Beta-galactoside alpha-2,6-sialyltransferase 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	[[[(2R,3S,4R,5R)-5-(4-Amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-cyclopentylmethyl]phosphonic acid	Ki	5852.0 [1]
	[(2S,3S)-3-(Acetamidomethyl)-1-[[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-2-phenylmethoxycyclopentyl]phosphonic acid	Ki	477.0 [1]
	3',4'-Dihydroxyflavonol	IC50	7500.0 [1]
	3',4'-Dihydroxyflavone	IC50	7100.0 [1]
	Stachybotrydial	IC50	610.0 [1]
	Trisodium;[[(2R,3R,4S)-3-acetamido-4-hydroxy-2-phenoxy-3,4-dihydro-2H-pyran-6-yl]-phosphonatomethyl] [(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl phosphate	Ki	690.0 [1]
	Stachybotrolide	IC50	8000.0 [1]
	Trisodium;[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2-benzamido-1-phosphonatoethyl) phosphate	Ki	174.0 [1]
	Trisodium;[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2-oxo-1-phosphonato-2-pyrrolidin-1-ylethyl) phosphate	Ki	165.0 [1]
	Trisodium;[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl [phenyl(phosphonato)methyl] phosphate	Ki	1000.0 [1]
	Trisodium;[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl [2-(2,5-dioxopyrrolidin-1-yl)-1-phosphonatoethyl] phosphate	Ki	224.0 [1]
	Trisodium;[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2-oxo-1-phosphonato-2-piperidin-1-ylethyl) phosphate	Ki	45.0 [1]
	Trisodium;[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2-anilino-2-oxo-1-phosphonatoethyl) phosphate	Ki	122.0 [1]
	(4S)-5-[[(3R,5R,8R,9S,10S,13R,14S,17R)-17-[(2R)-4-Carboxybutan-2-yl]-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl]oxy]-4-[(4-nitro-2,1,3-benzoxadiazol-7-yl)amino]-5-oxopentanoic acid	IC50	1500.0 [1]
	(2R,3S,4As,7R,8R,8aS)-2,3,4'-trihydroxy-4,4,7,8a-tetramethylspiro[2,3,4a,5,6,7-hexahydro-1H-naphthalene-8,2'-3,8-dihydrofuro[3,4-g][1]benzofuran]-6'-one	IC50	18500.0 [1]
	[[(1S,3S,4R)-3-Acetamido-4-hydroxycyclopentyl]-[[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxymethyl]phosphonic acid	Ki	4314.0 [1]
	[[(1S,3S,4R)-3-Acetamido-4-phenylmethoxycyclopentyl]-[[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxymethyl]phosphonic acid	Ki	1629.0 [1]
	[[(1R,3S,4R)-3-Acetamido-4-phenylmethoxycyclopentyl]-[[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxymethyl]phosphonic acid	Ki	1510.0 [1]
	[[(1R,3S,4R)-3-(Acetamidomethyl)-4-phenylmethoxycyclopentyl]-[[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxymethyl]phosphonic acid	Ki	865.0 [1]
	[[[(2R,3S,4R,5R)-5-(4-Amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-(3-phenoxyphenyl)methyl]phosphonic acid	Ki	19.0 [1]
	[(R)-[[(2R,3S,4R,5R)-5-(4-Amino-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-(3-phenoxyphenyl)methyl]phosphonic acid	Ki	19.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 21 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Beta-galactoside alpha-2,6-sialyltransferase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/beta-galactoside-alpha-2-6-sialyltransferase-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Beta-galactoside alpha-2,6-sialyltransferase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/beta-galactoside-alpha-2-6-sialyltransferase-1-inhibitors-ic50-ki.
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