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Alpha-1d adrenergic receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
PrazosinIC500.88 [1]
TamsulosinIC501.4 [1]
Methyl 5-[3-(4,4-diphenylpiperidin-1-yl)propylcarbamoyl]-2,6-dimethyl-4-(4-nitrophenyl)-1,4-dihydropyridine-3-carboxylateKi1047.0 [1]
CyclazosinKi0.17 [1], 3.24 [2], 31.62 [3]
3-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-1,5-dihydropyrimido[5,4-b]indole-2,4-dioneKi0.36 [1], 2.75e+18 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseAlpha-1d adrenergic receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.11 Jan2026https://www.aatbio.com/data-sets/alpha-1d-adrenergic-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026January 11). Quest DatabaseAlpha-1d adrenergic receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/alpha-1d-adrenergic-receptor-inhibitors-ic50-ki.
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