Beta-1,4-mannosyl-glycoprotein 4-beta-N-acetylglucosaminyltransferase Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	N-(2-Cyclobutyltriazol-4-yl)-2-[2-(3-methoxyphenyl)acetyl]-1,3-dihydroisoindole-5-sulfonamide	IC50	100.0 [1], 204.17 [2]
	2-[2-(3-Methoxyphenyl)acetyl]-N-[2-(oxan-3-yl)triazol-4-yl]-1,3-dihydroisoindole-5-sulfonamide	IC50	79.43 [1], 794.33 [2]
	N-[2-(3,3-Difluorocyclobutyl)triazol-4-yl]-2-[2-(3-methoxyphenyl)acetyl]-1,3-dihydroisoindole-5-sulfonamide	IC50	63.1 [1], 389.05 [2]
	N-[5-[(2,4-Difluorophenyl)sulfamoyl]-1-(2-phenylethyl)-2,3-dihydroindol-7-yl]acetamide	IC50	30000.0 [1]
	N-[2-(3-Fluorophenyl)ethyl]-2-[2-(3-methoxyphenyl)acetyl]-1,3-dihydroisoindole-5-sulfonamide	IC50	630.96 [1]
	N-[2-(3-Fluorophenyl)ethyl]-2-[2-(3-methoxyphenyl)acetyl]-N-methyl-1,3-dihydroisoindole-5-sulfonamide	IC50	2511.89 [1]
	2-[2-(3-Methoxyphenyl)acetyl]-N-(2-methyltriazol-4-yl)-1,3-dihydroisoindole-5-sulfonamide	IC50	3981.07 [1]
	2-[2-(3-Methoxyphenyl)acetyl]-N-(2-phenyltriazol-4-yl)-1,3-dihydroisoindole-5-sulfonamide	IC50	6.31 [1]
	N-[2-(4-Fluorophenyl)triazol-4-yl]-2-[2-(3-methoxyphenyl)acetyl]-1,3-dihydroisoindole-5-sulfonamide	IC50	6.31 [1]
	2-[2-(3-Methoxyphenyl)acetyl]-N-(2-propan-2-yltriazol-4-yl)-1,3-dihydroisoindole-5-sulfonamide	IC50	630.96 [1]
	2-[2-(3-Methoxyphenyl)acetyl]-N-[2-(oxetan-3-yl)triazol-4-yl]-1,3-dihydroisoindole-5-sulfonamide	IC50	398.11 [1]
	(3S)-N-(2,4-Difluorophenyl)-3-ethyl-3-methyl-2,5-dioxo-1,4-dihydro-1,4-benzodiazepine-7-sulfonamide	IC50	50.12 [1]
	(3S)-N-[4-(Difluoromethoxy)phenyl]-3-ethyl-3-methyl-2,5-dioxo-1,4-dihydro-1,4-benzodiazepine-7-sulfonamide	IC50	125.89 [1]
	3-Ethyl-3-methyl-2,5-dioxo-N-phenyl-1,4-dihydro-1,4-benzodiazepine-7-sulfonamide	IC50	2511.89 [1]
	N-(4-Chlorophenyl)-3-ethyl-3-methyl-2,5-dioxo-1,4-dihydro-1,4-benzodiazepine-7-sulfonamide	IC50	398.11 [1]
	[(3R)-1-[8-[1-(4-Chloropyrazol-1-yl)ethyl]-7H-purin-2-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone	IC50	50000.0 [1]
	[(3R)-1-[2-[(1S)-1-(4-Chloropyrazol-1-yl)ethyl]-1H-imidazo[4,5-b]pyridin-5-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone	IC50	50000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

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References

This online tool may be cited as follows

MLA	"Quest Database™ Beta-1,4-mannosyl-glycoprotein 4-beta-N-acetylglucosaminyltransferase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/beta-1-4-mannosyl-glycoprotein-4-beta-n-acetylglucosaminyltransferase-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Beta-1,4-mannosyl-glycoprotein 4-beta-N-acetylglucosaminyltransferase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/beta-1-4-mannosyl-glycoprotein-4-beta-n-acetylglucosaminyltransferase-inhibitors-ic50-ki.
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