Bromodomain adjacent to zinc finger domain protein 2A Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic Acid	IC50	31622.78 [1]
	1-(7-(2-Methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanone	IC50	400.0 [1]
	4-(4-(1-Methyl-1H-pyrazol-4-yl)-1-(2-(1-methyl-1H-pyrazol-4-yl)ethyl)-1H-imidazol-5-yl)benzonitrile	IC50	130.0 [1]
	4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	100000.0 [1]
	4-{1-[2-(4-Methyl-1h-1,2,3-Triazol-1-Yl)ethyl]-4-Phenyl-1h-Imidazol-5-Yl}benzonitrile	IC50	51000.0 [1]
	1-[1-(Pyridin-2-Yl)indolizin-3-Yl]ethan-1-One	IC50	1500.0 [1]
	N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamide	IC50	10000.0 [1]
	1-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-3-methyl-2,5,6,7-tetrahydropyrrolo[3,4-c]pyridin-4-one	IC50	10000.0 [1]
	4-[5-(1-Methylpyrazol-4-yl)-3-[2-(4-methyltriazol-1-yl)ethyl]imidazol-4-yl]benzonitrile	IC50	600.0 [1]
	4-[3-[2-(4-Methyltriazol-1-yl)ethyl]-5-pyridin-4-ylimidazol-4-yl]benzonitrile	IC50	4000.0 [1]
	4-[3-[2-(4-Methyltriazol-1-yl)ethyl]-5-pyridin-3-ylimidazol-4-yl]benzonitrile	IC50	50000.0 [1]
	4-[3-[2-(4-Methyltriazol-1-yl)ethyl]-5-(1,3-thiazol-5-yl)imidazol-4-yl]benzonitrile	IC50	7800.0 [1]
	4-[5-(3-Methyl-1,2-oxazol-5-yl)-3-[2-(4-methyltriazol-1-yl)ethyl]imidazol-4-yl]benzonitrile	IC50	50000.0 [1]
	4-[3-[2-(4-Methyltriazol-1-yl)ethyl]imidazol-4-yl]benzonitrile	IC50	50000.0 [1]
	4-[3-Methyl-5-(1-methylpyrazol-4-yl)imidazol-4-yl]benzonitrile	IC50	50000.0 [1]
	3-Fluoro-4-[5-(1-methylpyrazol-4-yl)-3-[(4-methyltriazol-1-yl)methyl]imidazol-4-yl]benzonitrile	IC50	1010.0 [1]
	2-Fluoro-4-[5-(1-methylpyrazol-4-yl)-3-[(4-methyltriazol-1-yl)methyl]imidazol-4-yl]benzonitrile	IC50	450.0 [1]
	4-Methyl-1-[[4-(1-methylpyrazol-4-yl)-5-(4-nitrophenyl)imidazol-1-yl]methyl]triazole	IC50	1380.0 [1]
	3-(3-Acetylindolizin-1-yl)benzamide	IC50	1800.0 [1]
	1-[1-[2-(Hydroxymethyl)phenyl]indolizin-3-yl]ethanone	IC50	1800.0 [1]
	1-[1-[4-(Hydroxymethyl)phenyl]indolizin-3-yl]ethanone	IC50	1200.0 [1]
	1-[1-[4-(Dimethylamino)phenyl]indolizin-3-yl]ethanone	IC50	1100.0 [1]
	1-[1-(2-Methylsulfonylphenyl)indolizin-3-yl]ethanone	IC50	720.0 [1]
	1-[1-[2-(Hydroxymethyl)phenyl]-7-methylindolizin-3-yl]ethanone	IC50	1000.0 [1]
	1-[1-[2-(Hydroxymethyl)phenyl]-7-methoxyindolizin-3-yl]ethanone	IC50	1200.0 [1]
	1-[1-[2-(Hydroxymethyl)phenyl]-7-morpholin-4-ylindolizin-3-yl]ethanone	IC50	1700.0 [1]
	3-Acetyl-1-[2-(hydroxymethyl)phenyl]indolizine-7-carboxamide	IC50	4100.0 [1]
	1-[7-Methoxy-1-(2-methylsulfonylphenyl)indolizin-3-yl]ethanone	IC50	580.0 [1]
	1-[1-(3-Methoxyphenyl)indolizin-3-yl]ethanone	IC50	30000.0 [1]
	1-[1-(2-Hydroxyphenyl)indolizin-3-yl]ethanone	IC50	7200.0 [1]
	1-[1-(3-Hydroxyphenyl)indolizin-3-yl]ethanone	IC50	3300.0 [1]
	1-[7-Methyl-1-(2-methylsulfonylphenyl)indolizin-3-yl]ethanone	IC50	890.0 [1]
	1-[1-[2-(Hydroxymethyl)-4-methoxyphenyl]indolizin-3-yl]ethanone	IC50	1400.0 [1]
	Tert-butyl N-[[3-acetyl-1-(2-methylsulfonylphenyl)indolizin-7-yl]methyl]carbamate	IC50	160.0 [1]
	1-(1-Thiophen-2-ylindolizin-3-yl)ethanone	IC50	8600.0 [1]
	1-{1-[2-(Hydroxymethyl)phenyl]-7-Phenoxyindolizin-3-Yl}ethanone	IC50	4100.0 [1]
	1-{1-[2-(Methylsulfonyl)phenyl]-7-Phenoxyindolizin-3-Yl}ethanone	IC50	550.0 [1]
	3-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-1-methyl-6H-pyrrolo[2,3-c]pyridin-7-one	IC50	10000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 38 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Bromodomain adjacent to zinc finger domain protein 2A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 26 Apr. 2024, https://www.aatbio.com/data-sets/bromodomain-adjacent-to-zinc-finger-domain-protein-2a-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, April 26). Quest Database™ Bromodomain adjacent to zinc finger domain protein 2A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bromodomain-adjacent-to-zinc-finger-domain-protein-2a-inhibitors-ic50-ki.
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