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Alpha-2a adrenergic receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
YohimbineIC503.67 [1], 8.4 [2]
YohimbineKi3.1 [1], 7.5 [2]
TerazosinKi549.54 [1], 550.0 [2], 1500.0 [3], 3702.0 [4], 5187.0 [5]
ClozapineKi24.0 [1], 34.0 [2], 185.0 [3], 1000.0 [4]
PhentolamineKi1.7 [1], 2.25 [2], 2.6 [3], 55.9 [4]

References
This online resource may be cited as follows
MLA
"Quest DatabaseAlpha-2a adrenergic receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/alpha-2a-adrenergic-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseAlpha-2a adrenergic receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/alpha-2a-adrenergic-receptor-inhibitors-ic50-ki.
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