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BCoR-BCL6 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
BCL6-IN-8cIC50100.0 [1], 720.0 [2]
5-[2-Chloro-4-nitro-5-(oxan-4-yloxy)anilino]-1,3-dihydroindol-2-oneIC50130.0 [1], 1200.0 [2]
5-[2-Chloro-5-(3-hydroxypropylamino)-4-nitroanilino]-1,3-dihydrobenzimidazol-2-oneIC50240.0 [1], 100000.0 [2]
7-Nitro-N~4~-phenyl-2,1,3-benzoxadiazole-4,6-diamineIC5069000.0 [1]
2-[5-(5-Bromo-2-oxoindol-3-yl)-4-hydroxy-2-sulfanylidene-1,3-thiazol-3-yl]butanedioic acidIC50200000.0 [1]
3-[4-Chloro-2-nitro-5-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)amino]anilino]propanoic acidIC50130.0 [1]
Ethyl 3-[4-chloro-2-nitro-5-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)amino]anilino]propanoateIC50430.0 [1]
3-Chloro-4-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)amino]benzonitrileIC50110000.0 [1]
5-[2-Chloro-4-nitro-5-(oxan-4-yloxy)anilino]-1,3-dihydrobenzimidazol-2-oneIC50220.0 [1]
5-[4-Nitro-2-(trifluoromethyl)anilino]-1,3-dihydrobenzimidazol-2-oneIC50300000.0 [1]
5-(2-Bromo-4-nitroanilino)-1,3-dihydrobenzimidazol-2-oneIC5083000.0 [1]
Methyl 3-chloro-4-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)amino]benzoateIC508600.0 [1]
5-[2-Chloro-4-nitro-5-(oxan-4-ylamino)anilino]-1,3-dihydrobenzimidazol-2-oneIC50130.0 [1]
3-Chloro-4-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)amino]benzamideIC5043000.0 [1]
5-Nitro-2-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)amino]benzonitrileIC504300.0 [1]
5-[2-Chloro-4-nitro-5-(pyridin-3-ylmethylamino)anilino]-1,3-dihydrobenzimidazol-2-oneIC50150.0 [1]
3-Chloro-4-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)amino]benzoic acidIC5062000.0 [1]
5-[(2-Chloranyl-4-Nitro-Phenyl)amino]-1,3-Dihydrobenzimidazol-2-OneIC504500.0 [1]
3-((7-((4-Fluorophenyl)amino)-4-nitrobenzo[c][1,2,5]oxadiazol-5-yl)amino)propan-1-olIC5014000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ BCoR-BCL6 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/bcor-bcl6-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ BCoR-BCL6 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bcor-bcl6-inhibitors-ic50-ki.
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