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Bile acid receptor FXR Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
GuggulsteroneIC5012000.0 [1], 44900.0 [2], 89360.0 [3], 89400.0 [4], 100000.0 [5]
GuggulsteroneKi5000.0 [1]
E-GuggulsteroneIC504100.0 [1], 41000.0 [2], 44000.0 [3], 100000.0 [4]
E-GuggulsteroneKi5000.0 [1]
(E)-3-(2-Chloro-4-((3-(2,6-dichlorophenyl)-5-isopropylisoxazol-4-yl)methoxy)styryl)benzoic acidIC5019.8 [1], 64.0 [2], 112.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseBile acid receptor FXR Inhibitors (IC50, Ki)." AAT Bioquest, Inc.6 Dec2025https://www.aatbio.com/data-sets/bile-acid-receptor-fxr-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 6). Quest DatabaseBile acid receptor FXR Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bile-acid-receptor-fxr-inhibitors-ic50-ki.
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