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Androgen Receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
BicalutamideIC50330.0 [1]
BicalutamideKi19.0 [1], 35.0 [2], 64.0 [3]
AndrostanoloneIC502.1 [1], 13.1 [2], 10000.0 [3]
HydroxyflutamideIC5043.0 [1]
HydroxyflutamideKi2.0 [1], 43.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseAndrogen Receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.27 Dec2025https://www.aatbio.com/data-sets/androgen-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 27). Quest DatabaseAndrogen Receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/androgen-receptor-inhibitors-ic50-ki.
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