenosine kinase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/adenosine-kinase-inhibitors-ic50-ki.
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