 | Salmeterol | IC50 | 5.01 [1] |
 | 1-[(7-Methyl-2,3-dihydro-1H-inden-4-yl)oxy]-3-(propan-2-ylamino)-2-butanol | IC50 | 0.49 [1], 0.74 [2], 1.2 [3], 2.3 [4], 2.5 [5] |
| 1-[(7-Methyl-2,3-dihydro-1H-inden-4-yl)oxy]-3-(propan-2-ylamino)-2-butanol | Ki | 0.13 [1], 1.0 [2] |
 | Propranolol | IC50 | 50.12 [1] |
| Propranolol | Ki | 0.46 [1], 0.77 [2], 1.74 [3], 3.69 [4] |
 | Isoprenaline | Ki | 2.44 [1], 46.0 [2], 169.0 [3], 192.0 [4], 676.08 [5] |
 | Salbutamol | IC50 | 1995.26 [1] |
| Salbutamol | Ki | 510.0 [1], 557.0 [2], 1828.0 [3] |
 | 2-(4-((2R)-2-(((2R)-2-(3-Chlorophenyl)-2-hydroxyethyl)amino)propyl)phenoxy)acetic acid | IC50 | 3000.0 [1] |
| 2-(4-((2R)-2-(((2R)-2-(3-Chlorophenyl)-2-hydroxyethyl)amino)propyl)phenoxy)acetic acid | Ki | 630.0 [1], 2850.0 [2] |
 | R,R-Fenoterol | IC50 | 0.14 [1] |
| R,R-Fenoterol | Ki | 4.0 [1], 345.0 [2], 346.74 [3] |
 | 5-[(1R)-1-Hydroxy-2-[[(2R)-1-(4-methoxyphenyl)propan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 0.17 [1] |
| 5-[(1R)-1-Hydroxy-2-[[(2R)-1-(4-methoxyphenyl)propan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 4.09 [1], 474.0 [2], 478.63 [3] |
 | 5-[(1R)-1-Hydroxy-2-[[(2S)-1-(4-methoxyphenyl)propan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 2.01 [1] |
| 5-[(1R)-1-Hydroxy-2-[[(2S)-1-(4-methoxyphenyl)propan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 26.1 [1], 1930.0 [2], 1949.84 [3] |
 | (S,R)-(+)-Fenoterol | IC50 | 6.74 [1] |
| (S,R)-(+)-Fenoterol | Ki | 1828.1 [1], 10232.93 [2], 10330.0 [3] |
 | (R,S)-(-)-Fenoterol | IC50 | 6.09 [1] |
| (R,S)-(-)-Fenoterol | Ki | 183.0 [1], 3695.0 [2], 3715.35 [3] |
 | (S,S)-(+)-Fenoterol | IC50 | 184.2 [1] |
| (S,S)-(+)-Fenoterol | Ki | 3372.87 [1], 27542.29 [2], 27749.0 [3] |
 | Indacaterol | Ki | 20.6 [1], 76.0 [2] |
 | 1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol | IC50 | 6.1 [1] |
| 1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol | Ki | 43.65 [1] |
 | CID 9829836 | IC50 | 190.0 [1], 3000.0 [2] |
| CID 9829836 | Ki | 160.0 [1] |
 | L-796568 Free base | IC50 | 670.0 [1], 2300.0 [2] |
 | 2-(2-Amino-1,3-thiazol-4-yl)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]acetamide | IC50 | 20000.0 [1] |
 | 5-[(1S)-1-Hydroxy-2-[[(2R)-1-(4-methoxyphenyl)propan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 3.16 [1] |
| 5-[(1S)-1-Hydroxy-2-[[(2R)-1-(4-methoxyphenyl)propan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 91.3 [1], 5248.07 [2] |
 | 5-[(1S)-1-Hydroxy-2-[[(2S)-1-(4-methoxyphenyl)propan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 337.2 [1] |
| 5-[(1S)-1-Hydroxy-2-[[(2S)-1-(4-methoxyphenyl)propan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 2870.0 [1], 15848.93 [2] |
 | 5-[(1R)-1-Hydroxy-2-[[(2S)-1-naphthalen-1-ylpropan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 1.19 [1] |
| 5-[(1R)-1-Hydroxy-2-[[(2S)-1-naphthalen-1-ylpropan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 338.84 [1], 341.0 [2] |
 | 5-[(1R)-1-Hydroxy-2-[[(2R)-1-naphthalen-1-ylpropan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 229.1 [1] |
| 5-[(1R)-1-Hydroxy-2-[[(2R)-1-naphthalen-1-ylpropan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 239.88 [1], 241.0 [2] |
 | 5-[(1R)-1-Hydroxy-2-[[(2R)-1-(4-methoxynaphthalen-1-yl)propan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 3.98 [1] |
| 5-[(1R)-1-Hydroxy-2-[[(2R)-1-(4-methoxynaphthalen-1-yl)propan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 13.3 [1], 280.0 [2] |
 | 5-[(1R)-1-Hydroxy-2-[[(2R)-1-(4-hydroxyphenyl)butan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 1.44 [1] |
| 5-[(1R)-1-Hydroxy-2-[[(2R)-1-(4-hydroxyphenyl)butan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 39.1 [1], 1270.0 [2] |
 | 5-[(1R)-1-Hydroxy-2-[[(2S)-1-(4-hydroxyphenyl)butan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 17.88 [1] |
| 5-[(1R)-1-Hydroxy-2-[[(2S)-1-(4-hydroxyphenyl)butan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 294.0 [1], 5760.0 [2] |
 | 5-[(1R)-1-Hydroxy-2-[[(2S)-1-(4-methoxynaphthalen-1-yl)propan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 4.37 [1] |
| 5-[(1R)-1-Hydroxy-2-[[(2S)-1-(4-methoxynaphthalen-1-yl)propan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 12.7 [1], 320.0 [2] |
 | 5-[(1S)-1-Hydroxy-2-[[(2R)-1-naphthalen-1-ylpropan-2-yl]amino]ethyl]benzene-1,3-diol | IC50 | 14.8 [1] |
| 5-[(1S)-1-Hydroxy-2-[[(2R)-1-naphthalen-1-ylpropan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 1778.28 [1], 1784.0 [2] |
 | (6Ar,7R)-1,2-dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-7-ol | IC50 | 1.4 [1], 6.9 [2] |
| (6Ar,7R)-1,2-dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-7-ol | Ki | 13.0 [1] |
 | Epinephrine | Ki | 196.0 [1], 360.0 [2] |
 | Atenolol | Ki | 9549.93 [1], 10061.0 [2] |
 | Pindolol | Ki | 0.38 [1], 0.4 [2] |
 | Timolol | Ki | 0.2 [1], 0.21 [2] |
 | Clenbuterol | Ki | 28.0 [1], 570.0 [2] |
 | Levalbuterol | Ki | 3801.89 [1], 4677.35 [2] |
 | Darifenacin | Ki | 15.9 [1], 61.0 [2] |
 | 1-(Isopropylamino)-3-(1-naphthyloxy)-2-propanol | IC50 | 0.78 [1] |
| 1-(Isopropylamino)-3-(1-naphthyloxy)-2-propanol | Ki | 0.24 [1] |
 | 4-(3-Hexyl-2-oxoimidazol-1-yl)-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamide | IC50 | 12000.0 [1] |
 | Milveterol | Ki | 3.16 [1] |
 | 1-Hexyl-3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]urea | IC50 | 3000.0 [1] |
 | 4-(3-Hexyl-2-oxoimidazolidin-1-yl)-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamide | IC50 | 2300.0 [1] |
 | 1-[4-(Diphenylmethyl)piperazin-1-yl]-3-[(3-methyl-1H-indol-4-yl)oxy]propan-2-ol | Ki | 0.3 [1], 0.31 [2] |
 | 1-(3,5-Diiodo-4-methoxybenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diol | Ki | 2.04 [1] |
 | [3-[(2R)-2-[[(2R)-2-Hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate | Ki | 48.0 [1] |
 | N-[4-[2-[[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-octyl-2-oxoimidazolidin-1-yl)benzenesulfonamide | IC50 | 380.0 [1] |
 | CID 16118894 | IC50 | 120.0 [1] |
 | 1-(4-Methoxyphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol | Ki | 700.0 [1] |
 | N-[4-[2-[[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-octyl-2-oxoimidazol-1-yl)benzenesulfonamide | IC50 | 330.0 [1] |
 | 1-(Benzo[b]thiophen-2-yl)-N-methylmethanamine | Ki | 43200.0 [1], 373000.0 [2] |
 | 7-((R)-2-((1S,2S)-2-(Benzyloxy)cyclopentylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one | Ki | 2.5 [1], 6.1 [2] |
 | 4-[4-(3,4-Difluorophenyl)-1,3-thiazol-2-yl]-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamide | IC50 | 1700.0 [1] |
 | 2-(Hydroxymethyl)-4-[2-hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]phenol | IC50 | 2250.0 [1] |
| 2-(Hydroxymethyl)-4-[2-hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]phenol | Ki | 14.0 [1] |
 | 1-[2-(2-Phenylphenoxy)ethylamino]propan-2-ol | Ki | 9.0 [1], 470.0 [2] |
 | 6-[2-[[2-Hydroxy-3-(1H-indol-4-yloxy)propyl]amino]propoxy]-4H-1,4-benzoxazin-3-one | Ki | 0.63 [1], 1.58 [2] |
 | 6-[2-[3-(1H-Indol-4-yloxy)propylamino]ethoxy]-4H-1,4-benzoxazin-3-one | Ki | 1000.0 [1] |
 | 4-[(2S)-2-Hydroxy-3-[[1-(4-methoxyphenyl)-2-methylpropan-2-yl]amino]propoxy]-1,3-dihydrobenzimidazol-2-one | IC50 | 0.0 [1], 1.3 [2] |
 | 7-[(1R)-2-[[(1R,2R)-2-Cyclopentylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one | Ki | 0.6 [1], 0.8 [2] |
 | (6S)-N-[4-[[(2S,5R)-5-[(R)-Hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamide | IC50 | 20000.0 [1] |
 | (4R)-N-[4-[[(2S,5R)-5-[(R)-Hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide | IC50 | 20000.0 [1] |
 | 4-(3,5-Diiodo-4-methoxybenzyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-amine | IC50 | 56.0 [1] |
| 4-(3,5-Diiodo-4-methoxybenzyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-amine | Ki | 426.58 [1] |
 | 1H-Indole-3-ethanamine, 5-methoxy-1-methyl- | Ki | 20400.0 [1], 36200.0 [2] |
 | Ethyl (1S,5R)-3-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylate | IC50 | 13400.0 [1], 20000.0 [2] |
 | N-(1-Benzothiophen-2-ylmethyl)-3-methyloxetan-3-amine | Ki | 1000000.0 [1] |
 | N-[2-(5-Methoxy-1-methylindol-3-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]propan-1-amine | Ki | 10400.0 [1], 25000.0 [2] |
 | N-[[2-Fluoro-5-(trifluoromethoxy)phenyl]methyl]-2-(5-methoxy-1-methylindol-3-yl)ethanamine | Ki | 80400.0 [1], 83800.0 [2] |
 | 1-(2-Methylphenyl)-N-[(4-pyrimidin-2-ylphenyl)methyl]ethanamine | Ki | 4390.0 [1], 268000.0 [2] |
 | 3-(4-Chlorophenyl)-N-[2-(5-methoxy-1-methylindol-3-yl)ethyl]propan-1-amine | Ki | 520.0 [1], 3900.0 [2] |
 | 2-(Furan-2-yl)-2-[[4-(1,3-thiazol-2-yl)phenyl]methylamino]ethanol | Ki | 95400.0 [1], 1000000.0 [2] |
 | 4,4,4-Trifluoro-N-[[4-(1,3-thiazol-2-yl)phenyl]methyl]butan-2-amine | Ki | 52300.0 [1], 393000.0 [2] |
 | 5-[(1S)-1-Hydroxy-2-[[(2R)-1-phenylpropan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 22908.68 [1], 23125.0 [2] |
 | 5-[(1S)-1-Hydroxy-2-[[(2S)-1-phenylpropan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 28624.0 [1], 28840.32 [2] |
 | (S)-(+)-5-(1-Hydroxy-2-phenethylaminoethyl)-1,3-benzenediol | Ki | 20417.38 [1], 20562.0 [2] |
 | 5-[(1S)-1-Hydroxy-2-[[(2S)-1-naphthalen-1-ylpropan-2-yl]amino]ethyl]benzene-1,3-diol | Ki | 2511.89 [1], 2535.0 [2] |
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