 | 1-Bromo-4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid | Ki | 2.0 [1] |
 | 4-[2-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid | Ki | 15.0 [1] |
 | Coformycin | Ki | 3000.0 [1] |
 | 3-[2-(8-Hydroxy-7,8-dihydro-6H-imidazo[4,5-d][1,3]diazepin-3-yl)-ethyl]-benzoic acid | Ki | 500.0 [1] |
 | 2-Benzyl-6-(8-hydroxy-7,8-dihydro-6H-imidazo[4,5-d][1,3]diazepin-3-yl)-hexanoic acid | Ki | 410.0 [1] |
 | 2-[4-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]-2-[[2-(trifluoromethyl)phenyl]methyl]propanedioic acid | Ki | 41.0 [1] |
 | 6-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)-2-phenylmethoxycarbonylhexanoic acid | Ki | 360.0 [1] |
 | 4-[2-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]naphthalene-2-carboxylic acid | Ki | 20.0 [1] |
 | 2-[4-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]-2-[[3-(trifluoromethyl)phenyl]methyl]propanedioic acid | Ki | 29.0 [1] |
 | 2-[4-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]-2-[[4-(trifluoromethyl)phenyl]methyl]propanedioic acid | Ki | 40.0 [1] |
 | 2-Carbamoyl-6-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)-2-methylhexanoic acid | Ki | 7800.0 [1] |
 | Ethyl 4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 1300.0 [1] |
 | Ethyl 4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-1-methoxy-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 2300.0 [1] |
 | Ethyl 4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-1-propan-2-yloxy-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 3800.0 [1] |
 | 2-Benzyl-2-[4-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]propanedioic acid | Ki | 170.0 [1] |
 | Ethyl 1-bromo-4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 1000.0 [1] |
 | 4-[2-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-1-phenylmethoxy-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid | Ki | 9.0 [1] |
 | 1,3-Dichloro-4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid | Ki | 50.0 [1] |
 | 6-Bromo-4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]naphthalene-2-carboxylic acid | Ki | 960.0 [1] |
 | Ethyl 4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-1-phenylmethoxy-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 300.0 [1] |
 | 2-(Cyclohexylcarbamoyl)-6-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)-2-methylhexanoic acid | Ki | 5200.0 [1] |
 | 6-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)-2-methyl-2-(2-phenylethylcarbamoyl)hexanoic acid | Ki | 2100.0 [1] |
 | Ethyl 4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-8-(trifluoromethyl)naphthalene-2-carboxylate | Ki | 35000.0 [1] |
 | Diethyl 2-benzyl-2-[4-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]propanedioate | Ki | 2600.0 [1] |
 | Dibenzyl 2-[4-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]-2-[[2-(trifluoromethyl)phenyl]methyl]propanedioate | Ki | 250.0 [1] |
 | 2-(Benzylcarbamoyl)-6-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)hexanoic acid | Ki | 2400.0 [1] |
 | 6-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)-2-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]hexanoic acid | Ki | 1200.0 [1] |
 | Ethyl 6-bromo-4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]naphthalene-2-carboxylate | Ki | 14000.0 [1] |
 | Diethyl 2-[4-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]-2-methylpropanedioate | Ki | 44800.0 [1] |
 | Methyl 4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]naphthalene-2-carboxylate | Ki | 1800.0 [1] |
 | 4-[2-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-3-methoxy-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid | Ki | 40.0 [1] |
 | Ethyl 1,3-dichloro-4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 500.0 [1] |
 | 4-[2-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-1-propan-2-yloxy-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid | Ki | 90.0 [1] |
 | 4-[2-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-1-methoxy-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid | Ki | 30.0 [1] |
 | Diethyl 2-[4-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]-2-[[2-(trifluoromethyl)phenyl]methyl]propanedioate | Ki | 360.0 [1] |
 | Ethyl 4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-3-methoxy-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 2400.0 [1] |
 | Benzyl 4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 5000.0 [1] |
 | 6-(8-Hydroxy-7,8-dihydro-6H-imidazo[4,5-d][1,3]diazepin-3-yl)-hexanoic acid | Ki | 4200.0 [1] |
 | 2-[4-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]propanedioic acid | Ki | 5100.0 [1] |
 | 2-[4-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]-2-methylpropanedioic acid | Ki | 6000.0 [1] |
 | 6-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)-2-methyl-2-phenylmethoxycarbonylhexanoic acid | Ki | 900.0 [1] |
 | 4-[2-(8-Hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-8-(trifluoromethyl)naphthalene-2-carboxylic acid | Ki | 220.0 [1] |
 | Benzyl 1,3-dichloro-4-[2-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxylate | Ki | 300.0 [1] |
 | 2-[(4-Chlorophenyl)methylcarbamoyl]-6-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)hexanoic acid | Ki | 1300.0 [1] |
 | Dibenzyl 2-[4-(8-hydroxy-7,8-dihydro-4H-imidazo[4,5-d][1,3]diazepin-3-yl)butyl]-2-methylpropanedioate | Ki | 5200.0 [1] |
 | 3-(2-Imidazo[2,1-f][1,2,4]triazin-7-ylethyl)benzoic acid | IC50 | 370000.0 [1] |
 | 4-(2-Imidazo[2,1-f][1,2,4]triazin-7-ylethyl)-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid | IC50 | 900.0 [1] |
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