X
Navigation Menu
Products
Services
Tools
Resources
logo
AAT Bioquest

 
search
logo
AAT Bioquest
Contact us
Company
Telephone:1-408-733-1055
Fax:1-408-733-1304
Hours:Monday to Friday
8:30 - 17:30 PST (GMT-8)
Location:5775 W Las Positas Blvd.
Pleasanton, CA, 94588
USA

Email us
Sales:sales@aatbio.com
Technical Support:support@aatbio.com
Website:websupport@aatbio.com
General Inquiries:info@aatbio.com
Order info
United States of America
Telephone:1-408-733-1055
Fax:1-408-733-1304
Email:sales@aatbio.com
Purchase Order:sales@aatbio.com

International
Click here to see all available distributors
Products
Services
Tools
Resources
 
search
calculatorCalculator

Arachidonate 15-lipoxygenase Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
Nordihydroguaiaretic acidIC501100.0 [1]
5-(Methylamino)-2-naphthalen-1-yl-1,3-oxazole-4-carbonitrileIC50200.0 [1], 50000.0 [2]
5-(Methylamino)-2-naphthalen-1-yl-1,3-oxazole-4-carbonitrileKi100.0 [1], 1200.0 [2]
6,11-Dihydro[1]benzothiopyrano[4,3-b]indoleIC50810.0 [1]
6,11-Dihydro[1]benzothiopyrano[4,3-b]indoleKi3810.0 [1]
1H-Imidazole-5-carboxylic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterKi870.0 [1], 1400.0 [2], 8100.0 [3]
Ethyl 6-chloro-3-[(3S)-3,7-dimethyloctanoyl]-1H-indole-2-carboxylateIC5090.0 [1]
Ethyl 6-chloro-3-[(3S)-3,7-dimethyloctanoyl]-1H-indole-2-carboxylateKi30.0 [1], 36.0 [2]
BaicaleinIC509100.0 [1]
BaicaleinKi600.0 [1]
alpha-MangostinIC503100.0 [1], 50000.0 [2]
IndolizineIC5025000.0 [1]
IndolizineKi25000.0 [1]
PuupehenoneIC50760.0 [1], 6000.0 [2]
12-Oxo-ETEIC503000.0 [1]
12-Oxo-ETEKi36800.0 [1]
Phenol, 2,3,5-tribromo-6-(3,5-dibromo-2-hydroxyphenoxy)-IC502200.0 [1], 2500.0 [2]
2,3,4,5-Tetrabromo-6-(3,5-dibromo-2-hydroxyphenoxy)phenolIC50790.0 [1], 1300.0 [2]
JaspaquinolIC50300.0 [1], 19000.0 [2]
4-Fluorobenzoic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterKi10.0 [1]
N-(2-Chlorophenyl)-1H-pyrazole-3-carboxamideIC50618.0 [1], 645.0 [2]
Tribromobisphenol AIC505000.0 [1], 7000.0 [2]
Phenol, 2,3,4,5-tetrabromo-6-(2,4-dibromophenoxy)-IC50700.0 [1], 1800.0 [2]
Jaspic acidIC501400.0 [1], 4700.0 [2]
CID 24825377Ki73.0 [1]
4-[2-(3-Carboxy-4-hydroxynaphthalen-1-yl)-2-oxoacetyl]-1-hydroxynaphthalene-2-carboxylic acidIC5025000.0 [1], 50000.0 [2]
4-Ethyl-6-(4-phenoxy-1H-pyrazol-3-yl)-1,3-BenzenediolIC509200.0 [1]
2-[4-[2-[[Ethyl-[(3S)-1-[1-(4-fluorophenyl)ethyl]pyrrolidin-3-yl]sulfamoyl]amino]ethyl]-5-thiophen-2-yl-1H-pyrazol-3-yl]pyrazineKi1.0 [1]
2,6-Dichloro-4-[1,2,2-tris(3,5-dichloro-4-hydroxyphenyl)ethyl]phenolIC509400.0 [1], 50000.0 [2]
Isojaspic acidIC505300.0 [1], 16000.0 [2]
3-N-(2-Chloro-4-fluorophenyl)-1-N-hexyl-5-methylpyrazole-1,3-dicarboxamideIC5085.0 [1], 395.0 [2]
N-Quinolin-3-yl-1H-pyrazole-5-carboxamideIC5092.0 [1], 180.0 [2]
1h-Pyrazole-3-carboxamide,n-6-quinolinyl-IC50837.0 [1], 970.0 [2]
N-Quinolin-2-yl-1H-pyrazole-5-carboxamideIC50334.0 [1], 3740.0 [2]
1-N-(1,3-Benzodioxol-5-yl)-3-N-(2-chloro-4-fluorophenyl)pyrazole-1,3-dicarboxamideIC5047.0 [1], 109.0 [2]
N-(2-Chloro-4-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]sulfonylpyrazole-3-carboxamideIC501062.0 [1], 1944.0 [2]
4-Bromo-N-(2-chloro-4-fluorophenyl)-1H-pyrazole-5-carboxamideIC5039.0 [1], 290.0 [2]
4-Bromo-5-chloro-N-(2-chloro-4-fluorophenyl)-1H-pyrazole-3-carboxamideIC501.0 [1], 10.0 [2]
N-(2-Chloro-4-fluorophenyl)-4-iodo-1H-pyrazole-5-carboxamideIC50184.0 [1], 551.0 [2]
N-(2-Chloro-4-fluorophenyl)-5-iodo-1H-pyrazole-3-carboxamideIC5027.0 [1], 150.0 [2]
N-(2-Chloro-4-fluorophenyl)-4-nitro-1H-pyrazole-5-carboxamideIC50616.0 [1], 5900.0 [2]
6-Chloro-2-(5-chloro-1H-pyrazol-3-yl)-1,3-benzoxazoleIC504.0 [1], 131.0 [2]
6-Chloro-2-(4,5-dichloro-1H-pyrazol-3-yl)-1,3-benzoxazoleIC502.0 [1], 34.0 [2]
3-Acetyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC502310.0 [1]
3-Acetyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi930.0 [1]
3-Propanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC501780.0 [1]
3-Propanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi720.0 [1]
3-Butanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC50730.0 [1]
3-Butanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi290.0 [1]
Ethyl 6-chloro-3-[(3R)-3,7-dimethyloctanoyl]-1H-indole-2-carboxylateIC50300.0 [1]
Ethyl 6-chloro-3-[(3R)-3,7-dimethyloctanoyl]-1H-indole-2-carboxylateKi120.0 [1]
3-Dodecanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC50430.0 [1]
3-Dodecanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi170.0 [1]
3-Decanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC50200.0 [1]
3-Decanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi80.0 [1]
3-Octanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC50270.0 [1]
3-Octanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi100.0 [1]
3-Hexanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC50540.0 [1]
3-Hexanoyl-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi210.0 [1]
3-(p-Methylphenylacetyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC502080.0 [1]
3-(p-Methylphenylacetyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi830.0 [1]
3-(p-Chlorophenylacetyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC501190.0 [1]
3-(p-Chlorophenylacetyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi480.0 [1]
3-(p-Fluorophenylacetyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC50770.0 [1]
3-(p-Fluorophenylacetyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi310.0 [1]
3-(3-Phenylpropanoyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC50560.0 [1]
3-(3-Phenylpropanoyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi220.0 [1]
4-Chloro-N-(2-chloro-4-fluorophenyl)-1H-pyrazole-5-carboxamideIC5033.0 [1], 85.0 [2]
5-Chloro-N-(2-chloro-4-fluorophenyl)-1H-pyrazole-3-carboxamideIC5022.0 [1], 71.0 [2]
N-(2-Chloro-4-fluorophenyl)-5-(trifluoromethyl)-1H-pyrazole-3-carboxamideIC50112.0 [1], 1000.0 [2]
4,5-Dichloro-N-(2-chloro-4-fluorophenyl)-1H-pyrazole-3-carboxamideIC5014.0 [1], 32.0 [2]
N-Quinolin-3-yl-2H-triazole-4-carboxamideIC501020.0 [1], 1400.0 [2]
N-(2-Chloro-4-fluorophenyl)-1H-1,2,3-triazole-5-carboxamideIC5068.0 [1], 571.0 [2]
N-(2,4-Dichlorophenyl)-1H-1,2,3-triazole-4-carboxamideIC5056.0 [1], 99.0 [2]
N-(4-Fluorophenyl)-2H-triazole-4-carboxamideIC50947.0 [1], 2426.0 [2]
N-(2-Chlorophenyl)-2H-triazole-4-carboxamideIC50392.0 [1], 6976.0 [2]
N-(2,5-Dichlorophenyl)-1H-1,2,3-triazole-5-carboxamideIC5079.0 [1], 22530.0 [2]
N-(5-Fluoropyridin-2-yl)-2H-triazole-4-carboxamideIC503110.0 [1], 3965.0 [2]
N-(5-Fluoropyridin-2-yl)-1H-pyrazole-5-carboxamideIC50118.0 [1], 550.0 [2]
N-(5-Chloropyridin-2-yl)-1H-pyrazole-5-carboxamideIC5026.0 [1], 43.0 [2]
N-[4-(Trifluoromethyl)phenyl]-1H-pyrazole-5-carboxamideIC50448.0 [1], 519.0 [2]
Benzoxazole, 2-(1H-pyrazol-3-yl)-IC50638.0 [1], 3273.0 [2]
6-Chloro-2-(1H-pyrazol-5-yl)-1,3-benzoxazoleIC5013.0 [1], 20.0 [2]
5-Chloro-2-(1H-pyrazol-5-yl)-1,3-benzoxazoleIC50124.0 [1], 443.0 [2]
N-(3,4-Dichlorophenyl)-1H-pyrazole-3-carboxamideIC50180.0 [1], 1320.0 [2]
(1R,3R)-5-[3-[5-[(1R,3R)-6,8-Dihydroxy-1,3-dimethyl-1,2,3,4-tetrahydroisoquinolin-5-yl]-1-hydroxy-8-methoxy-6-methylnaphthalen-2-yl]-4-hydroxy-5-methoxy-7-methylnaphthalen-1-yl]-1,3-dimethyl-1,2,3,4-tetrahydroisoquinoline-6,8-diolIC507600.0 [1], 50000.0 [2]
2-Amino-N-butyl-5-phenylthiophene-3-carboxamideIC5012400.0 [1]
2-Amino-N-butyl-5-phenylthiophene-3-carboxamideKi3300.0 [1]
3-(Phenylacetyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterIC50600.0 [1]
3-(Phenylacetyl)-6-chloro-1H-indole-2-carboxylic acid ethyl esterKi250.0 [1]
4-Amino-N-(2-chloro-4-fluorophenyl)-1H-pyrazole-5-carboxamideIC5069.0 [1], 641.0 [2]
3-Amino-N-(2-chloro-4-fluorophenyl)-1H-pyrazole-5-carboxamideIC50334.0 [1], 5980.0 [2]
N-Pyridin-2-yl-1H-pyrazole-5-carboxamideIC501207.0 [1], 3410.0 [2]
3-N-(2-Chloro-4-fluorophenyl)-1-N-pentylpyrazole-1,3-dicarboxamideIC50130.0 [1], 408.0 [2]
6-{[3-(2-Chloro-4-fluorophenylcarbamoyl)pyrazole-1-carbonyl]-amino}-hexanoic acid ethyl esterIC50141.0 [1], 250.0 [2]
N-(2-Chloro-4-fluorophenyl)-1H-pyrazole-5-carboxamideIC5024.0 [1], 81.0 [2]
N-[4-Fluoro-2-(trifluoromethyl)phenyl]-1H-pyrazole-5-carboxamideIC5094.0 [1], 168.0 [2]
2-(2,3-Dichlorophenyl)-5-(methylamino)-1,3-oxazole-4-carbonitrileIC50460.0 [1], 50000.0 [2]
2-(3,4-Dichlorophenyl)-5-(methylamino)-1,3-oxazole-4-carbonitrileIC50810.0 [1], 50000.0 [2]
5-(Methylamino)-2-naphthalen-1-yl-1,3-thiazole-4-carbonitrileIC50550.0 [1], 50000.0 [2]
Items per page: 1 - 10 of 100
⟨⟩

References

This online tool may be cited as follows

MLA

"Quest Database™ Arachidonate 15-lipoxygenase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/arachidonate-15-lipoxygenase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Arachidonate 15-lipoxygenase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/arachidonate-15-lipoxygenase-inhibitors-ic50-ki.
BibTeXEndNoteRefMan
Location: Home / Datasets / Arachidonate 15-lipoxygenase Inhibitors (IC50, Ki)
AboutPrivacyTerms of UseTerms of SalesDistributors
Copyright © 2024 AAT Bioquest, Inc. All Rights Reserved.