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Alpha-2c adrenergic receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
YohimbineIC5027.1 [1]
YohimbineKi2.3 [1]
ClonidineKi9.33 [1], 30.0 [2], 56.23 [3], 160.0 [4]
TerazosinKi78.0 [1], 170.0 [2], 213.0 [3], 223.87 [4], 878.0 [5]
(3R,3As)-7,8-dimethoxy-3-[[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazoleKi0.5 [1], 4.8 [2], 6.2 [3], 8.8 [4]

References
This online resource may be cited as follows
MLA
"Quest DatabaseAlpha-2c adrenergic receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.16 Jun2026https://www.aatbio.com/data-sets/alpha-2c-adrenergic-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026June 16). Quest DatabaseAlpha-2c adrenergic receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/alpha-2c-adrenergic-receptor-inhibitors-ic50-ki.
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