Aurora kinase A/Targeting protein for Xklp2 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	3-[4-[4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethylpyrazol-3-yl]phenyl]-1,1-dimethylurea	IC50	1100.0 [1]
	3-[4-[4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethylpyrazol-3-yl]phenyl]-1,1-dimethylurea	Ki	490.0 [1]
	Tak-901	IC50	21.0 [1]
	1-[3-[5-Chloro-4-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]phenyl]-N,N-dimethylmethanamine	IC50	6.2 [1]
	3-(4-(1-Ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl)phenyl)-1,1-dimethylurea	IC50	10000.0 [1]
	N,N-Dimethyl-1-[4-[4-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]phenyl]methanamine	IC50	76.0 [1]
	4-(4-Fluorophenyl)-N-[4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]phthalazin-1-amine	IC50	41.0 [1]
	1-[4-[5-Chloro-4-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]phenyl]-N,N-dimethylmethanamine	IC50	7.9 [1]
	4-(1H-Pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine	IC50	584.0 [1]
	1H-Pyrrolo[2,3-b]pyridine, 4-(1-methyl-1H-pyrazol-4-yl)-	IC50	982.0 [1]
	N,N-Dimethyl-1-[3-[4-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]phenyl]methanamine	IC50	128.0 [1]
	N-[3-Methyl-4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]-3-(trifluoromethyl)benzamide	IC50	586.0 [1]
	2-Chloro-N-[3-methyl-4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]benzamide	IC50	25000.0 [1]
	3-Chloro-N-[3-methyl-4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]benzamide	IC50	1546.0 [1]
	4-Chloro-N-[3-methyl-4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]benzamide	IC50	2342.0 [1]
	N-[3-Methyl-4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]-2-phenoxybenzamide	IC50	1544.0 [1]
	N-[3-Methyl-4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]-3-phenoxybenzamide	IC50	964.0 [1]
	2-Anilino-N-[3-methyl-4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]benzamide	IC50	62.0 [1]
	2-Anilino-N-[2-methyl-4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]benzamide	IC50	1000.0 [1]
	2-Anilino-N-[4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]benzamide	IC50	16.0 [1]
	N-[4-[3-[2-(Methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]-4-phenylphthalazin-1-amine	IC50	149.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 21 ⟨⟩

---

---

References

This online tool may be cited as follows

MLA	"Quest Database™ Aurora kinase A/Targeting protein for Xklp2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/aurora-kinase-a-targeting-protein-for-xklp2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Aurora kinase A/Targeting protein for Xklp2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/aurora-kinase-a-targeting-protein-for-xklp2-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan