Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| 3-[4-[4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethylpyrazol-3-yl]phenyl]-1,1-dimethylurea | IC50 | 1100.0 [1] | |
| 3-[4-[4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethylpyrazol-3-yl]phenyl]-1,1-dimethylurea | Ki | 490.0 [1] | |
| Tak-901 | IC50 | 21.0 [1] | |
| 1-[3-[5-Chloro-4-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]phenyl]-N,N-dimethylmethanamine | IC50 | 6.2 [1] | |
| 3-(4-(1-Ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl)phenyl)-1,1-dimethylurea | IC50 | 10000.0 [1] | |
MLA | "Quest Database™ Aurora kinase A/Targeting protein for Xklp2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 14 Dec. 2025, https://www.aatbio.com/data-sets/aurora-kinase-a-targeting-protein-for-xklp2-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 14). Quest Database™ Aurora kinase A/Targeting protein for Xklp2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/aurora-kinase-a-targeting-protein-for-xklp2-inhibitors-ic50-ki. | |
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