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Aminopeptidase N Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
UbenimexIC5020120.0 [1]
Angiotensin IVKi56.23 [1], 830.0 [2], 841.0 [3], 1202264434617410.0 [4]
OpiorphinIC508000.0 [1], 8100.0 [2]
CID 44593458IC50141900.0 [1]
7-Amino-5,7,8,9-tetrahydro-benzocyclohepten-6-one hydrochlorideKi1000.0 [1], 2000.0 [2]
N-Hydroxy-2-(naphthalen-2-ylsulfanyl)-acetamideIC503400.0 [1]
N-Hydroxy-2-(naphthalen-2-ylsulfanyl)-acetamideKi3500.0 [1]
[1-Amino-2-(cyclohexylamino)ethyl]phosphonic acidKi691.0 [1], 870.0 [2]
(2S)-2-Amino-4-methylsulfinylbutane-1-thiol;2,2,2-trifluoroacetic acidKi11.0 [1]
5-Amino-2-benzyl-7-methyl-4-oxo-octanoic acidKi79000.0 [1], 260000.0 [2]
(2S)-2-Amino-4-methylsulfanylbutane-1-thiol;2,2,2-trifluoroacetic acidKi11.0 [1]
trans-1-Benzenesulfonyl-4-hydroxy-pyrrolidine-2-carboxylic acid methyl esterIC5053800.0 [1]
2-Amino-4-methylsulfanylbutane-1-thiolIC5011.0 [1]
2-Amino-4-methylsulfanylbutane-1-thiolKi8.0 [1]
3-Amino-3,4-dihydro-1H-naphthalen-2-one;hydrochlorideKi500.0 [1]
trans-4-Hydroxy-1-methanesulfonyl-pyrrolidine-2-carboxylic acid methyl esterIC5041600.0 [1]
CID 53494934Ki0.06 [1], 0.35 [2]
(2S,4R)-Methyl 4-hydroxy-1-tosylpyrrolidine-2-carboxylateIC5038400.0 [1]
(2S)-5-(Diaminomethylideneamino)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]pentanoyl]amino]-3-phenylpropanoyl]amino]-3-hydroxybutanoyl]amino]pentanoic acidIC50100000.0 [1]
(5S)-5-Amino-2,7-dimethyl-4-oxooctanoic acidKi660000.0 [1], 940000.0 [2]
(2S)-N-Hydroxy-4-methyl-2-[[1-[(2-phenylmethoxyphenyl)methyl]triazol-4-yl]methylcarbamoylamino]pentanamideIC50740.0 [1], 1300.0 [2]
(2S)-N-Hydroxy-4-methyl-2-[[1-[(3-phenylmethoxyphenyl)methyl]triazol-4-yl]methylcarbamoylamino]pentanamideIC50870.0 [1], 4900.0 [2]
2-[[(2S)-2-[[(2S,3R)-3-Amino-2-hydroxy-4-phenylbutanoyl]amino]-4-methylpentanoyl]amino]acetic acid;hydrochlorideIC505370.0 [1], 13570.0 [2]
(5-Fluoro-2,4-dioxopyrimidin-1-yl)methyl 2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanoyl]amino]-4-methylpentanoyl]amino]acetate;hydrochlorideIC501680.0 [1], 5690.0 [2]
(2S)-N-Hydroxy-2-[[1-[(2-methoxyphenyl)methyl]triazol-4-yl]methylcarbamoylamino]-4-methylpentanamideIC506500.0 [1], 15300.0 [2]
(2S)-N-Hydroxy-2-[[1-[1-(2-methoxyphenyl)ethyl]triazol-4-yl]methylcarbamoylamino]-4-methylpentanamideIC504800.0 [1], 12300.0 [2]
(2S)-2-[[1-[(2-Ethoxyphenyl)methyl]triazol-4-yl]methylcarbamoylamino]-N-hydroxy-4-methylpentanamideIC502100.0 [1], 5000.0 [2]
(2S)-N-Hydroxy-4-methyl-2-[[1-[(2-methylphenyl)methyl]triazol-4-yl]methylcarbamoylamino]pentanamideIC506900.0 [1], 20600.0 [2]
(5-Fluoro-2,4-dioxopyrimidin-1-yl)methyl (2S)-2-[[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanoyl]amino]-4-methylpentanoateIC5065290.0 [1], 164170.0 [2]
CurcuminIC5015500.0 [1]
PuromycinIC5041000.0 [1]
SitagliptinIC50100000.0 [1]
(1E,4Z,6E)-5-Hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneIC5010000.0 [1]
AmastatinKi200.0 [1]
(2-Mercaptomethyl-3-phenyl-propionyl)-glycineKi10000.0 [1]
ActinoninKi170.0 [1]
KelatorphanKi7000.0 [1]
Butylboronic acidKi10000.0 [1]
TosedostatIC50680.0 [1]
ProbestinKi19.0 [1]
Leucine Phosphonic AcidKi2.62 [1]
(1-Amino-2-phenylethyl)phosphonic acidKi27500.0 [1]
Glutamate thiolKi17000.0 [1]
PhenylalanylleucineIC501000000.0 [1]
4-Amino-N-(2,6-dimethylphenyl)phthalimideIC5056300.0 [1]
2-(2,6-Diethylphenyl)-4H-isoquinoline-1,3-dioneKi120.0 [1]
Phosphonic acid, (1-amino-3-phenylpropyl)-Ki0.79 [1]
2-[[(1-Amino-3-phenylpropyl)-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi2.0 [1]
2-(5'-Bromo-2'-oxospiro[1,3-dioxolane-2,3'-indole]-1'-yl)-N-hydroxyacetamideIC5012400.0 [1]
Inhibitor 19 [PMID: 21476495]Ki240.0 [1]
2-[2,6-Di(propan-2-yl)phenyl]-3-sulfanylideneisoindol-1-oneIC50309200.0 [1]
2-[[(1-Amino-3-phenylpropyl)-hydroxyphosphoryl]methyl]-3-(4-hydroxyphenyl)propanoic acidKi7.2 [1]
CID 118720630Ki2.4 [1]
CID 127052870Ki65.0 [1]
2-Amino-3-phenyl-1-propanethiolIC5030.0 [1]
[(1S)-1-Amino-3-methylbutyl]phosphonic acidKi167.0 [1]
(S)-4-Amino-5-mercaptovaleric acidKi120.0 [1]
2-[(1-Cyanophenanthren-3-yl)methyl]phenanthrene-1-carbonitrileKi2010.0 [1]
2-(2,6-Dimethyl-phenyl)-4-hydroxy-isoindole-1,3-dioneIC50264500.0 [1]
(S)-N-(1-(2-(Hydroxyamino)-2-oxoethyl)-2,6-dioxopiperidin-3-yl)-3,4,5-trimethoxybenzamideIC503100.0 [1]
(2R)-2-[4-[[[(2S)-3-[(3R)-3-Amino-4-(2,4,5-trifluorophenyl)butanoyl]-1,3-thiazolidine-2-carbonyl]amino]methyl]anilino]-3-methylbutanoic acidIC50100000.0 [1]
Cyclohexanecarboxylic acid, 4-(2-amino-3-mercaptopropyl)-Ki2300.0 [1]
3-(2-Amino-3-mercaptopropyl)cyclohexanecarboxylic acidKi210.0 [1]
4-(2-Amino-3-mercaptopropyl)benzoic acidKi7300.0 [1]
[4-(2-Amino-3-mercapto-propyl)-phenyl]-acetic acidKi2700.0 [1]
3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-butyramideKi20000.0 [1]
(2S)-2-Amino-N-[(3S)-1-[2-(hydroxyamino)-2-oxoethyl]-2,6-dioxopiperidin-3-yl]-3-phenylpropanamide;hydrochlorideIC501800.0 [1]
4-Amino-2-(2,6-dimethyl-phenyl)-isoindole-1,3-dioneIC50108900.0 [1]
(1-Amino-3-phenylpropyl)-hydroxy-oxophosphaniumKi0.16 [1]
N-{(2s)-3-[(1r)-1-Aminoethyl](Hydroxy)phosphoryl-2-Benzylpropanoyl}-L-PhenylalanineKi2.2 [1]
2-[[[1-Amino-3-(3,5-dimethylphenyl)propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi4.8 [1]
2-[[[1-Amino-3-(3-hydroxyphenyl)propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi146.0 [1]
2-[[[1-Amino-3-(4-hydroxyphenyl)propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi24.2 [1]
2-[[[1-Amino-3-[4-(hydroxymethyl)phenyl]propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi1.7 [1]
2-[[(1-Amino-3-pyridin-3-ylpropyl)-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi2.1 [1]
2-[[(1-Amino-3-pyridin-4-ylpropyl)-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi1.3 [1]
2-[[(1-Amino-3-phenylpropyl)-hydroxyphosphoryl]methyl]-3-(3,5-dimethylphenyl)propanoic acidKi27.8 [1]
2-[[3-(Aminomethyl)phenyl]methyl]-3-[(1-amino-3-phenylpropyl)-hydroxyphosphoryl]propanoic acidKi2.1 [1]
2-[[4-(Aminomethyl)phenyl]methyl]-3-[(1-amino-3-phenylpropyl)-hydroxyphosphoryl]propanoic acidKi0.69 [1]
(1-Amino-2-methylpropyl)-(1-hydroxy-3-phenylpropyl)phosphinic acidIC50500.0 [1]
(1-Amino-2-morpholin-4-ylethyl)phosphonic acidKi37700.0 [1]
2-[[[1-Amino-2-(2-methylpropylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi499.0 [1]
2-[[[1-Amino-2-(cyclohexylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi275.0 [1]
[1-Amino-2-(oxolan-2-ylmethylamino)ethyl]phosphonic acidKi782.0 [1]
(1-Amino-2-piperidin-1-ylethyl)phosphonic acidKi6040.0 [1]
[1-Amino-2-[(2-aminocyclohexyl)amino]ethyl]phosphonic acidKi13500.0 [1]
[1-Amino-2-(1-phenylethylamino)ethyl]phosphonic acidKi391.0 [1]
[1-Amino-2-[2-(dimethylamino)ethylamino]ethyl]phosphonic acidKi5740.0 [1]
2-Benzyl-3-[1,2-diaminoethyl(hydroxy)phosphoryl]propanoic acidKi4450.0 [1]
[1-Amino-2-(cycloheptylamino)ethyl]phosphonic acidKi397.0 [1]
[1-Amino-2-(2-phenylethylamino)ethyl]phosphonic acidKi1220.0 [1]
2-[[[1-Amino-2-(propylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi1110.0 [1]
[1-Amino-2-(2-piperazin-1-ylethylamino)ethyl]phosphonic acidKi3220.0 [1]
[1-Amino-2-[(4-tert-butylphenyl)methylamino]ethyl]phosphonic acidKi2550.0 [1]
[1-Amino-2-[(4-aminophenyl)methylamino]ethyl]phosphonic acidKi1490.0 [1]
2-[[[1-Amino-2-(cycloheptylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi207.0 [1]
[1-Amino-2-[(4-methoxyphenyl)methylamino]ethyl]phosphonic acidKi357.0 [1]
2-[[[1-Amino-2-[2-(4-methoxyphenyl)ethylamino]ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi78.0 [1]
[1-Amino-2-(hexylamino)ethyl]phosphonic acidKi297.0 [1]
[1-Amino-2-[[4-(aminomethyl)phenyl]methylamino]ethyl]phosphonic acidKi2890.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Aminopeptidase N Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/aminopeptidase-n-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Aminopeptidase N Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/aminopeptidase-n-inhibitors-ic50-ki.
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