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Alpha-2b adrenergic receptor Inhibitors (IC50, Ki)

Structure
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Compound Name
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▼
Standard Type
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Standard Values (in nM)
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▼
YohimbineKi4.6 [1]
IdazoxanIC5019.5 [1]
IdazoxanKi22.91 [1], 100.0 [2]
TerazosinKi26.0 [1], 30.9 [2], 195.0 [3], 418.0 [4]
2-[1-(2-Prop-2-enylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi338.84 [1]
Methyl 5-[3-(4,4-diphenylpiperidin-1-yl)propylcarbamoyl]-2,6-dimethyl-4-(4-nitrophenyl)-1,4-dihydropyridine-3-carboxylateKi794.33 [1], 800.0 [2], 1088.0 [3], 1170.0 [4]
2-[1-(2-Biphenylyloxy)ethyl]-2-imidazolineKi501.19 [1]
ClonidineKi6.17 [1], 31.62 [2], 38.0 [3]
PrazosinKi13.0 [1], 133.0 [2], 365.0 [3]
PhentolamineKi7.6 [1], 8.23 [2], 48.0 [3]
3-[2-[1-(4,5-Dihydro-1H-imidazol-2-yl)ethoxy]phenyl]phenolKi354.81 [1]
2-[1-[2-(3-Nitrophenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazoleKi660.69 [1]
2-[(1S)-1-(2-Prop-2-enylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi398.11 [1]
2-[(1R)-1-(2-Prop-2-enylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi562.34 [1]
2-[1-[2-(Cyclopropylmethyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazoleKi407.38 [1]
ClozapineKi11.0 [1], 100.0 [2]
RisperidoneKi12.0 [1], 1000.0 [2]
OlanzapineKi100.0 [1], 192.0 [2]
QuetiapineKi45.8 [1], 1000.0 [2]
BrimonidineKi34.67 [1], 478.0 [2]
OxymetazolineKi581.0 [1], 5370.32 [2]
RilmenidineKi42.66 [1], 70.79 [2]
ClemastineKi142.0 [1], 478.63 [2]
CirazolineKi524.81 [1]
NiguldipineKi420.0 [1], 5000.0 [2]
Unii-22xbk6DY1EKi142.0 [1]
N,N-Diallyl-5-methoxytryptamineKi10000.0 [1]
1H-Imidazole, 4,5-dihydro-2-(1-phenoxyethyl)-Ki165.96 [1]
2-(1-Benzofuran-6-yl)-N-[[(1R)-5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl]methyl]-N-methylethanamineKi11.0 [1]
2-[(1S)-1-(2-Phenylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi588.84 [1]
4-(5-Fluoro-2-indanylmethyl)-2-imidazolineKi23.0 [1]
5-N-[3-(4,4-Diphenylpiperidin-1-yl)propyl]-3-N,2,6-trimethyl-4-(4-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxamideKi912.0 [1], 933.25 [2]
2-[(1R)-1-(2-Phenylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi1258.93 [1]
(3R,3As)-7,8-dimethoxy-3-[[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazoleKi14.0 [1], 42.0 [2]
(3R,3As)-7,8-dimethoxy-3-[[4-[(E)-2-methyl-3-phenylprop-2-enyl]piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazoleKi3.0 [1]
(3R,3As)-7,8-dimethoxy-3-[[4-[(E)-3-phenylbut-2-enyl]piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazoleKi14.0 [1]
5-N-[3-(4,4-Diphenylpiperidin-1-yl)propyl]-2,6-dimethyl-4-(4-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxamideKi275.0 [1], 416.87 [2]
1-Benzyl-4-chroman-2-ylmethyl-piperazineKi72.8 [1], 180.0 [2]
2-[1-[2-(3-Fluorophenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazoleKi269.15 [1]
3-[2-[1-(4,5-Dihydro-1H-imidazol-2-yl)ethoxy]phenyl]pyridineKi933.25 [1]
2-[1-(2-Thiophen-3-ylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi416.87 [1]
(R)-3-NitrobiphenylineKi741.31 [1]
2-[(1S)-1-[2-(3-Nitrophenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazoleKi1584.89 [1]
(3R,3As)-7,8-dimethoxy-3-[[4-(naphthalen-2-ylmethyl)piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazoleKi14.0 [1]
2-[1-(2-Cyclopropylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi309.03 [1]
2-[(1S)-1-(2-Cyclopropylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi263.03 [1]
2-[(1R)-1-(2-Cyclopropylphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi562.34 [1]
2-(1-(2-Bromophenoxy)ethyl)-4,5-dihydro-1H-imidazoleKi354.81 [1]
2-[1-(2-Cyclopropyloxyphenoxy)ethyl]-4,5-dihydro-1H-imidazoleKi1047.13 [1]
2-[(1R)-1-[2-(Cyclopropylmethyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazoleKi338.84 [1]
2-[(1S)-1-[2-(Cyclopropylmethyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazoleKi407.38 [1]
5-O-[3-(4,4-Diphenylpiperidin-1-yl)propyl] 3-O-methyl 2,6-dimethyl-4-(4-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylateKi570.0 [1], 758.0 [2]
N-[2-[4-[[(3S)-2,3-Dihydro-1,4-benzodioxin-3-yl]methyl]-1,4-diazepan-1-yl]ethyl]-2-phenoxypyridine-3-carboxamideKi14.3 [1], 31.3 [2]
1-((2,3-Dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-4-(2-methoxyphenyl)piperazineKi17.0 [1], 194.0 [2]
N-[2-[4-(2,3-Dihydro-1,4-benzodioxin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl]-2-phenoxypyridine-3-carboxamideKi49.0 [1], 132.0 [2]
2-(3-Cyanophenoxy)-N-[2-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl]pyridine-3-carboxamideKi27.5 [1], 36.0 [2]
2-(Tert-butylamino)-N-[2-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl]pyridine-3-carboxamideKi28.0 [1], 103.0 [2]
2-Butoxy-N-[2-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl]pyridine-3-carboxamideKi10.5 [1], 13.3 [2]
6-Butoxy-N-[2-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl]pyridine-2-carboxamideKi10.9 [1], 14.1 [2]
1-(2,3-Dihydro-1,4-benzodioxin-3-ylmethyl)-4-[2-[(2-phenoxypyridin-3-yl)methoxy]ethyl]-1,4-diazepaneKi69.5 [1], 132.0 [2]
5-[[4-(2,3-Dihydro-1,4-benzodioxin-3-ylmethyl)-1,4-diazepan-1-yl]methyl]-3-(2-phenoxypyridin-3-yl)-1,2,4-oxadiazoleKi5.2 [1], 15.3 [2]
EpinephrineKi397.0 [1]
TamoxifenKi1606.0 [1]
ChlorpromazineKi12.0 [1]
HaloperidolKi618.0 [1]
FluoxetineKi698.0 [1]
ChloroquineKi31622.78 [1]
TiclopidineKi139.0 [1]
AmiodaroneKi5886.0 [1]
CelecoxibKi692.0 [1]
AmitriptylineKi3.69 [1]
KetoconazoleKi8239.0 [1]
DiethylstilbestrolKi5340.0 [1]
BromocriptineKi16.0 [1]
DobutamineKi1354.0 [1]
MifepristoneKi12082.0 [1]
SertralineKi82.8 [1]
RauwolscineKi4.7 [1]
CorynanthineKi455.0 [1]
RaloxifeneKi1688.0 [1]
ClomipheneKi721.0 [1]
HydroxychloroquineKi72443.6 [1]
CarvedilolKi43.0 [1]
AripiprazoleKi1000.0 [1]
ClomipramineKi46.0 [1]
CandesartanKi1754.4 [1]
QuinacrineKi833.0 [1]
DisulfiramKi1469.0 [1]
PromethazineKi24.0 [1]
IsotretinoinKi3019.0 [1]
MianserinKi24.0 [1]
SelegilineKi172.0 [1]
DanazolKi10574.0 [1]
MiconazoleKi1642.0 [1]
MethysergideKi2175.0 [1]
ClotrimazoleKi3725.0 [1]
MirtazapineIC50223.87 [1]
DroperidolKi101.0 [1]
ThioridazineKi174.0 [1]
FluphenazineKi13.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Alpha-2b adrenergic receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/alpha-2b-adrenergic-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Alpha-2b adrenergic receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/alpha-2b-adrenergic-receptor-inhibitors-ic50-ki.
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