 | 5-Benzyl-2-(5-benzyl-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl)-3-methylnaphthalene-1,4,6,7-tetrone | IC50 | 122.0 [1], 650.0 [2] |
| 5-Benzyl-2-(5-benzyl-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl)-3-methylnaphthalene-1,4,6,7-tetrone | Ki | 430.0 [1] |
 | Apogossypolone | IC50 | 2170.0 [1] |
| Apogossypolone | Ki | 1470.0 [1] |
 | 2,3,5-Trihydroxy-7-methyl-N-(2-phenylpropyl)-6-[1,6,7-trihydroxy-3-methyl-5-(2-phenylpropylcarbamoyl)naphthalen-2-yl]naphthalene-1-carboxamide | IC50 | 420.0 [1], 730.0 [2] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-morpholino-1H-pyrrole-2,5-dione | IC50 | 450.0 [1], 800.0 [2] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dione | IC50 | 600.0 [1], 800.0 [2] |
 | 3-Chloro-1-(3-chlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dione | IC50 | 1200.0 [1], 2100.0 [2] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-(dimethylamino)pyrrole-2,5-dione | IC50 | 300.0 [1], 400.0 [2] |
 | CID 1180669 | IC50 | 50000.0 [1] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-piperidin-1-ylpyrrole-2,5-dione | IC50 | 50000.0 [1] |
 | N-[2-(4-Ethylphenyl)ethyl]-6-[5-[2-(4-ethylphenyl)ethylcarbamoyl]-3-methyl-1,4,6,7-tetraoxonaphthalen-2-yl]-2,3,5,8-tetrahydroxy-7-methylnaphthalene-1-carboxamide | IC50 | 1250.0 [1] |
| N-[2-(4-Ethylphenyl)ethyl]-6-[5-[2-(4-ethylphenyl)ethylcarbamoyl]-3-methyl-1,4,6,7-tetraoxonaphthalen-2-yl]-2,3,5,8-tetrahydroxy-7-methylnaphthalene-1-carboxamide | Ki | 870.0 [1] |
 | 3-Methyl-5-(2-phenylacetyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-phenylacetyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | IC50 | 690.0 [1] |
| 3-Methyl-5-(2-phenylacetyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-phenylacetyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | Ki | 460.0 [1] |
 | 2,3,5,8-Tetrahydroxy-7-methyl-6-[3-methyl-1,4,6,7-tetraoxo-5-(2-phenylpropylcarbamoyl)naphthalen-2-yl]-N-(2-phenylpropyl)naphthalene-1-carboxamide | IC50 | 710.0 [1] |
| 2,3,5,8-Tetrahydroxy-7-methyl-6-[3-methyl-1,4,6,7-tetraoxo-5-(2-phenylpropylcarbamoyl)naphthalen-2-yl]-N-(2-phenylpropyl)naphthalene-1-carboxamide | Ki | 470.0 [1] |
 | 3-Methyl-5-(2-phenylethyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-phenylethyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | IC50 | 9720.0 [1] |
| 3-Methyl-5-(2-phenylethyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-phenylethyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | Ki | 6470.0 [1] |
 | 5-[(4-Chlorophenyl)methyl]-2-[5-[(4-chlorophenyl)methyl]-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl]-3-methylnaphthalene-1,4,6,7-tetrone | IC50 | 700.0 [1] |
| 5-[(4-Chlorophenyl)methyl]-2-[5-[(4-chlorophenyl)methyl]-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl]-3-methylnaphthalene-1,4,6,7-tetrone | Ki | 470.0 [1] |
 | 3-Methyl-5-(2-methylpropyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-methylpropyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | IC50 | 1410.0 [1] |
| 3-Methyl-5-(2-methylpropyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-methylpropyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | Ki | 930.0 [1] |
 | 3-Methyl-5-[2-(4-methylphenyl)ethyl]-2-[1,4,6,7-tetrahydroxy-3-methyl-5-[2-(4-methylphenyl)ethyl]naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | IC50 | 14700.0 [1] |
| 3-Methyl-5-[2-(4-methylphenyl)ethyl]-2-[1,4,6,7-tetrahydroxy-3-methyl-5-[2-(4-methylphenyl)ethyl]naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | Ki | 9330.0 [1] |
 | 3-Methyl-5-(3-phenylpropyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(3-phenylpropyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | IC50 | 5270.0 [1] |
| 3-Methyl-5-(3-phenylpropyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(3-phenylpropyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetrone | Ki | 3530.0 [1] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-(4-phenylpiperazin-1-yl)pyrrole-2,5-dione | IC50 | 4100.0 [1], 4900.0 [2] |
 | 3-Chloro-1-(3,5-dichlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dione | IC50 | 1900.0 [1], 2400.0 [2] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-(pyrrolidino)-1H-pyrrole-2,5-dione | IC50 | 50000.0 [1] |
 | CID 16654638 | IC50 | 2600.0 [1], 8700.0 [2] |
 | CID 16654639 | IC50 | 11100.0 [1], 23900.0 [2] |
 | 3-Chloranyl-1-(2-chlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dione | IC50 | 1000.0 [1], 3300.0 [2] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-[4-(3-methylphenyl)piperazin-1-yl]pyrrole-2,5-dione | IC50 | 10000.0 [1] |
 | CID 16654652 | IC50 | 300.0 [1], 400.0 [2] |
 | CID 16654653 | IC50 | 600.0 [1], 800.0 [2] |
 | 3-Chloranyl-1-(3,4-dichlorophenyl)-4-[(3S)-3-methylpiperazin-1-yl]pyrrole-2,5-dione | IC50 | 1100.0 [1], 2200.0 [2] |
 | CID 16654655 | IC50 | 250.0 [1], 690.0 [2] |
 | 3-Chloranyl-1-(3,4-dichlorophenyl)-4-(4-ethylpiperazin-1-yl)pyrrole-2,5-dione | IC50 | 1000.0 [1], 1700.0 [2] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-(4-piperonylpiperazino)-3-pyrroline-2,5-quinone | IC50 | 2100.0 [1], 4100.0 [2] |
 | CID 16654662 | IC50 | 1300.0 [1], 2400.0 [2] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrrole-2,5-dione | IC50 | 10000.0 [1] |
 | CID 16654669 | IC50 | 240.0 [1], 620.0 [2] |
 | CID 16654670 | IC50 | 6200.0 [1], 9600.0 [2] |
 | CID 16654672 | IC50 | 8300.0 [1], 10000.0 [2] |
 | CID 16654674 | IC50 | 3300.0 [1], 10500.0 [2] |
 | CID 16654677 | IC50 | 1200.0 [1], 5000.0 [2] |
 | CID 16654679 | IC50 | 2000.0 [1], 5600.0 [2] |
 | CID 16654730 | IC50 | 10800.0 [1], 12600.0 [2] |
 | CID 16654772 | IC50 | 3900.0 [1], 6800.0 [2] |
 | 3-Chloro-1-(2,4-dichlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dione | IC50 | 1400.0 [1], 2600.0 [2] |
 | 1-(4-Chlorophenyl)-3-(4-methylpiperazin-1-yl)-1H-pyrrole-2,5-dione | IC50 | 10000.0 [1] |
 | 1-(3,4-Dichlorophenyl)-3-(4-methylpiperazin-1-yl)pyrrolidine-2,5-dione | IC50 | 10000.0 [1] |
 | 3-Chloro-1-(3,4-dichlorophenyl)-4-(2-hydroxyethylamino)pyrrole-2,5-dione | IC50 | 50000.0 [1] |
 | 3-Chloro-1-(3-chloropyridin-4-yl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dione | IC50 | 29000.0 [1], 35600.0 [2] |
 | Abt-737 | Ki | 20000.0 [1] |
 | (2Z)-2-[(5Z)-5-[(3,5-Dimethyl-1H-pyrrol-2-yl)methylidene]-4-methoxypyrrol-2-ylidene]indole | Ki | 1000.0 [1] |
 | Apogossypol | IC50 | 10000.0 [1] |
 | 2-[4-[(4-Bromophenyl)sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | Ki | 5330.0 [1] |
 | Sabutoclax | IC50 | 620.0 [1] |
 | 2-(1-Hydroxy-4-(thiophene-2-sulfonamido)naphthalen-2-ylthio)acetic acid | Ki | 6140.0 [1] |
 | 2-[1-Hydroxy-4-[[(4-phenoxyphenyl)sulfonyl]amino]-2-naphthylthio]acetic acid | Ki | 3360.0 [1] |
 | 7-[1,3-Dimethyl-5-[[4-(4-methylsulfonylpiperazin-1-yl)phenoxy]methyl]pyrazol-4-yl]-1-(2-morpholin-4-ylethyl)-3-(3-naphthalen-1-yloxypropyl)indole-2-carboxylic acid | Ki | 660.0 [1] |
 | (4S)-4-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-3-(prop-2-enoylamino)propanoyl]amino]-3-methylpentanoyl]amino]propanoyl]amino]-5-amino-5-oxopentanoyl]amino]-5-[[(2S)-1-[[(2S)-1-[[(3S,9S,12S,21S)-21-[[(2S)-1-[[(2S)-4-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-3-(carboxymethyl)-12,21-dimethyl-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclohenicos-16-en-12-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-oxopentanoic acid | IC50 | 8.5 [1] |
 | (4S)-4-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-methylpentanoyl]amino]propanoyl]amino]-5-amino-5-oxopentanoyl]amino]-5-[[(2S)-1-[[(2S)-1-[[(3S,9S,12S,21S)-21-[[(2S)-1-[[(2S)-4-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-3-(carboxymethyl)-12,21-dimethyl-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclohenicos-16-en-12-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-oxopentanoic acid | IC50 | 110.0 [1] |
 | 2,3,5-Trihydroxy-7-methyl-N-(2-phenylethyl)-6-[1,6,7-trihydroxy-3-methyl-5-(2-phenylethylcarbamoyl)naphthalen-2-yl]naphthalene-1-carboxamide | IC50 | 550.0 [1] |
 | N-[2-(4-Ethylphenyl)ethyl]-6-[5-[2-(4-ethylphenyl)ethylcarbamoyl]-1,6,7-trihydroxy-3-methylnaphthalen-2-yl]-2,3,5-trihydroxy-7-methylnaphthalene-1-carboxamide | IC50 | 1300.0 [1] |
 | N-(2,3-Dihydro-1H-inden-2-yl)-6-[5-(2,3-dihydro-1H-inden-2-ylcarbamoyl)-1,6,7-trihydroxy-3-methylnaphthalen-2-yl]-2,3,5-trihydroxy-7-methylnaphthalene-1-carboxamide | IC50 | 670.0 [1] |
 | 3-Methyl-5-(2-phenylethyl)-2-[1,6,7-trihydroxy-3-methyl-5-(2-phenylethyl)naphthalen-2-yl]naphthalene-1,6,7-triol | IC50 | 5000.0 [1] |
 | N-[1-(4-Chlorophenyl)ethyl]-6-[5-[1-(4-chlorophenyl)ethylcarbamoyl]-1,6,7-trihydroxy-3-methylnaphthalen-2-yl]-2,3,5-trihydroxy-7-methylnaphthalene-1-carboxamide | IC50 | 400.0 [1] |
 | N-(Cyclohexylmethyl)-6-[5-(cyclohexylmethylcarbamoyl)-1,6,7-trihydroxy-3-methylnaphthalen-2-yl]-2,3,5-trihydroxy-7-methylnaphthalene-1-carboxamide | IC50 | 2000.0 [1] |
 | 2-[1-Hydroxy-4-[(4-phenylphenyl)sulfonylamino]naphthalen-2-yl]sulfanylacetic acid | Ki | 2340.0 [1] |
 | 2,3,5-Trihydroxy-7-methyl-N-[(2S)-2-phenylpropyl]-6-[1,6,7-trihydroxy-3-methyl-5-[[(2S)-2-phenylpropyl]carbamoyl]naphthalen-2-yl]naphthalene-1-carboxamide | IC50 | 750.0 [1] |
 | 2-[4-[[4-(4-Chlorophenyl)phenyl]sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | Ki | 1110.0 [1] |
 | 2-[1-Hydroxy-4-[(3-phenylphenyl)sulfonylamino]naphthalen-2-yl]sulfanylacetic acid | Ki | 3180.0 [1] |
 | 2-[1-Hydroxy-4-[(2-phenylphenyl)sulfonylamino]naphthalen-2-yl]sulfanylacetic acid | Ki | 17260.0 [1] |
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