Alpha-ketoglutarate-dependent dioxygenase alkB homolog 3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	1-(1,3-Benzothiazol-2-yl)-3,4-dimethyl-1H-pyrazol-5-ol	IC50	10000.0 [1]
	4-Benzyl-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	670.0 [1]
	DMT1 blocker 1	IC50	1700.0 [1]
	2,3-Bis(4-methylphenyl)-5-methyl-1H-indene-1-one	IC50	50000.0 [1]
	2-Bromo-3-(4-methoxyphenyl)-5-methylinden-1-one	IC50	43170.0 [1]
	2-(3,5-Dimethoxyphenyl)-3-(4-methoxyphenyl)-5-(4-methylphenyl)inden-1-one	IC50	50000.0 [1]
	2-Chloro-3-(4-methoxyphenyl)-5-phenylinden-1-one	IC50	50000.0 [1]
	2-Bromo-3-(3,5-dimethoxyphenyl)-5-methylinden-1-one	IC50	50000.0 [1]
	2,3-Bis(3,4-dichlorophenyl)-5-methylinden-1-one	IC50	32300.0 [1]
	2,3-Bis(3,4-dimethoxyphenyl)-5-phenylinden-1-one	IC50	50000.0 [1]
	2-Chloro-3-(4-methoxyphenyl)-5-(4-methylphenyl)inden-1-one	IC50	9800.0 [1]
	2,3-Bis(3-methoxyphenyl)-5-phenylinden-1-one	IC50	50000.0 [1]
	2,3-Bis(3-methoxyphenyl)-5-(4-methylphenyl)inden-1-one	IC50	13100.0 [1]
	2-(3,5-Dimethoxyphenyl)-3-(4-methoxyphenyl)-5-phenylinden-1-one	IC50	50000.0 [1]
	2-Bromo-5-methyl-3-naphthalen-1-ylinden-1-one	IC50	50000.0 [1]
	2,3-Bis(4-methoxyphenyl)-5-phenylinden-1-one	IC50	50000.0 [1]
	2,3-Bis(4-methoxyphenyl)-5-methylinden-1-one	IC50	50000.0 [1]
	2,3-Bis(3-methoxyphenyl)-5-methylinden-1-one	IC50	50000.0 [1]
	3-(3,5-Dimethoxyphenyl)-2-(4-methoxyphenyl)-5-methylinden-1-one	IC50	50000.0 [1]
	2,3-Bis(3,4-dimethoxyphenyl)-5-(4-methylphenyl)inden-1-one	IC50	50000.0 [1]
	2-Chloro-3-(4-methoxyphenyl)-5-methylinden-1-one	IC50	50000.0 [1]
	2-Bromo-5-methyl-3-(4-methylphenyl)inden-1-one	IC50	50000.0 [1]
	2,3-Bis(3,4-dimethoxyphenyl)-5-methylinden-1-one	IC50	50000.0 [1]
	2-(3,5-Dimethoxyphenyl)-3-(4-methoxyphenyl)-5-methylinden-1-one	IC50	50000.0 [1]
	2-Bromo-3-(3,4-dimethoxyphenyl)-5-methylinden-1-one	IC50	50000.0 [1]
	1-(1H-Benzimidazol-2-yl)-4-(4-tert-butylbenzyl)-3-methyl-1H-pyrazol-5-ol	IC50	4100.0 [1]
	1-(1H-Benzimidazol-2-yl)-3,4-dimethyl-1H-pyrazol-5-ol	IC50	4000.0 [1]
	1-(1H-Benzimidazol-2-yl)-4-(2-chlorobenzyl)-3-methyl-1H-pyrazol-5-ol	IC50	10000.0 [1]
	1-(1H-Benzimidazol-2-yl)-4-(4-chlorobenzyl)-3-methyl-1H-pyrazol-5-ol	IC50	10000.0 [1]
	1-(1H-Benzimidazol-2-yl)-4-(3-chlorobenzyl)-3-methyl-1H-pyrazol-5-ol	IC50	540.0 [1]
	2-(1,3-Benzoxazol-2-yl)-4,5-dimethyl-1H-pyrazol-3-one	IC50	10000.0 [1]
	1-(1H-Benzimidazol-2-yl)-4-benzyl-3-methyl-1H-pyrazol-5-ol	IC50	480.0 [1]
	4,5-Dimethyl-2-pyridin-2-yl-1H-pyrazol-3-one	IC50	10000.0 [1]
	2,3,5-Triphenyl-1H-indene-1-one	IC50	50000.0 [1]
	3,4-Dimethyl-1-phenyl-3-pyrazolin-5-one	IC50	10000.0 [1]
	4,5-Dimethyl-2-pyrimidin-2-yl-1H-pyrazol-3-one	IC50	10000.0 [1]
	1-(1H-Benzimidazol-2-yl)-3-phenyl-1H-pyrazol-5-ol	IC50	7200.0 [1]
	2-Bromo-5-methyl-3-phenylinden-1-one	IC50	50000.0 [1]
	5-Methyl-2,3-diphenyl-1H-inden-1-one	IC50	50000.0 [1]
	1-(1H-Benzimidazol-2-yl)-3-methyl-1H-pyrazol-5-ol	IC50	3600.0 [1]
	2-[2-(1H-Benzimidazol-2-yl)-5-methyl-3-oxo-1H-pyrazol-4-yl]acetic acid	IC50	15000.0 [1]
	2-(6-Chloro-1H-benzimidazol-2-yl)-4,5-diphenyl-1H-pyrazol-3-one	IC50	2000.0 [1]
	4-Benzyl-2-(6-tert-butyl-1H-benzimidazol-2-yl)-5-methyl-1H-pyrazol-3-one	IC50	640.0 [1]
	4-[(3,4-Dichlorophenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	720.0 [1]
	2-(1H-Benzimidazol-2-yl)-4-[(3,4-dichlorophenyl)methyl]-5-methyl-1H-pyrazol-3-one	IC50	3100.0 [1]
	4,5-Dimethyl-2-(4-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	10000.0 [1]
	2-(1H-Benzimidazol-2-yl)-4-[(2,4-dichlorophenyl)methyl]-5-methyl-1H-pyrazol-3-one	IC50	10000.0 [1]
	2-(1H-Benzimidazol-2-yl)-4-[(4-methoxyphenyl)methyl]-5-methyl-1H-pyrazol-3-one	IC50	630.0 [1]
	4-Benzyl-5-methyl-2-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]-1H-pyrazol-3-one	IC50	610.0 [1]
	2-(6-Methyl-1H-benzimidazol-2-yl)-4,5-diphenyl-1H-pyrazol-3-one	IC50	5800.0 [1]
	4-[(4-Fluorophenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	780.0 [1]
	5-Methyl-2-(6-methyl-1H-benzimidazol-2-yl)-4-[(4-phenylphenyl)methyl]-1H-pyrazol-3-one	IC50	5300.0 [1]
	4,5-Dimethyl-2-(1-methylbenzimidazol-2-yl)-1H-pyrazol-3-one	IC50	10000.0 [1]
	4-Benzyl-5-methyl-2-(6-phenyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	810.0 [1]
	4-Benzyl-5-methyl-2-(4-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	5900.0 [1]
	4-[(4-Chlorophenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	750.0 [1]
	4-[(4-Tert-butylphenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	3700.0 [1]
	4-Benzyl-5-methyl-2-[6-(4-methylphenyl)-1H-benzimidazol-2-yl]-1H-pyrazol-3-one	IC50	2100.0 [1]
	4,5-Dimethyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	2600.0 [1]
	Methyl 2-[2-(1H-benzimidazol-2-yl)-5-methyl-3-oxo-1H-pyrazol-4-yl]acetate	IC50	4300.0 [1]
	2-(1H-Benzimidazol-2-yl)-4-benzyl-5-phenyl-1H-pyrazol-3-one	IC50	10000.0 [1]
	2-(1H-Benzimidazol-2-yl)-4-[(4-fluorophenyl)methyl]-5-methyl-1H-pyrazol-3-one	IC50	600.0 [1]
	2-(1H-Benzimidazol-2-yl)-5-methyl-4-[(4-phenylphenyl)methyl]-1H-pyrazol-3-one	IC50	720.0 [1]
	4-Benzyl-2-(6-chloro-1H-benzimidazol-2-yl)-5-methyl-1H-pyrazol-3-one	IC50	4500.0 [1]
	4-Benzyl-2-[6-(4-chlorophenyl)-1H-benzimidazol-2-yl]-5-methyl-1H-pyrazol-3-one	IC50	1500.0 [1]
	2-(1H-Benzimidazol-2-yl)-5-methyl-4-(naphthalen-2-ylmethyl)-1H-pyrazol-3-one	IC50	750.0 [1]
	2-(1H-Benzimidazol-2-yl)-4-methyl-5-phenyl-1H-pyrazol-3-one	IC50	10000.0 [1]
	4-Methyl-2-(6-methyl-1H-benzimidazol-2-yl)-5-phenyl-1H-pyrazol-3-one	IC50	3300.0 [1]
	2-(1H-Benzimidazol-2-yl)-5-methyl-4-[[4-(trifluoromethyl)phenyl]methyl]-1H-pyrazol-3-one	IC50	550.0 [1]
	4-Benzyl-2-(6-bromo-1H-benzimidazol-2-yl)-5-methyl-1H-pyrazol-3-one	IC50	490.0 [1]
	4-Benzyl-2-(4,5-dimethyl-1H-benzimidazol-2-yl)-5-methyl-1H-pyrazol-3-one	IC50	10000.0 [1]
	5-Methyl-2-(6-methyl-1H-benzimidazol-2-yl)-4-[[4-(trifluoromethyl)phenyl]methyl]-1H-pyrazol-3-one	IC50	570.0 [1]
	4-[(4-Methoxyphenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	680.0 [1]
	4-[(2-Chlorophenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one	IC50	910.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 74 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Alpha-ketoglutarate-dependent dioxygenase alkB homolog 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/alpha-ketoglutarate-dependent-dioxygenase-alkb-homolog-3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Alpha-ketoglutarate-dependent dioxygenase alkB homolog 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/alpha-ketoglutarate-dependent-dioxygenase-alkb-homolog-3-inhibitors-ic50-ki.
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