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Bombesin receptor subtype-3 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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CID 46200989IC503.6 [1]
2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]benzoic acidIC5011.0 [1]
2-(4-(2-(4-(2,2-Dimethylbutyl)-1H-imidazol-2-yl)ethyl)phenyl)-5-fluoropyridineIC5016.0 [1], 19.0 [2]
CID 49871766Ki3.7 [1]
2-(4-(2-(4-(2,2-Dimethylbutyl)-1H-imidazol-2-yl)ethyl)phenyl)pyridineIC5018.0 [1]
4-(Bicyclo[2.2.1]hept-2-ylamino)-3-({[(isopropylamino)carbonyl]amino}sulfonyl)pyridineIC50600.0 [1]
CID 56840673IC501.4 [1]
2-[4-[2-(5-Butyl-1H-imidazol-2-yl)-5-hydroxypentyl]phenyl]benzoic acidIC503676.0 [1]
(2S)-2-[[2-[2-[4-[3-(2-Aminoethylamino)-2-[(2-aminoethylamino)methyl]propyl]anilino]-2-oxoethoxy]acetyl]amino]-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-4-methylsulfanyl-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]pentanediamideIC5037.0 [1]
(2S)-2-[[2-[2-[4-[3-(2-Aminoethylamino)-2-[(2-aminoethylamino)methyl]propyl]anilino]-2-oxoethoxy]acetyl]amino]-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-1-oxohexan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]pentanediamideIC50100.0 [1]
1-[4-[[(1R,2S,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3-propan-2-ylureaIC50820.0 [1]
1-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3-propan-2-ylureaIC50510.0 [1]
3-[[2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]phenoxy]methyl]-1,4-dihydro-1,2,4-triazol-5-oneIC5031.0 [1]
3-[6-(4-Tert-butylphenyl)sulfonyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-7-yl]-4H-1,2,4-oxadiazol-5-oneIC5029.0 [1]
1-(4-(2-(4-(2,2-Dimethylbutyl)-1H-imidazol-2-yl)ethyl)phenyl)-1H-pyrazoleIC5033.0 [1]
5-[[2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]phenoxy]methyl]-2H-tetrazoleIC505.3 [1]
2-(4-Pyrazol-1-ylphenyl)-1-[5-[[1-(trifluoromethyl)cyclopropyl]methyl]-1H-imidazol-2-yl]propan-2-olIC5011.0 [1]
2-(4-(2-(4-(2,2-Dimethylbutyl)-1H-imidazol-2-yl)ethyl)phenyl)-6-methylpyridineIC506.3 [1]
7-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]-1,4,5,6-tetrahydropyrazolo[3,4-b]pyridineIC5018.0 [1]
1-[4-(2,2-Dimethylpropyl)-1h-imidazol-2-yl]-2-[4-(5-fluoropyridin-2-yl)phenyl]propan-2-olIC5017.0 [1]
1-[5-(2,2-Dimethylpropyl)-1H-imidazol-2-yl]-2-(4-pyrazol-1-ylphenyl)propan-2-olIC505.0 [1]
2-[4-(2,2-Dimethylpropyl)-1H-imidazol-2-yl]-1-[4-(5-fluoropyridin-2-yl)phenyl]propan-2-olIC5082.0 [1]
7,8-Dimethyl-6-(4-propan-2-ylphenyl)sulfonyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepineIC501.6 [1]
2-[3-[1-[6-[4-(Trifluoromethoxy)phenyl]sulfonyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-7-yl]cyclobutyl]-1,2,4-oxadiazol-5-yl]propan-2-olIC500.6 [1]
2-Methyl-2-[6-[4-(trifluoromethoxy)phenyl]sulfonyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-7-yl]propanamideIC500.5 [1]
2-[3-[2-(Trifluoromethyl)-6-[4-(trifluoromethyl)phenyl]sulfonyl-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-7-yl]-1,2,4-oxadiazol-5-yl]propan-2-olIC508.3 [1]
2-[3-[6-(4-Propan-2-ylphenyl)sulfonyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-7-yl]-1,2,4-oxadiazol-5-yl]propan-2-olIC501.7 [1]
Universal ligandIC501.1 [1]
(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-Amino-1-oxohexan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-[[(2R)-2-amino-3-phenylpropanoyl]amino]pentanediamideKi0.36 [1]
5-[[2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]phenoxy]methyl]-1,2-dihydro-1,2,4-triazole-3-thioneIC506.1 [1]
2-(4-(2-(4-(Cyclopentylmethyl)-1H-imidazol-2-yl)ethyl)phenyl)pyridineIC50177.0 [1]
3-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]pyridineIC507.5 [1]
4-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]pyridineIC50101.0 [1]
6-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]-1H-pyridin-2-oneIC5051.0 [1]
6-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]pyridin-2-amineIC507.3 [1]
6-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]pyridine-2-carbonitrileIC50140.0 [1]
5-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]-1,2-thiazoleIC5011.0 [1]
4-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]thiadiazoleIC5045.0 [1]
4-(4-(2-(4-(2,2-Dimethylbutyl)-1H-imidazol-2-yl)ethyl)phenyl)isothiazoleIC5010.0 [1]
2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]pyrazineIC5051.0 [1]
1-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]-1,2,4-triazoleIC50340.0 [1]
1-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]triazoleIC50390.0 [1]
2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]tetrazoleIC50205.0 [1]
1-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]piperidineIC5028.0 [1]
2-[4-[2-[5-(Cyclohexylmethyl)-1H-imidazol-2-yl]ethyl]phenyl]-4,5-difluorobenzoic acidIC5036.0 [1]
3-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]pyridine-2-carboxylic acidIC50560.0 [1]
6-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]pyridine-2-carboxylic acidIC502821.0 [1]
5-[2-[4-[2-[5-(Cyclopentylmethyl)-1H-imidazol-2-yl]ethyl]phenyl]phenyl]-2H-tetrazoleIC5015.0 [1]
2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]phenolIC5031.0 [1]
5-[2-[4-[2-[4-(Cyclopentylmethyl)-2H-imidazol-2-yl]ethyl]phenyl]phenyl]-1,3-thiazolidine-2,4-dioneIC50287.0 [1]
2-[2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]phenoxy]acetic acidIC50103.0 [1]
3-(4'-{2-[4-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl}biphenyl-2-yloxymethyl)-4H-[1,2,4]triazoleIC5022.0 [1]
5-[[2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]phenoxy]methyl]-1H-1,2,4-triazol-3-amineIC5027.0 [1]
5-[[2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]phenoxy]methyl]-3-(trifluoromethyl)-1H-1,2,4-triazoleIC50127.0 [1]
4-[[2-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]phenoxy]methyl]-2H-triazoleIC5083.0 [1]
3-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]-5,6-dihydrobenzo[d][2]benzazepin-7-oneIC5010.0 [1]
3-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]-6-methyl-5H-benzo[d][2]benzazepin-7-oneIC5020.0 [1]
(R)-1-(4-(2-(4-(2,2-Dimethylbutyl)-1H-imidazol-2-yl)ethyl)phenyl)piperidine-2-carboxylic acidIC505.3 [1]
(2R)-1-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]-2-(2H-tetrazol-5-yl)piperidineIC506.2 [1]
(2R)-1-[4-[2-[5-(2,2-Dimethylbutyl)-1H-imidazol-2-yl]ethyl]phenyl]-2-(1H-1,2,4-triazol-5-yl)piperidineIC5026.0 [1]
1-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3-tert-butylureaIC5068.0 [1]
1-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3-(2-methylbutan-2-yl)ureaIC5075.0 [1]
1-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3-(2,4,4-trimethylpentan-2-yl)ureaIC50530.0 [1]
1-Tert-butyl-3-[4-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonylureaIC50300.0 [1]
1-[4-[[(3R)-1-Azabicyclo[2.2.2]octan-3-yl]amino]pyridin-3-yl]sulfonyl-3-tert-butylureaIC5010000.0 [1]
1-Tert-butyl-3-[4-(2-phenylpropan-2-ylamino)pyridin-3-yl]sulfonylureaIC503000.0 [1]
1-[4-[[(1R,2S,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3-tert-butylureaIC50230.0 [1]
1-(1-Adamantyl)-3-[4-[[(1R,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonylureaIC50310.0 [1]
1-[2-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]phenyl]sulfonyl-3-tert-butylureaIC506200.0 [1]
1-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-2-tert-butylguanidineIC509700.0 [1]
4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]-N-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)pyridine-3-sulfonamideIC50770.0 [1]
4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]-N-(4-tert-butyl-1,3-thiazol-2-yl)pyridine-3-sulfonamideIC502500.0 [1]
4-(2-Bicyclo[2.2.1]heptanylamino)-N-(5-cyclobutyl-1H-1,2,4-triazol-3-yl)pyridine-3-sulfonamideIC50310.0 [1]
1-Tert-butyl-3-[4-(2,3-dihydro-1H-inden-1-ylamino)pyridin-3-yl]sulfonylureaIC503800.0 [1]
1-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3-tert-butyl-1-methylureaIC506700.0 [1]
4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]-N-(3-tert-butylphenyl)pyridine-3-sulfonamideIC50520.0 [1]
4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]-N-(5-tert-butyl-1H-pyrazol-3-yl)pyridine-3-sulfonamideIC50250.0 [1]
4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]-N-(5-cyclobutyl-1H-1,2,4-triazol-3-yl)pyridine-3-sulfonamideIC50290.0 [1]
1-[4-[[(1S,2S,4R)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3-tert-butylureaIC50630.0 [1]
1-Tert-butyl-3-[4-(pyrrolidin-1-ylamino)pyridin-3-yl]sulfonylureaIC5010000.0 [1]
N-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-3,3-dimethylbutanamideIC5010000.0 [1]
Tert-butyl N-[4-[[(1R,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonylcarbamateIC5010000.0 [1]
1-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]oxy]pyridin-3-yl]sulfonyl-3-tert-butylureaIC50990.0 [1]
3-[4-[[(1R,2R,4S)-2-Bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonyl-1-tert-butyl-1-methylureaIC50650.0 [1]
1-Tert-butyl-3-[4-[[(1R,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]pyridin-3-yl]sulfonylureaIC50660.0 [1]
1-[4-(Benzylamino)pyridin-3-yl]sulfonyl-3-tert-butylureaIC5010000.0 [1]
1-[4-[[(1S,2R,4R)-2-Bicyclo[2.2.1]heptanyl]oxy]pyridin-3-yl]sulfonyl-3-tert-butylureaIC50880.0 [1]
1-Tert-butyl-3-[4-(cyclohexylamino)pyridin-3-yl]sulfonylureaIC50400.0 [1]
10-(4-Tert-butylphenyl)sulfonyl-13-methyl-5-(trifluoromethyl)-2,4,10,12-tetrazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaeneIC505.3 [1]
7,8-Dimethyl-2-(trifluoromethyl)-6-[4-(trifluoromethyl)phenyl]sulfonyl-5,11-dihydropyrido[3,2-c][1,5]benzodiazepineIC506.8 [1]
6-(4-Tert-butylphenyl)sulfonyl-2,7,8-trimethyl-5,11-dihydropyrido[3,2-c][1,5]benzodiazepineIC5010.0 [1]
6-(4-Tert-butylphenyl)sulfonyl-7,8-dimethyl-5,11-dihydropyrido[3,2-c][1,5]benzodiazepineIC5040.0 [1]
7,8-Dimethyl-2-(trifluoromethyl)-6-[5-(trifluoromethyl)thiophen-3-yl]sulfonyl-5,11-dihydropyrido[3,2-c][1,5]benzodiazepineIC5014.0 [1]
4-Tert-butyl-2-[[7,8-dimethyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-6-yl]sulfonyl]-1,3-thiazoleIC5020.0 [1]
6-(4-Tert-butylphenyl)sulfonyl-7,8-dimethyl-5,11-dihydropyrido[3,2-c][1,5]benzodiazepine-2-carbonitrileIC504.4 [1]
10-(4-Tert-butylphenyl)sulfonyl-5-(trifluoromethyl)-2,4,10,16-tetrazatetracyclo[9.8.0.03,8.012,17]nonadeca-1(11),3(8),4,6,12(17),13,15,18-octaeneIC500.7 [1]
7,8-Dimethyl-6-[4-(trifluoromethoxy)phenyl]sulfonyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepineIC503.3 [1]
6-(4-Tert-butylphenyl)sulfonyl-2-chloro-7,8-dimethyl-5,11-dihydropyrido[3,2-c][1,5]benzodiazepineIC501.2 [1]
6-(4-Tert-butylphenyl)sulfonyl-2-chloro-3-fluoro-7,8-dimethyl-5,11-dihydropyrido[3,2-c][1,5]benzodiazepineIC508.9 [1]
N-Methyl-1-[6-[4-(trifluoromethoxy)phenyl]sulfonyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-7-yl]cyclobutane-1-carboxamideIC502.1 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Bombesin receptor subtype-3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/bombesin-receptor-subtype-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Bombesin receptor subtype-3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bombesin-receptor-subtype-3-inhibitors-ic50-ki.
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