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Bone morphogenetic protein 1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(R)-5-(6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl)-1,2,4-oxadiazole-3-carboxamideIC5026.0 [1], 44.0 [2]
(2R)-N-[(2S)-3,3-Dimethyl-1-oxo-1-[[(1R)-1-phenylethyl]amino]butan-2-yl]-N'-hydroxy-2-(3-phenylpropyl)butanediamideIC508765.0 [1]
(2R)-2-(3-Cyclohexylpropyl)-N-[(2S)-3,3-dimethyl-1-oxo-1-[[(1R)-1-phenylethyl]amino]butan-2-yl]-N'-hydroxybutanediamideIC50820.0 [1]
(R)-Ethyl 5-(6-cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl)-1,2,4-oxadiazole-3-carboxylateIC5036.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl)amino]-methyl}-1,2,4-oxadiazol-5-yl)hexanamideIC5011.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl)amino]-methyl}-1,2,4-oxadiazol-5-yl)hexanamideKi11.0 [1]
Benzyl N-[(4R)-4-[1,3-benzodioxol-5-ylmethyl-(4-methoxyphenyl)sulfonylamino]-5-(hydroxyamino)-5-oxopentyl]carbamateIC509.0 [1]
(2-Chlorophenyl)methyl N-[(4R)-4-[1,3-benzodioxol-5-ylmethyl-(4-methoxyphenyl)sulfonylamino]-5-(hydroxyamino)-5-oxopentyl]carbamateIC503.9 [1]
(2-Bromophenyl)methyl N-[(4R)-4-[1,3-benzodioxol-5-ylmethyl-(4-methoxyphenyl)sulfonylamino]-5-(hydroxyamino)-5-oxopentyl]carbamateIC5024.0 [1]
N-[(4R)-4-[1,3-Benzodioxol-5-ylmethyl-(4-methoxyphenyl)sulfonylamino]-5-(hydroxyamino)-5-oxopentyl]benzamideIC5098.0 [1]
N-[(4R)-4-[1,3-Benzodioxol-5-ylmethyl-(4-methoxyphenyl)sulfonylamino]-5-(hydroxyamino)-5-oxopentyl]benzamideKi100.0 [1]
Ethyl 5-[(3R)-1-(hydroxyamino)-1-oxo-6-phenylhexan-3-yl]-1,2,4-oxadiazole-3-carboxylateIC506600.0 [1]
5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-N,N-dimethyl-1,2,4-oxadiazole-3-carboxamideIC509.3 [1], 10.0 [2]
Ethyl 4-[(4R)-4-[1,3-benzodioxol-5-ylmethyl-(4-methoxy-2,3,6-trimethylphenyl)sulfonylamino]-5-(hydroxyamino)-5-oxopentanoyl]piperazine-1-carboxylateKi43.0 [1]
[3-Ethoxy-5-[5-[[[(2R)-2-[(1R)-1-[formyl(hydroxy)amino]propyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]phenyl]phosphonic acidIC501.0 [1]
[3-Ethoxy-5-[5-[[[(2R)-2-[(1R)-1-[formyl(hydroxy)amino]propyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]phenyl]phosphonic acidKi0.04 [1]
(2S)-2-[[2-Ethoxy-4-[5-[[[(2R)-2-[(1R)-1-[formyl(hydroxy)amino]propyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]benzoyl]amino]butanedioic acidIC501.0 [1]
(2S)-2-[[2-Ethoxy-4-[5-[[[(2R)-2-[(1R)-1-[formyl(hydroxy)amino]propyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]benzoyl]amino]butanedioic acidKi0.01 [1]
(S)-2-(4-Methoxyphenylsulfonylamino)-5-[3-[(R)-alpha-methylbenzyl]ureido]pentanehydroximic acidIC50110.0 [1]
3-[[4-(Benzylcarbamoylamino)phenyl]sulfonyl-[2-(4-methoxyphenyl)ethyl]amino]-N-hydroxypropanamideIC5010.0 [1], 1000.0 [2]
(2R)-N-Hydroxy-2-[(4-methoxyphenyl)sulfonyl-(pyridin-3-ylmethyl)amino]-3-methylbutanamide;hydrochlorideIC503000.0 [1]
CID 10370504IC5052000.0 [1]
2-[Benzyl-(4-methoxyphenyl)sulfonylamino]-N-hydroxyacetamideIC5016000.0 [1]
2-[Phenethyl[(4-methoxyphenyl)sulfonyl]amino]acetohydroximic acidIC5018000.0 [1]
2-[(4-Methoxybenzyl)[(4-methoxyphenyl)sulfonyl]amino]acetohydroximic acidIC5029000.0 [1]
2-[[2-(Hydroxyamino)-2-oxoethyl]-(4-methoxyphenyl)sulfonylamino]acetic acidIC50345000.0 [1]
2-[Butan-2-yl-(4-methoxyphenyl)sulfonylamino]-N-hydroxyacetamideIC50112000.0 [1]
2-[(4-Chlorobenzyl)[(4-methoxyphenyl)sulfonyl]amino]acetohydroximic acidIC5019000.0 [1]
2-(5-{(1R)-4-Cyclohexyl-1-[2-(hydroxyamino)-2-oxoethyl]butyl}-1,2,4-oxadiazol-3-yl)isonicotinic acidIC506.0 [1]
CID 44274134IC500.2 [1]
N-[[[(2R)-2-[[Formyl(hydroxy)amino]methyl]heptanoyl]amino]methyl]-7-methoxy-1-benzofuran-2-carboxamideIC50160.0 [1]
Methyl 4-[[(2R)-2-[1,3-benzodioxol-5-ylmethyl-(4-methoxyphenyl)sulfonylamino]-3-(hydroxyamino)-3-oxopropyl]carbamoyl]benzoateKi7.0 [1]
Benzyl 4-[(4R)-4-[1,3-benzodioxol-5-ylmethyl-(4-methoxy-2,3,6-trimethylphenyl)sulfonylamino]-5-(hydroxyamino)-5-oxopentanoyl]piperazine-1-carboxylateKi100.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(3-pyridinyl)-1,2,4-oxadiazol-5-yl]hexanamideIC5023.0 [1]
(3R)-3-[3-[(Tert-butylamino)methyl]-1,2,4-oxadiazol-5-yl]-6-cyclohexyl-N-hydroxyhexanamideIC5010.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]hexanamideIC5030.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-[(sulfamoylamino)methyl]-1,2,4-oxadiazol-5-yl]hexanamideIC5098.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(piperidine-1-carbonyl)-1,2,4-oxadiazol-5-yl]hexanamideIC5026.0 [1]
2-[5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-1,2,4-oxadiazol-3-yl]pyridine-4-carboxamideIC5017.0 [1]
(3R)-6-Cyclohexyl-3-[3-[(1,1-dioxo-1,2-thiazolidin-2-yl)methyl]-1,2,4-oxadiazol-5-yl]-N-hydroxyhexanamideIC5015.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-(3-{[(isopropylsulfonyl)amino]methyl}-1,2,4-oxadiazol-5-yl)hexanamideIC5021.0 [1]
5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-N-(4-methoxyphenyl)sulfonyl-1,2,4-oxadiazole-3-carboxamideIC5017.0 [1]
(3R)-6-Cyclohexyl-3-[3-[(cyclopropylamino)methyl]-1,2,4-oxadiazol-5-yl]-N-hydroxyhexanamideIC506.0 [1]
(R)-2-(6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl)-N,N-dimethyloxazole-4-carboxamideIC5045.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(2-pyridinyl)-1,2,4-oxadiazol-5-yl]hexanamideIC5025.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(2-pyrimidinyl)-1,2,4-oxadiazol-5-yl]hexanamideIC5023.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(4-morpholinylmethyl)-1,2,4-oxadiazol-5-yl]hexanamideIC505.0 [1]
N-Benzyl-5-[(3R)-6-cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-1,2,4-oxadiazole-3-carboxamideIC5057.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(5-pyrimidinyl)-1,2,4-oxadiazol-5-yl]hexanamideIC5014.0 [1]
(3R)-3-[3-[[Acetyl(methyl)amino]methyl]-1,2,4-oxadiazol-5-yl]-6-cyclohexyl-N-hydroxyhexanamideIC503.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(2-pyridinylmethyl)-1,2,4-oxadiazol-5-yl]hexanamideIC506.0 [1]
2-[5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-1,2,4-oxadiazol-3-yl]-N,N-dimethylpyridine-4-carboxamideIC5017.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-[(1H-pyrazol-4-ylsulfonylamino)methyl]-1,2,4-oxadiazol-5-yl]hexanamideIC5088.0 [1]
5-[5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-1,2,4-oxadiazol-3-yl]pyridine-3-carboxylic acidIC5017.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-[[methyl(methylsulfonyl)amino]methyl]-1,2,4-oxadiazol-5-yl]hexanamideIC5038.0 [1]
2-[5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-1,2,4-oxadiazol-3-yl]-N-methylpyridine-4-carboxamideIC5030.0 [1]
N-Benzyl-5-[(3R)-6-cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-N-methyl-1,2,4-oxadiazole-3-carboxamideIC5065.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-[(pyridin-3-ylsulfonylamino)methyl]-1,2,4-oxadiazol-5-yl]hexanamideIC5026.0 [1]
5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-N-(4-fluorophenyl)sulfonyl-1,2,4-oxadiazole-3-carboxamideIC5033.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-(3-{[(phenylsulfonyl)amino]methyl}-1,2,4-oxadiazol-5-yl)hexanamideIC5026.0 [1]
5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-N-(4-methylphenyl)sulfonyl-1,2,4-oxadiazole-3-carboxamideIC5014.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-(morpholine-4-carbonyl)-1,2,4-oxadiazol-5-yl]hexanamideIC5025.0 [1]
N-[(2R)-2-[1,3-Benzodioxol-5-ylmethyl-(4-methoxyphenyl)sulfonylamino]-3-(hydroxyamino)-3-oxopropyl]benzamideKi14.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-{3-[(isopropylamino)methyl]-1,2,4-oxadiazol-5-yl}hexanamideIC5029.0 [1]
(3R)-3-[3-[(Cyclobutylamino)methyl]-1,2,4-oxadiazol-5-yl]-6-cyclohexyl-N-hydroxyhexanamideIC506.0 [1]
(R)-2-(6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl)-N,N,5-trimethyloxazole-4-carboxamideIC5017.0 [1]
(R)-5-(6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl)-N-propyl-1,2,4-oxadiazole-3-carboxamideIC5032.0 [1]
(R)-6-Cyclohexyl-N-hydroxy-3-(3-(pyrrolidine-1-carbonyl)-1,2,4-oxadiazol-5-yl)hexanamideIC5043.0 [1]
(R)-2-(5-(6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl)-1,2,4-oxadiazole-3-carboxamido)acetic acidIC5021.0 [1]
(3R)-6-Cyclohexyl-3-[3-[(ethylsulfonylamino)methyl]-1,2,4-oxadiazol-5-yl]-N-hydroxyhexanamideIC5026.0 [1]
5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-N-(pyridin-2-ylmethyl)-1,2,4-oxadiazole-3-carboxamideIC5037.0 [1]
5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-N-(3,4-dimethoxyphenyl)sulfonyl-1,2,4-oxadiazole-3-carboxamideIC501.8 [1]
(3R)-3-[3-[(Carbamoylamino)methyl]-1,2,4-oxadiazol-5-yl]-6-cyclohexyl-N-hydroxyhexanamideIC50324.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-[[(1-hydroxy-2-methylpropan-2-yl)amino]methyl]-1,2,4-oxadiazol-5-yl]hexanamideIC508.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-[(4-hydroxypiperidin-1-yl)methyl]-1,2,4-oxadiazol-5-yl]hexanamideIC5013.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-[3-[(pyridin-2-ylsulfonylamino)methyl]-1,2,4-oxadiazol-5-yl]hexanamideIC50107.0 [1]
Benzyl N-[(2S)-2-[[(2S,3S)-2-[(3,4-dibromophenyl)sulfonylamino]-3-methylpentanoyl]amino]-3-(hydroxyamino)-3-oxopropyl]carbamateIC5026.0 [1]
3-[[4-(Dibenzylcarbamoylamino)phenyl]sulfonyl-[2-(4-methoxyphenyl)ethyl]amino]-N-hydroxypropanamideIC50380.0 [1]
[2-Ethoxy-4-[5-[[[(2R)-2-[(1R)-1-[formyl(hydroxy)amino]propyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]phenyl]phosphonic acidIC501.0 [1]
N-[[[(2R)-2-[(1R)-1-[Formyl(hydroxy)amino]propyl]heptanoyl]amino]methyl]-5-phenylfuran-2-carboxamideIC5032.0 [1]
3-Ethoxy-5-[5-[[[(2R)-2-[(1R)-1-[formyl(hydroxy)amino]propyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]benzoic acidIC501.0 [1]
5-(3-Ethoxyphenyl)-N-[[[(2R)-2-[[formyl(hydroxy)amino]methyl]heptanoyl]amino]methyl]furan-2-carboxamideIC501.0 [1]
(2S)-2-[[3-Ethoxy-5-[5-[[[(2R)-2-[(1R)-1-[formyl(hydroxy)amino]propyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]benzoyl]amino]butanedioic acidIC501.0 [1]
N-[[[(2R)-2-[[Formyl(hydroxy)amino]methyl]heptanoyl]amino]methyl]-5-(3-methoxyphenyl)furan-2-carboxamideIC5020.0 [1]
4-[5-[[[(2R)-2-[[Formyl(hydroxy)amino]methyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]benzoic acidIC501.0 [1]
3-[5-[[[(2R)-2-[[Formyl(hydroxy)amino]methyl]heptanoyl]amino]methylcarbamoyl]furan-2-yl]benzoic acidIC508.0 [1]
N-[[[(2R)-2-[[Formyl(hydroxy)amino]methyl]heptanoyl]amino]methyl]-5-phenylfuran-2-carboxamideIC5025.0 [1]
3-[[4-[(4-Chlorophenyl)carbamoylamino]phenyl]sulfonyl-[2-(4-methoxyphenyl)ethyl]amino]-N-hydroxypropanamideIC50300.0 [1]
(3R)-6-Cyclohexyl-3-[3-(2,4-dioxo-1H-pyrimidin-5-yl)-1,2,4-oxadiazol-5-yl]-N-hydroxyhexanamideIC5010.0 [1]
N-[[[(2S)-2-[[Formyl(hydroxy)amino]methyl]heptanoyl]amino]methyl]-7-methoxy-1-benzofuran-2-carboxamideIC504000.0 [1]
CID 135712681IC5039.0 [1]
N-[[[(2R)-2-[[Formyl(hydroxy)amino]methyl]pentanoyl]amino]methyl]-7-methoxy-1-benzofuran-2-carboxamideIC501250.0 [1]
N-[[[(2R)-2-[(1S)-1-[Formyl(hydroxy)amino]propyl]heptanoyl]amino]methyl]-7-methoxy-1-benzofuran-2-carboxamideIC5010000.0 [1]
N-[[[(2R)-2-Benzyl-3-[formyl(hydroxy)amino]propanoyl]amino]methyl]-7-methoxy-1-benzofuran-2-carboxamideIC50160.0 [1]
N-[[3-[Formyl(hydroxy)amino]propanoylamino]methyl]-7-methoxy-1-benzofuran-2-carboxamideIC506300.0 [1]
N-[[[(2R)-2-[(1R)-1-[Formyl(hydroxy)amino]propyl]heptanoyl]amino]methyl]-7-methoxy-1-benzofuran-2-carboxamideIC50126.0 [1]
Benzyl N-[(2S)-2-[[(2S,3S)-2-[(4-chloro-2,5-dimethylphenyl)sulfonylamino]-3-methylpentanoyl]amino]-3-(hydroxyamino)-3-oxopropyl]carbamateIC5067.0 [1]
(3R)-6-Cyclohexyl-N-hydroxy-3-(3-phenyl-1,2,4-oxadiazol-5-yl)hexanamideIC50116.0 [1]
Ethyl 4-[5-[(3R)-6-cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-1,2,4-oxadiazol-3-yl]benzoateIC50154.0 [1]
4-[5-[(3R)-6-Cyclohexyl-1-(hydroxyamino)-1-oxohexan-3-yl]-1,2,4-oxadiazol-3-yl]benzoic acidIC5032.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Bone morphogenetic protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/bone-morphogenetic-protein-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Bone morphogenetic protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bone-morphogenetic-protein-1-inhibitors-ic50-ki.
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