Bromodomain and PHD finger-containing protein 3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	4-Cyano-N-(1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	260.0 [1], 2000.0 [2]
	CID 122705990	IC50	2450.0 [1], 5550.0 [2]
	CID 91827373	IC50	140.0 [1], 1010.0 [2]
	4-Cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	1000.0 [1]
	N-(1-Methyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	7600.0 [1]
	4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	100000.0 [1]
	6-(3-Hydroxypropyl)-2-(1-methyl-2-oxo-3H-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dione	IC50	20000.0 [1]
	4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic Acid	IC50	1.0 [1]
	CID 40642506	IC50	5110.0 [1]
	CID 15990224	IC50	100000.0 [1]
	N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamide	IC50	15848.93 [1]
	4-Bromo-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-one	Ki	100.0 [1]
	3,4-Dimethoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzenesulfonamide	IC50	7000.0 [1]
	N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamide	IC50	10000.0 [1]
	1-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-3-methyl-2,5,6,7-tetrahydropyrrolo[3,4-c]pyridin-4-one	IC50	10000.0 [1]
	4-Cyano-2-methoxy-N-(7-methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	190.0 [1]
	3-Chloro-4-cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	2300.0 [1]
	4-Cyano-N-(8-fluoro-1,3-dimethyl-2-oxoquinolin-6-yl)-2-methoxybenzenesulfonamide	IC50	10000.0 [1]
	4-Cyano-N-(7-methoxy-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	2200.0 [1]
	N-(7-Methoxy-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	2200.0 [1]
	N-(4-Cyanophenyl)-1-methyl-2-oxoquinoline-6-sulfonamide	IC50	2200.0 [1]
	4-Cyano-N-(7-methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	280.0 [1]
	N-(7-Methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamide	IC50	590.0 [1]
	4-Cyano-N-(7-Methoxy-1,4-Dimethyl-2-Oxo-1,2-Dihydroquinolin-6-Yl)benzene-1-Sulfonamide	IC50	9300.0 [1]
	8-[[(3R,4R)-3-[(1,1-Dioxothian-4-yl)methoxy]-1-methylpiperidin-4-yl]amino]-3-methyl-5-(5-methylpyridin-3-yl)-1H-1,7-naphthyridin-2-one	Ki	794.33 [1]
	4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)-2-methoxybenzenesulfonamide	IC50	4600.0 [1]
	4-Cyano-2-methoxy-N-(1-methyl-2-oxo-3-propan-2-ylquinolin-6-yl)benzenesulfonamide	IC50	4600.0 [1]
	1-Methyl-2-oxo-N-phenylquinoline-6-sulfonamide	IC50	100000.0 [1]
	4-Cyano-N-(1-methyl-2-oxo-3-propan-2-ylquinolin-6-yl)benzenesulfonamide	IC50	16000.0 [1]
	N-(1,3-Dimethyl-2-oxo-7-pyrrolidin-1-ylquinolin-6-yl)-2-methoxybenzamide	IC50	12000.0 [1]
	3-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-1-methyl-6H-pyrrolo[2,3-c]pyridin-7-one	IC50	10000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 31 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Bromodomain and PHD finger-containing protein 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/bromodomain-and-phd-finger-containing-protein-3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Bromodomain and PHD finger-containing protein 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bromodomain-and-phd-finger-containing-protein-3-inhibitors-ic50-ki.
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