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Angiotensin II receptor Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
LosartanIC508.0 [1], 18.0 [2], 50.0 [3], 89.0 [4]
2-Ethyl-5,7-dimethyl-3-((4-(2-(2H-tetrazol-5-yl)phenyl)phenyl)methyl)imidazo(4,5-b)pyridineIC500.1 [1], 0.3 [2], 6.0 [3]
Losartan carboxylic acidIC500.3 [1], 1.8 [2]
4'-((2-Butyl-4-chloro-5-(hydroxymethyl)-1H-imidazol-1-yl)methyl)-(1,1'-biphenyl)-2-carboxylic acidIC50230.0 [1], 480.0 [2]
2-[4-(2-Butylbenzimidazol-1-yl)methylphenyl]benzoic acidIC502300.0 [1]
2-Butyl-1-({4-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]phenyl}methyl)-1H-1,3-benzodiazoleIC5096.0 [1]
2-Butyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5H-imidazo[4,5-c]pyridin-4-oneIC500.8 [1], 16.0 [2]
Losartan potassiumIC503.0 [1]
IrbesartanIC503.0 [1]
SaralasinIC500.07 [1]
(Sar1,Ile8)-Angiotensin IIIC500.21 [1]
2-Ethyl-4-((2'-(1H-1,2,3,4-tetrazol-5-yl)biphenyl-4-yl)methoxy)quinoline hydrochlorideIC5031.0 [1]
NaluzotanKi2000.0 [1]
Angiotensin II, 1-sar-5-ile-8-ala-IC505.8 [1]
7-Methyl-2-propyl-3-((2'-(1H-tetrazol-5-yl)(1,1'-biphenyl)-4-yl)methyl)-3H-imidazo(4,5-b)pyridineIC501.0 [1]
2-Propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5-[2-(2,2,2-trifluoroacetyl)pyrrol-1-yl]imidazole-4-carboxylic acidIC503.8 [1]
2-[2-Butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]-N,N-dimethylacetamideIC500.2 [1]
5,7-Dimethyl-2-propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-b]pyridineIC500.3 [1]
Angiotensin II, sar(1)-val(5)-ile(8)-IC500.45 [1]
2-Butyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5-(thiophen-2-ylmethyl)imidazo[4,5-c]pyridin-4-oneIC502.0 [1]
3-Butyl-2-[2'-(1H-tetrazole-5-yl)-4-biphenylylmethyl]-2,3-diazaspiro[4.4]nonane-1,4-dioneIC5022.0 [1]
2-Ethyl-4-(2'-(1H-tetrazol-5-yl)biphenyl-4-ylmethoxy)-5,6,7,8-tetrahydroquinolineIC505.0 [1]
2-[2-Butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]-N,N-diphenylacetamideIC507.0 [1]
2BotbmipIC500.08 [1]
2-Butyl-5-methylsulfanyl-3-[[4-[2-(propylcarbamoylsulfamoyl)phenyl]phenyl]methyl]imidazole-4-carboxylic acidIC50920.0 [1]
Methyl 4-[[2-butyl-5-[(Z)-[1-butyl-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoateIC50350.0 [1]
2-Cyclopropyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5H-imidazo[4,5-c]pyridin-4-oneIC502.0 [1]
4-[[2-Butyl-5-[(Z)-[2,5-dioxo-3-(thiophen-2-ylmethyl)imidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC5018.0 [1]
2-[2-Butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]acetic acidIC500.7 [1]
4-[[2-Butyl-5-[(Z)-[3-[(4-chlorophenyl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC5028.0 [1]
N,N-Dimethyl-2-[4-oxo-2-propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]acetamideIC500.1 [1]
4-[[5-[(E)-(3-Benzyl-2,5-dioxoimidazolidin-4-ylidene)methyl]-2-butylimidazol-1-yl]methyl]benzoic acidIC50100.0 [1]
2-[2-Butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]acetamideIC500.4 [1]
4-[[2-Butyl-5-[(Z)-[1-butyl-3-[(5-methylthiophen-3-yl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC509.2 [1]
4-[[5-[(Z)-[3-[(2-Amino-1,3-thiazol-4-yl)methyl]-1-butyl-2,5-dioxoimidazolidin-4-ylidene]methyl]-2-butylimidazol-1-yl]methyl]benzoic acidIC502.9 [1]
2-Butyl-5-[(2-nitrophenyl)methyl]-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC502.0 [1]
4-[[2-Butyl-5-[(Z)-[3-(3-methylbutyl)-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC5032.0 [1]
4-[[5-[(Z)-(3-Benzyl-2,5-dioxoimidazolidin-4-ylidene)methyl]-2-butylimidazol-1-yl]methyl]benzoic acidIC5035.0 [1]
2-[2-Ethyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]-N,N-dimethylacetamideIC500.3 [1]
Methyl 4-[[2-butyl-5-[(Z)-[1-butyl-2,5-dioxo-3-(thiophen-2-ylmethyl)imidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoateIC50370.0 [1]
2-Butyl-5-[(2-chlorophenyl)methyl]-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC503.0 [1]
2-Propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5H-imidazo[4,5-c]pyridin-4-oneIC500.7 [1]
2-Butyl-5-[(3-chlorophenyl)methyl]-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC503.0 [1]
2-[2-Butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]-N-phenylacetamideIC501.0 [1]
Ethyl 2-[[2-butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]methyl]benzoateIC502.0 [1]
2-Butyl-5-methyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC500.7 [1]
4-[[2-Butyl-5-[(Z)-(1,3-dibutyl-2,5-dioxoimidazolidin-4-ylidene)methyl]imidazol-1-yl]methyl]benzoic acidIC5014.0 [1]
5-[(2-Aminophenyl)methyl]-2-butyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC502.0 [1]
4-[[2-Butyl-5-[(Z)-[1-butyl-3-[(5-methylthiophen-2-yl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC505.3 [1]
2-Butyl-3-[[4-[2-(butylcarbamoylsulfamoyl)phenyl]phenyl]methyl]-5-methylsulfanylimidazole-4-carboxylic acidIC5097.0 [1]
Methyl 4-[[2-butyl-5-[(Z)-[1-hexyl-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoateIC50100.0 [1]
2-[2-Cyclopropyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]-N,N-dimethylacetamideIC500.5 [1]
Methyl 4-[[2-butyl-5-[(Z)-[1-butyl-3-(1,2-oxazol-5-ylmethyl)-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoateIC50100.0 [1]
Methyl 4-[[5-[(Z)-[3-[(2-amino-1,3-thiazol-4-yl)methyl]-1-butyl-2,5-dioxoimidazolidin-4-ylidene]methyl]-2-butylimidazol-1-yl]methyl]benzoateIC50290.0 [1]
4-[[2-Butyl-5-[(Z)-(3-butyl-2,5-dioxoimidazolidin-4-ylidene)methyl]imidazol-1-yl]methyl]benzoic acidIC5028.0 [1]
Methyl 4-[[2-butyl-5-[(Z)-(3-butyl-2,5-dioxoimidazolidin-4-ylidene)methyl]imidazol-1-yl]methyl]benzoateIC5030.0 [1]
N-[4-[[2-Butyl-5-[(Z)-(3-butyl-2,5-dioxoimidazolidin-4-ylidene)methyl]imidazol-1-yl]methyl]phenyl]-1,1,1-trifluoromethanesulfonamideIC50120.0 [1]
Methyl 4-[[2-butyl-5-[(Z)-[2,5-dioxo-3-(thiophen-2-ylmethyl)imidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoateIC5028.0 [1]
Methyl 4-[[2-butyl-5-[(Z)-[1-butyl-2,5-dioxo-3-(pyridin-2-ylmethyl)imidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoateIC50490.0 [1]
2-Butyl-5-[(2-fluorophenyl)methyl]-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC502.0 [1]
4-[[2-Butyl-5-[(Z)-[1-butyl-3-[(4-methylthiophen-2-yl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC5021.0 [1]
N-Tert-butyl-2-[2-butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]acetamideIC500.1 [1]
Methyl 4-[[2-butyl-5-[(Z)-(1,3-dibutyl-2,5-dioxoimidazolidin-4-ylidene)methyl]imidazol-1-yl]methyl]benzoateIC50460.0 [1]
4-[[2-Butyl-5-[(Z)-[1-butyl-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC502.6 [1]
N-[2-[4-[(2-Butyl-1,4-dioxo-2,3-diazaspiro[4.4]nonan-3-yl)methyl]phenyl]phenyl]sulfonylbenzamideIC5012.0 [1]
Methyl 4-[[2-butyl-5-[(Z)-[1-butyl-3-[(4-chlorophenyl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoateIC50500.0 [1]
2-[4-[(2-Butylimidazol-1-yl)methyl]phenyl]benzoic acidIC509400.0 [1]
2-Butyl-3-[[4-[2-(methylcarbamoylsulfamoyl)phenyl]phenyl]methyl]-5-methylsulfanylimidazole-4-carboxylic acidIC502400.0 [1]
Methyl 4-[[2-butyl-5-[(Z)-[1-butyl-3-(furan-3-ylmethyl)-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoateIC50100.0 [1]
4-[[2-Butyl-5-[(Z)-[1-butyl-2,5-dioxo-3-(thiophen-2-ylmethyl)imidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC5013.0 [1]
(5Z)-1-Butyl-5-[[2-butyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazol-4-yl]methylidene]imidazolidine-2,4-dioneIC5040.0 [1]
2-Butyl-3-[[4-[2-(ethylcarbamoylsulfamoyl)phenyl]phenyl]methyl]-5-methylsulfanylimidazole-4-carboxylic acidIC501900.0 [1]
2-Ethyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5H-imidazo[4,5-c]pyridin-4-oneIC502.0 [1]
N,N-Diethyl-2-[2-ethyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]acetamideIC500.3 [1]
2-Butyl-5-phenacyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC504.0 [1]
2-[2-Butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]-N-methyl-N-phenylacetamideIC500.3 [1]
2-Butyl-5-ethyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC500.6 [1]
2-[[2-Butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]methyl]benzoic acidIC500.8 [1]
4-[[2-Butyl-5-[(E)-[3-(3-methylbutyl)-2,5-dioxoimidazolidin-4-ylidene]methyl]imidazol-1-yl]methyl]benzoic acidIC5074.0 [1]
2-Butyl-5-[(4-chlorophenyl)methyl]-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC5010.0 [1]
3-Phenyl-2-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-2,3-diazaspiro[4.4]nonane-1,4-dioneIC5089.0 [1]
N-[2-[4-[(1,4-Dioxo-2-pentyl-2,3-diazaspiro[4.4]nonan-3-yl)methyl]phenyl]phenyl]sulfonylbenzamideIC5028.0 [1]
N-Pentanoyl-2-[4-(3-butyl-1,4-dioxo-2,3-diazaspiro[4.4]nonane-2-ylmethyl)phenyl]benzenesulfonamideIC5015.0 [1]
N-[2-[4-[(1,4-Dioxo-2-propyl-2,3-diazaspiro[4.4]nonan-3-yl)methyl]phenyl]phenyl]sulfonylbenzamideIC5052.0 [1]
N-[2-[4-[(2-Butyl-4,4-dimethyl-3,5-dioxopyrazolidin-1-yl)methyl]phenyl]phenyl]sulfonylbenzamideIC5026.0 [1]
Methyl 2-[2-butyl-4-oxo-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-5-yl]acetateIC500.2 [1]
2-Butyl-5-(2-oxo-2-pyrrolidin-1-ylethyl)-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazo[4,5-c]pyridin-4-oneIC500.2 [1]
1-[2-[4-[(2-Butyl-1,4-dioxo-2,3-diazaspiro[4.4]nonan-3-yl)methyl]phenyl]phenyl]sulfonyl-3-cyclohexylureaIC5038.0 [1]
2,6-Diethyl-3-iodo-4-[[[2'-(1H-tetrazol-5-yl)-1,1'-biphenyl-4-yl]methyl]oxy]pyridineIC5014.0 [1]
2-Butyl-5-pyrrol-1-yl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazole-4-carboxylic acidIC507.0 [1]
2-Butyl-5-pyrrol-1-yl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazole-4-carbonitrileIC50100.0 [1]
1-[[2'-(2H-Tetrazol-5-yl)-1,1'-biphenyl-4-yl]methyl]-2-butyl-4-[1H-pyrrol-1-yl]-1H-imidazoleIC50400.0 [1]
[2-Butyl-5-pyrrol-1-yl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazol-4-yl]-phenylmethanoneIC505400.0 [1]
Methyl 2-butyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5-[2-(2,2,2-trifluoroacetyl)pyrrol-1-yl]imidazole-4-carboxylateIC5052.0 [1]
2-Butyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5-[2-(2,2,2-trifluoroacetyl)pyrrol-1-yl]imidazole-4-carboxylic acidIC504.0 [1]
Ethyl 2-propyl-5-pyrrol-1-yl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazole-4-carboxylateIC50330.0 [1]
2-Propyl-5-pyrrol-1-yl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazole-4-carboxylic acidIC505.4 [1]
2-Propyl-5-pyrrol-1-yl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]imidazole-4-carbonitrileIC501500.0 [1]
5-[2-[4-[(2-Propyl-4-pyrrol-1-ylimidazol-1-yl)methyl]phenyl]phenyl]-2H-tetrazoleIC503500.0 [1]
2-Propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-5-[2-(2,2,2-trifluoroacetyl)pyrrol-1-yl]imidazole-4-carbonitrileIC50780.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Angiotensin II receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/angiotensin-ii-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Angiotensin II receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/angiotensin-ii-receptor-inhibitors-ic50-ki.
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