beta-catenin-B-cell lymphoma 9 protein complex Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Carnosic acid	Ki	5300.0 [1]
	[3-Cyclohexyl-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]methanone;dihydrochloride	IC50	5600.0 [1]
	[3-(4-Fluorophenyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-[3-fluoro-5-[(3R)-pyrrolidin-3-yl]oxybenzoyl]piperazin-1-yl]methanone;dihydrochloride	Ki	35000.0 [1]
	[3-(4-Fluorophenyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-fluoro-5-piperidin-4-ylbenzoyl)piperazin-1-yl]methanone;dihydrochloride	Ki	20000.0 [1]
	[3-(3,4-Difluorophenyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]methanone;dihydrochloride	Ki	57000.0 [1]
	[4-(3-Fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]-[3-(4-methylcyclohexyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]methanone;dihydrochloride	Ki	37000.0 [1]
	[4-(3-Fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]-[4-[(3S)-pyrrolidin-3-yl]oxy-3-[4-(trifluoromethyl)cyclohexyl]phenyl]methanone;dihydrochloride	Ki	16000.0 [1]
	[3-(4-Fluorophenyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]methanone;dihydrochloride	Ki	19000.0 [1]
	[4-[5-(4-Fluorophenyl)-6-[(3S)-pyrrolidin-3-yl]oxypyridine-3-carbonyl]piperazin-1-yl]-(3-fluoro-5-piperazin-1-ylphenyl)methanone;dihydrochloride	Ki	82000.0 [1]
	[3-(2-Aminoethyl)-5-fluorophenyl]-[4-[5-(4-fluorophenyl)-6-[(3S)-pyrrolidin-3-yl]oxypyridine-3-carbonyl]piperazin-1-yl]methanone;dihydrochloride	Ki	500000.0 [1]
	[4-[3-(2-Aminoethyl)-5-fluorobenzoyl]piperazin-1-yl]-[3-(4-fluorophenyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]methanone;dihydrochloride	Ki	67000.0 [1]
	[3-(4-Fluorophenyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-[3-fluoro-5-[(3S)-pyrrolidin-3-yl]oxybenzoyl]piperazin-1-yl]methanone;dihydrochloride	Ki	48000.0 [1]
	[4-(3-Chloro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]-[3-cyclohexyl-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]methanone;dihydrochloride	Ki	76000.0 [1]
	[3-Cyclohexyl-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-methyl-5-piperazin-1-ylbenzoyl)piperazin-1-yl]methanone;dihydrochloride	Ki	25000.0 [1]
	[3-Cyclohexyl-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-[3-piperazin-1-yl-5-(trifluoromethyl)benzoyl]piperazin-1-yl]methanone;dihydrochloride	Ki	69000.0 [1]
	[4-(3-Bromo-5-piperazin-1-ylbenzoyl)piperazin-1-yl]-[3-cyclohexyl-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]methanone;dihydrochloride	Ki	55000.0 [1]
	3-(3,4-Difluorophenyl)-N-[3-(4-fluorophenyl)-4-pyrrolidin-3-yloxyphenyl]-4-[(3S)-pyrrolidin-3-yl]oxybenzamide	Ki	2100.0 [1]
	4-(2-Aminoethoxy)-3-(4-fluorophenyl)benzamide	Ki	130000.0 [1]
	[3-(4-Ethylcyclohexyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]methanone	Ki	170000.0 [1]
	[3-(4,4-Dimethylcyclohexyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]methanone	Ki	70000.0 [1]
	[3-(4,4-Difluorocyclohexyl)-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]methanone	Ki	45000.0 [1]
	[3-Cyclopentyl-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]-[4-(3-fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]methanone	Ki	53000.0 [1]
	[4-(3-Fluoro-5-piperazin-1-ylbenzoyl)piperazin-1-yl]-[3-methyl-4-[(3S)-pyrrolidin-3-yl]oxyphenyl]methanone	Ki	490000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

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References

This online tool may be cited as follows

MLA	"Quest Database™ beta-catenin-B-cell lymphoma 9 protein complex Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/beta-catenin-b-cell-lymphoma-9-protein-complex-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ beta-catenin-B-cell lymphoma 9 protein complex Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/beta-catenin-b-cell-lymphoma-9-protein-complex-inhibitors-ic50-ki.
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