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Annexin A2/S100-A10 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC5014000.0 [1], 14125.38 [2]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC50178000.0 [1]
CID 5903185IC50275422.87 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-methylphenyl)acetamideIC5013000.0 [1]
N-(2,4-Dimethylphenyl)-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC5015000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)acetamideIC50129000.0 [1]
CID 655941IC5010000.0 [1]
3-(4-Aminophenylthio)-1-{[3-(4-aminophenylthio)phenyl]sulfonyl}benzeneIC501800.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-ylphenyl)acetamideIC504000.0 [1]
5-Benzyl-4-methyl-2-{[(4-methylphenyl)sulfonyl]amino}thiophene-3-carboxamideIC502100.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methylphenyl)acetamideIC5011000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamideIC5023000.0 [1]
N-(4-Bromophenyl)-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC507000.0 [1]
(4E)-5-(4-Tert-butylphenyl)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)pyrrolidine-2,3-dioneIC5028183.83 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Acetamido-4-methylsulfanylbutanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]-3-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-4-carboxybutanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoyl]amino]-3-sulfanylpropanoyl]amino]-6-aminohexanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]pentanedioic acidIC501202.26 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methyl-1,3-thiazol-2-yl)acetamideIC5030000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(5-methyl-1,2-oxazol-3-yl)acetamideIC5043000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(trifluoromethyl)phenyl]acetamideIC5028000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC509000.0 [1]
N-(4-Chlorophenyl)-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC5017000.0 [1]
N-(3,4-Dimethylphenyl)-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC5032000.0 [1]
N-(3,4-Dimethylphenyl)-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC5052000.0 [1]
2-[[4-(4-Chlorophenyl)-5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(3,4-dimethylphenyl)acetamideIC5059000.0 [1]
N-(3,4-Dimethylphenyl)-3-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamideIC5024000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-ylphenyl)acetamideIC5010000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-ylphenyl)acetamideIC507000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-ylphenyl)acetamideIC5015000.0 [1]
2-[[4-(4-Chlorophenyl)-5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-ylphenyl)acetamideIC5027000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(trifluoromethyl)phenyl]acetamideIC508000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(trifluoromethyl)phenyl]acetamideIC5010000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(trifluoromethyl)phenyl]acetamideIC504000.0 [1]
2-[[4-(4-Chlorophenyl)-5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(trifluoromethyl)phenyl]acetamideIC508000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC507000.0 [1]
N-(4-Chlorophenyl)-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamideIC5022000.0 [1]
2-[[5-[(4,6-Dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)acetamideIC50154000.0 [1]
N-(3,4-Dimethylphenyl)-2-[[4-(furan-2-ylmethyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamideIC501000000.0 [1]
N-(3,4-Dimethylphenyl)-3-[[4-(furan-2-ylmethyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]propanamideIC501000000.0 [1]
2-[[4-(Furan-2-ylmethyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-ylphenyl)acetamideIC5040000.0 [1]
2-[[4-(3-Methoxypropyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-ylphenyl)acetamideIC50164000.0 [1]
N-(3,4-Dimethylphenyl)-2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]acetamideIC5027000.0 [1]
4-Hydroxy-1-(3-imidazol-1-ylpropyl)-2-phenyl-3-(thiophene-2-carbonyl)-2H-pyrrol-5-oneIC50100000.0 [1]
5-[3-(Allyloxy)phenyl]-4-(2-furylcarbonyl)-3-hydroxy-1-(2-methoxyethyl)-1,5-dihydro-2H-pyrrol-2-oneIC50100000.0 [1]
(4E)-1-(2-Hydroxyethyl)-4-[hydroxy-(4-methylphenyl)methylidene]-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC5012022.64 [1]
5-(4-Chlorophenyl)-3-hydroxy-1-(2-hydroxypropyl)-4-(4-methylbenzoyl)-1,5-dihydro-2H-pyrrol-2-oneIC50117489.76 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-propan-2-ylpyrrolidine-2,3-dioneIC501000000.0 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-naphthalen-2-ylpyrrolidine-2,3-dioneIC50128824.96 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-(3-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC5011481.54 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-(4-propylphenyl)pyrrolidine-2,3-dioneIC5018197.01 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-[4-(trifluoromethoxy)phenyl]pyrrolidine-2,3-dioneIC509549.93 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-[4-(trifluoromethyl)phenyl]pyrrolidine-2,3-dioneIC506309.57 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dioneIC508317.64 [1]
(4E)-5-[2,4-Bis(trifluoromethyl)phenyl]-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)pyrrolidine-2,3-dioneIC507585.78 [1]
(4E)-5-[3,5-Bis(trifluoromethyl)phenyl]-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)pyrrolidine-2,3-dioneIC503890.45 [1]
(4E)-5-(3-Chlorophenyl)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)pyrrolidine-2,3-dioneIC50104712.85 [1]
(4E)-5-(3,5-Dichlorophenyl)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)pyrrolidine-2,3-dioneIC506918.31 [1]
(4E)-5-[4-Chloro-3-(trifluoromethyl)phenyl]-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)pyrrolidine-2,3-dioneIC507585.78 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-methylpropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC501000000.0 [1]
(4E)-4-[Hydroxy-(3-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC5079432.82 [1]
(4E)-4-[Hydroxy-(4-methoxyphenyl)methylidene]-1-(2-hydroxypropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC50616595.0 [1]
(4E)-4-[Hydroxy-(3-methoxyphenyl)methylidene]-1-(2-hydroxypropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC506918.31 [1]
(4E)-4-[(2-Ethoxyphenyl)-hydroxymethylidene]-1-(2-hydroxypropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC507079.46 [1]
4-[(E)-Hydroxy-[1-(2-hydroxypropyl)-4,5-dioxo-2-(4-propan-2-ylphenyl)pyrrolidin-3-ylidene]methyl]benzonitrileIC5056234.13 [1]
(4E)-4-[(4-Chlorophenyl)-hydroxymethylidene]-1-(2-hydroxypropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC502691.53 [1]
(4E)-4-[Hydroxy(pyridin-3-yl)methylidene]-1-prop-2-enyl-5-[4-(trifluoromethyl)phenyl]pyrrolidine-2,3-dioneIC501000000.0 [1]
(4E)-4-[Hydroxy-(6-methylpyridin-3-yl)methylidene]-1-prop-2-enyl-5-[4-(trifluoromethyl)phenyl]pyrrolidine-2,3-dioneIC5028183.83 [1]
(4E)-4-[(4-Chlorophenyl)-hydroxymethylidene]-1-prop-2-enyl-5-[4-(trifluoromethyl)phenyl]pyrrolidine-2,3-dioneIC506309.57 [1]
(4E)-4-[Hydroxy(pyridin-3-yl)methylidene]-1-(3-methoxypropyl)-5-[4-(trifluoromethyl)phenyl]pyrrolidine-2,3-dioneIC501000000.0 [1]
(4E)-4-[Hydroxy-(6-methylpyridin-3-yl)methylidene]-1-(3-methoxypropyl)-5-[4-(trifluoromethyl)phenyl]pyrrolidine-2,3-dioneIC50269153.48 [1]
(4E)-5-[3-Fluoro-4-(trifluoromethyl)phenyl]-4-[hydroxy-(6-methylpyridin-3-yl)methylidene]-1-(3-methoxypropyl)pyrrolidine-2,3-dioneIC50181970.09 [1]
(4E)-4-[(4-Chlorophenyl)-hydroxymethylidene]-5-[3-fluoro-4-(trifluoromethyl)phenyl]-1-(3-methoxypropyl)pyrrolidine-2,3-dioneIC50186208.71 [1]
(4E)-4-[(2-Ethoxyphenyl)-hydroxymethylidene]-1-(3-methoxypropyl)-5-[4-(trifluoromethyl)phenyl]pyrrolidine-2,3-dioneIC5010715.19 [1]
(4E)-4-[(2-Ethoxyphenyl)-hydroxymethylidene]-5-[3-fluoro-4-(trifluoromethyl)phenyl]-1-(3-methoxypropyl)pyrrolidine-2,3-dioneIC504897.79 [1]
N-[(6,8-Dimethyl-1,2-dihydroquinolin-3-yl)methyl]-2-(3-methylphenyl)ethanamineIC50100000.0 [1]
(4E)-1-(2-Hydroxypropyl)-4-[hydroxy(pyridin-3-yl)methylidene]-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC50794328.23 [1]
Ethyl 5-cyano-2-methyl-6-[(5-oxo-1,2-dihydropyrazol-3-yl)methylsulfanyl]-4-thiophen-2-yl-3,4-dihydropyridine-3-carboxylateIC5018000.0 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(3-methoxypropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC502884.03 [1]
3-Hydroxy-1-[3-(1H-imidazol-1-yl)propyl]-5-phenyl-4-(phenylcarbonyl)-1,5-dihydro-2H-pyrrol-2-oneIC50100000.0 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-5-(4-propan-2-ylphenyl)-1-prop-2-enylpyrrolidine-2,3-dioneIC506456.54 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-5-(4-hydroxyphenyl)-1-(2-hydroxypropyl)pyrrolidine-2,3-dioneIC501000000.0 [1]
(4E)-5-(4-Ethylphenyl)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)pyrrolidine-2,3-dioneIC5015848.93 [1]
(4E)-4-[Hydroxy(phenyl)methylidene]-1-(2-hydroxypropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC5014454.4 [1]
3-Hydroxy-1-(2-hydroxypropyl)-4-(4-methylbenzoyl)-5-phenyl-1,5-dihydro-2H-pyrrol-2-oneIC50251188.64 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-methoxyethyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dioneIC507585.78 [1]
(4E)-4-[Hydroxy-(4-methylphenyl)methylidene]-1-(2-hydroxypropyl)-5-(4-methylphenyl)pyrrolidine-2,3-dioneIC5085113.8 [1]
6-Methyl-3-(1,3,4,9-tetrahydropyrido[3,4-b]indol-2-ylmethyl)chromen-4-oneIC50100000.0 [1]
N-(3-Methylphenyl)-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}acetamideIC5020000.0 [1]
N-(2,4-Dimethylphenyl)-2-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]acetamideIC5015000.0 [1]
N-(2-Fluorophenyl)-2-[4-(4-methylbenzyl)piperazin-1-yl]acetamideIC50100000.0 [1]
N-(2,5-Dimethylphenyl)-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}acetamideIC508800.0 [1]
2-[(5-Methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]-N-(4-propan-2-ylphenyl)acetamideIC50138000.0 [1]
2-({5-[(2-Methylphenoxy)methyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetamideIC5024000.0 [1]
Items per page: 1 - 10 of 91
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References

This online tool may be cited as follows

MLA

"Quest Database™ Annexin A2/S100-A10 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/annexin-a2-s100-a10-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Annexin A2/S100-A10 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/annexin-a2-s100-a10-inhibitors-ic50-ki.
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