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Adenosylhomocysteinase Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
Neplanocin AIC5010.0 [1]
Neplanocin AKi3.8 [1]
DHCeAIC50877.0 [1], 4125.0 [2], 8700.0 [3]
DHCeAKi41.0 [1], 49.0 [2]
(1S,2R,3S,4R)-4-(6-Aminopurin-9-yl)cyclopentane-1,2,3-triolIC501100.0 [1], 3100.0 [2]
(1S,2R,3S,4R)-4-(6-Aminopurin-9-yl)cyclopentane-1,2,3-triolKi160.0 [1]
(1R,2S,3R)-3-(6-Amino-9H-purin-9-yl)cyclopentane-1,2-diolIC501.5 [1], 55.0 [2], 18000.0 [3]
(1R,2S,3R)-3-(6-Amino-9H-purin-9-yl)cyclopentane-1,2-diolKi12.0 [1]
2-FluoronoraristeromycinIC5013000.0 [1], 63000.0 [2]
2-FluoronoraristeromycinKi7900.0 [1]
AristeromycinIC50303.0 [1], 4850.0 [2]
AristeromycinKi110.0 [1]
5'-DehydroadenosineKi39.0 [1], 43.0 [2]
(1s,2r,5s)-5-(6-Amino-9h-purin-9-yl)-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diolIC50240.0 [1], 470.0 [2], 480.0 [3]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[1,3-dihydroisoindol-2-yl(methyl)amino]-2-oxoethyl]anilino]-N-[2-(methylamino)ethyl]acetamide;hydrochlorideIC505.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[1,3-dihydroisoindol-2-yl(methyl)amino]-2-oxoethyl]anilino]-N-[2-(methylamino)ethyl]acetamide;hydrochlorideKi1.5 [1]
5-(6-Amino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carbaldehydeKi39.0 [1], 43.0 [2]
(1S,2R,5R)-5-(6-Aminopurin-9-yl)-3-(chloromethyl)cyclopent-3-ene-1,2-diolIC50195.0 [1], 939.0 [2]
2-[N-[2-[Benzyl(methyl)amino]-2-oxoethyl]-5-chloro-2-(4-chlorophenoxy)anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC50530.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[cyclohexyl(methyl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC50380.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[methyl(2-phenylethyl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC50340.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC50970.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[(2-fluorophenyl)methylamino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC508780.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-(2,3-dihydro-1H-inden-2-ylamino)-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC5011360.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-(1,3-dihydroisoindol-2-yl)-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC50100000.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC5017000.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-(N-methylanilino)-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC502700.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[2,3-dihydro-1H-inden-2-yl(methyl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC5052.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[methyl(1,2,3,4-tetrahydronaphthalen-2-yl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC5081.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[methyl-(4-phenylcyclohexyl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC50530.0 [1]
2-[N-[2-[(1-Acetylpiperidin-4-yl)-methylamino]-2-oxoethyl]-5-chloro-2-(4-chlorophenoxy)anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC504600.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[methyl-(1-methylsulfonylpiperidin-4-yl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC50230.0 [1]
Methyl 4-[[2-[5-chloro-2-(4-chlorophenoxy)-N-[2-oxo-2-(2-pyrrolidin-1-ylethylamino)ethyl]anilino]acetyl]-methylamino]piperidine-1-carboxylateIC50890.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[1,3-dihydroisoindol-2-yl(methyl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC5013.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[3,4-dihydro-1H-isoquinolin-2-yl(methyl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC50200.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[methyl-(4-methylsulfonylpiperazin-1-yl)amino]-2-oxoethyl]anilino]-N-(2-pyrrolidin-1-ylethyl)acetamideIC5049.0 [1]
Methyl 4-[[2-[5-chloro-2-(4-chlorophenoxy)-N-[2-oxo-2-(2-pyrrolidin-1-ylethylamino)ethyl]anilino]acetyl]-methylamino]piperazine-1-carboxylateIC5044.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[2,3-dihydro-1H-inden-2-yl(methyl)amino]-2-oxoethyl]anilino]-N-(3-pyrrolidin-1-ylpropyl)acetamideIC50330.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[2,3-dihydro-1H-inden-2-yl(methyl)amino]-2-oxoethyl]anilino]-N-(2-piperidin-1-ylethyl)acetamideIC50320.0 [1]
2-[5-Chloro-2-(4-chlorophenoxy)-N-[2-[2,3-dihydro-1H-inden-2-yl(methyl)amino]-2-oxoethyl]anilino]-N-[2-(dimethylamino)ethyl]acetamideIC50130.0 [1]
(1S,2R,3S,4R)-4-(4-Amino-7-fluoroimidazo[4,5-c]pyridin-1-yl)cyclopentane-1,2,3-triolIC509.4 [1], 24.0 [2]
2-Amino-4-[3-[(3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]imidazol-4-yl]-1H-pyrimidin-6-oneKi128000.0 [1], 217000.0 [2]
(1R,2S,3S)-3-(8-Aminoimidazo[1,2-a]pyrazin-3-yl)cyclopentane-1,2-diolIC501.5 [1], 250.0 [2]
(1R,2S,3R)-3-(4-Amino-7-chloroimidazo[4,5-c]pyridin-1-yl)cyclopentane-1,2-diolIC502.2 [1], 16.0 [2]
(1R,2S,3R)-3-(4-Amino-7-methylimidazo[4,5-c]pyridin-1-yl)cyclopentane-1,2-diolIC5036.0 [1], 236.0 [2]
(1R,2S,3R)-3-(6-Amino-2-fluoropurin-9-yl)cyclopentane-1,2-diolIC5098.0 [1], 2124.0 [2]
(1R,2S,3R)-3-(4-Amino-6,7-difluoroimidazo[4,5-c]pyridin-1-yl)cyclopentane-1,2-diolIC50189.0 [1], 3644.0 [2]
(1S,2S,3R,5S)-3-(4-Amino-7-fluoroimidazo[4,5-c]pyridin-1-yl)-5-fluorocyclopentane-1,2-diolIC5041.0 [1], 269.0 [2]
(1R,2S,3S)-3-(4-Amino-7-fluoro-1H-imidazo[4,5-c]pyridin-1-yl)-4-fluorocyclopentane-1,2-diolIC502.7 [1], 455.0 [2]
(1S,2R,5R)-5-(4-Amino-7-fluoroimidazo[4,5-c]pyridin-1-yl)cyclopent-3-ene-1,2-diolIC5028.0 [1], 9690.0 [2]
(1R,2S,3R)-3-(4-Amino-7-fluoro-1H-imidazo[4,5-c]pyridin-1-yl)cyclopentane-1,2-diolIC501.3 [1], 40.0 [2]
(1R,2S,3R)-3-(6-Amino-8-fluoropurin-9-yl)cyclopentane-1,2-diolIC5010000.0 [1]
(1R,2S,3R)-3-(6-Amino-8-chloropurin-9-yl)cyclopentane-1,2-diolIC502100.0 [1], 10000.0 [2]
(1R,2S,3R)-3-(6-Amino-8-bromopurin-9-yl)cyclopentane-1,2-diolIC5010000.0 [1]
(1S,2S,3R,5R)-3-(4-Amino-7-fluoroimidazo[4,5-c]pyridin-1-yl)-5-fluorocyclopentane-1,2-diolIC50672.0 [1], 10000.0 [2]
(1R,2R,3S,4R)-4-(4-Amino-7-fluoroimidazo[4,5-c]pyridin-1-yl)cyclopentane-1,2,3-triolIC50878.0 [1], 10000.0 [2]
(1R,2R,3S,4R,5S)-4-(4-Amino-7-fluoroimidazo[4,5-c]pyridin-1-yl)bicyclo[3.1.0]hexane-2,3-diolIC501960.0 [1], 10000.0 [2]
GuanosineKi1472000.0 [1]
InosineKi925000.0 [1]
3-DeazaadenosineIC504000.0 [1]
3-DeazaneplanocinIC50440.0 [1]
(S)-9-(2,3-Dihydroxypropyl)adenineIC50280.0 [1]
Adenosine dialdehydeKi3.3 [1]
AdenoxIC5040.0 [1]
3-DeazaaristeromycinKi4.0 [1]
IlimaquinoneIC5040000.0 [1]
5'-Amino-5'-deoxyadenosineIC5075020.0 [1]
5'-N-MethylcarboxamidoadenosineKi1930.0 [1]
(1S,2R,5R)-5-(6-Aminopurin-9-yl)-3-(2-hydroxyethyl)cyclopent-3-ene-1,2-diolIC50480.0 [1]
(Z)-4-(6-Aminopurin-9-yl)but-2-en-1-olKi125.0 [1]
Adenosine-5'-carboxylic acidKi410.0 [1]
(2S,3S,4R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolane-2-carboxamideKi2600.0 [1]
(1R,2S,3S,4R,5R)-3-(6-Aminopurin-9-yl)-4-fluoro-5-(hydroxymethyl)cyclopentane-1,2-diolIC508.0 [1]
Deazaneplanocin AIC50100000.0 [1]
9-(4-Hydroxy-3-(hydroxymethyl)-2-butenyl)adenineKi110.0 [1]
9-(4-Hydroxy-2-butyn)-adenineIC501000.0 [1]
9-(trans-4-Hydroxy-2-buten-1-yl)adenineKi330.0 [1]
5-MethylenearisteromycinIC5015700.0 [1]
(2S,3S,4R)-5-(6-Aminopurin-9-yl)-N-benzyl-3,4-dihydroxyoxolane-2-carboxamideKi43400.0 [1]
3-(7-Amino-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-5-hydroxymethyl-cyclopentane-1,2-diolKi22000.0 [1]
(1R,2R,3S,4R)-4-(6-Aminopurin-9-yl)cyclopentane-1,2,3-triolIC507600.0 [1]
(1S,2R,5R)-5-(4-Aminoimidazo[4,5-c]pyridin-1-yl)-3-(2-hydroxyethyl)cyclopent-3-ene-1,2-diolIC503760.0 [1]
(2S,3S,4R)-5-(6-Aminopurin-9-yl)-N-butyl-3,4-dihydroxyoxolane-2-carboxamideKi19800.0 [1]
5-(6-Amino-purin-9-yl)-3-methyl-cyclopent-3-ene-1,2-diolKi9150.0 [1]
5-(6-Amino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carbaldehyde oximeKi670.0 [1]
(1S,2R,5S)-5-(6-Amino-purin-9-yl)-4-fluoro-cyclopent-3-ene-1,2-diolIC508900.0 [1]
(2S,3S)-4-(6-Amino-purin-9-yl)-2,3-dihydroxy-butyraldehydeKi8800.0 [1]
(E)-4-(6-Aminopurin-9-yl)-2-methyl-but-2-en-1-olKi500.0 [1]
Methyl (2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolane-2-carboxylateKi1700.0 [1]
3-(6-Amino-purin-9-yl)-5-hydroxymethyl-cyclopentane-1,2,4-triolIC5028000.0 [1]
CID 16075366IC50180.0 [1]
5-(4-Amino-imidazo[4,5-c]pyridin-1-yl)-3-hydroxymethyl-cyclopent-3-ene-1,2-diolIC5031.0 [1]
(2R,3R,4S,5R)-2-(6-Aminopurin-9-yl)-5-(azidomethyl)oxolane-3,4-diolIC5028940.0 [1]
(3R,4S,5R)-2-(6-Aminopurin-9-yl)-5-ethynyloxolane-3,4-diolKi681.0 [1]
(2S,3S,4R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxy-N-phenyloxolane-2-carboxamideKi48500.0 [1]
(1R,2S,3R,5S)-3-(6-Aminopurin-9-yl)-5-azido-cyclopentane-1,2-diolIC50123000.0 [1]
(1S,2R,3S,5R)-3-Amino-5-(6-aminopurin-9-yl)cyclopentane-1,2-diolIC5076000.0 [1]
(2S,1R,3R,5R)-3-(6-Aminopurin-9-yl)-5-methylcyclopentane-1,2-diolKi5020.0 [1]
3-(6-Amino-purin-9-yl)-5-methyl-cyclopentane-1,2-diolKi27.0 [1]
3-(6-Amino-purin-9-yl)-5-ethyl-cyclopentane-1,2-diolKi586.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Adenosylhomocysteinase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/adenosylhomocysteinase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Adenosylhomocysteinase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/adenosylhomocysteinase-inhibitors-ic50-ki.
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