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B-cell lymphoma 6 protein Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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3-[5-(5-Chloro-2-oxoindol-3-yl)-4-hydroxy-2-sulfanylidene-1,3-thiazol-3-yl]propanoic acidIC5031622.78 [1], 49000.0 [2]
5-[[5-Chloro-2-(pyridin-3-ylmethylamino)pyrimidin-4-yl]amino]-1,3-dihydroindol-2-oneIC50480.0 [1], 8600.0 [2]
(12S,14S,17E)-12-(Hydroxymethyl)-24-oxo-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaene-7-carbonitrileIC502.9 [1], 1995.26 [2]
(12S,14S,17E)-7-Chloro-12-(hydroxymethyl)-23-methyl-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC504.9 [1], 6309.57 [2]
(12S,14S,17E)-23-Benzyl-7-chloro-12-(hydroxymethyl)-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC5011.0 [1], 199.53 [2]
(12S,14S,17E)-7-Chloro-12-(hydroxymethyl)-23-(pyridin-4-ylmethyl)-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC509.9 [1], 398.11 [2]
(12S,14S,17E)-12-(Hydroxymethyl)-23-[(3-methoxyphenyl)methyl]-24-oxo-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaene-7-carbonitrileIC5011.0 [1], 125.89 [2]
(12S,14S,17E)-7-Chloro-12-(hydroxymethyl)-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC501.5 [1], 3981.07 [2]
(12S,14S,17E)-7-Chloro-12-(hydroxymethyl)-23-(3-morpholin-4-ylpropyl)-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC500.87 [1], 1258.93 [2]
(14S)-24-Oxo-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,21(29),22(27)-heptaene-7-carbonitrileIC5024.0 [1], 15848.93 [2]
(12S,14S)-12-(Hydroxymethyl)-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,21(29),22(27)-heptaen-24-oneIC5055.0 [1], 10000.0 [2]
(12S,14S,17E)-7-Chloro-12-(hydroxymethyl)-23-[(4-methylphenyl)methyl]-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC5029.0 [1], 794.33 [2]
(12S,14S,17E)-7-Chloro-23-(cyclopropylmethyl)-12-(hydroxymethyl)-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC5036.0 [1], 5011.87 [2]
(12S,14S)-12-(Hydroxymethyl)-24-oxo-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,21(29),22(27)-heptaene-7-carbonitrileIC502.4 [1], 6309.57 [2]
(12S,14S,17E)-7-Chloro-23-[(3,3-difluorocyclobutyl)methyl]-12-(hydroxymethyl)-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC505.0 [1], 501.19 [2]
(12S,14S,17E)-7-Chloro-12-(hydroxymethyl)-23-[(3-methoxyphenyl)methyl]-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC5012.0 [1], 100.0 [2]
2-[(12S,14S,17E)-7-Chloro-23-[(3,3-difluorocyclobutyl)methyl]-24-oxo-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-12-yl]acetic acidIC5016.0 [1], 3162.28 [2]
(12S,14S)-7-Chloro-12-(hydroxymethyl)-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,21(29),22(27)-heptaen-24-oneIC503.3 [1], 3981.07 [2]
(12S,14S,17E)-7-Chloro-12-(hydroxymethyl)-23-[(2-methylphenyl)methyl]-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-24-oneIC5013.0 [1], 79.43 [2]
2-[5-(5-Bromo-2-oxoindol-3-yl)-4-hydroxy-2-sulfanylidene-1,3-thiazol-3-yl]butanedioic acidIC50212000.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxybutanoyl]amino]-3-carboxypropanoyl]amino]-3-methylpentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-4-methylsulfanylbutanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-methylbutanoyl]pyrrolidine-2-carboxylic acidIC501.0 [1]
1-[2-(1H-Indol-3-yl)ethyl]-3-[3-[(4-methylpiperazin-1-yl)methyl]-1-(2-morpholin-4-yl-2-oxoethyl)indol-6-yl]thioureaIC5027000.0 [1]
2-[(2S)-1-[3-Cyano-7-[(2-oxo-3,4-dihydro-1H-quinolin-6-yl)amino]pyrazolo[1,5-a]pyrimidin-5-yl]pyrrolidin-2-yl]acetic acidIC50350.0 [1]
2-[6-[2-(1H-Indol-3-yl)ethylcarbamothioylamino]-3-[(4-methylpiperazin-1-yl)methyl]indol-1-yl]-N-propan-2-ylacetamideIC50142000.0 [1]
2-[(12S,14S,17E)-7-Cyano-24-oxo-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaen-12-yl]acetic acidIC501.7 [1]
(5S,8E)-6,11-Dioxa-2,17,19,20,24-pentazapentacyclo[16.6.1.12,5.112,16.019,23]heptacosa-1(24),8,12,14,16(26),18(25),20,22-octaene-22-carbonitrileIC502300.0 [1]
N-[4-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]phenyl]acetamideIC5061000.0 [1]
7-(Cyclopropylamino)-5-pyrrolidin-1-ylpyrazolo[1,5-a]pyrimidine-3-carbonitrileIC5099000.0 [1]
7-Anilino-5-pyrrolidin-1-ylpyrazolo[1,5-a]pyrimidine-3-carbonitrileIC50100000.0 [1]
5-[(2R)-2-(Hydroxymethyl)pyrrolidin-1-yl]-7-[(2-oxo-3,4-dihydro-1H-quinolin-6-yl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileIC50590.0 [1]
(3S,5S,8E)-3-(Hydroxymethyl)-6,11-dioxa-2,17,19,20,24-pentazapentacyclo[16.6.1.12,5.112,16.019,23]heptacosa-1(24),8,12,14,16(26),18(25),20,22-octaene-22-carbonitrileIC50390.0 [1]
(15R)-17,25-Dioxo-21-oxa-2,4,5,9,11,18,24-heptazahexacyclo[20.7.1.13,10.04,8.011,15.023,28]hentriaconta-1(29),3(31),5,7,9,22(30),23(28)-heptaene-7-carbonitrileIC50210.0 [1]
2-[(4Z)-4-(5-Bromo-2-oxo-1H-indol-3-ylidene)-2-sulfanylidene-1,3-thiazolidin-3-yl]butanedioic acidIC50212000.0 [1]
2-[(2S)-1-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]pyrrolidin-2-yl]acetic acidIC5064000.0 [1]
7-Anilino-5-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileIC5024000.0 [1]
(2R)-1-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]pyrrolidine-2-carboxylic acidIC5045000.0 [1]
(3R,5S,8E)-3-(Hydroxymethyl)-6,11-dioxa-2,17,19,20,24-pentazapentacyclo[16.6.1.12,5.112,16.019,23]heptacosa-1(24),8,12,14,16(26),18(25),20,22-octaene-22-carbonitrileIC5010000.0 [1]
5-[(2S)-2-(Hydroxymethyl)pyrrolidin-1-yl]-7-[(2-oxo-3,4-dihydro-1H-quinolin-6-yl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileIC50370.0 [1]
(5S,8E,27R)-27-(Hydroxymethyl)-6,11-dioxa-2,17,19,20,24-pentazapentacyclo[16.6.1.12,5.112,16.019,23]heptacosa-1(24),8,12,14,16(26),18(25),20,22-octaene-22-carbonitrileIC508200.0 [1]
7-(Cyclopropylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrileIC5099000.0 [1]
(14S,17E)-24-Oxo-15,20-dioxa-2,4,5,9,11,23-hexazahexacyclo[19.7.1.13,10.111,14.04,8.022,27]hentriaconta-1(28),3(31),5,7,9,17,21(29),22(27)-octaene-7-carbonitrileIC5015.0 [1]
7-[(2-Oxo-3,4-dihydro-1H-quinolin-6-yl)amino]-5-pyrrolidin-1-ylpyrazolo[1,5-a]pyrimidine-3-carbonitrileIC502900.0 [1]
1-[2-(1H-Indol-3-yl)ethyl]-3-[1-[2-(2-methylmorpholin-4-yl)-2-oxoethyl]-3-[(4-methylpiperazin-1-yl)methyl]indol-6-yl]thioureaIC5062000.0 [1]
2-[[2-[6-[2-(1H-Indol-3-yl)ethylcarbamothioylamino]-3-[(4-methylpiperazin-1-yl)methyl]indol-1-yl]acetyl]amino]acetic acidIC50112000.0 [1]
1-[2-(1H-Indol-3-yl)ethyl]-3-[3-[(4-methylpiperazin-1-yl)methyl]-1-(2-oxo-2-piperidin-1-ylethyl)indol-6-yl]thioureaIC5034000.0 [1]
Methyl 2-[6-[2-(1H-indol-3-yl)ethylcarbamothioylamino]-3-[(4-methylpiperazin-1-yl)methyl]indol-1-yl]acetateIC5080000.0 [1]
2-[[2-[6-[2-(1H-Indol-3-yl)ethylcarbamothioylamino]indol-1-yl]acetyl]amino]acetic acidIC50170000.0 [1]
Items per page: 1 - 10 of 47
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References

This online tool may be cited as follows

MLA

"Quest Database™ B-cell lymphoma 6 protein Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/b-cell-lymphoma-6-protein-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ B-cell lymphoma 6 protein Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/b-cell-lymphoma-6-protein-inhibitors-ic50-ki.
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