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Bromodomain-containing protein 1 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
CID 122705990IC506.0 [1], 67.0 [2], 97.0 [3], 825.0 [4]
6-(3-Hydroxypropyl)-2-(1-methyl-2-oxo-3H-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5010000.0 [1], 20000.0 [2]
4-Cyano-N-(1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5048.0 [1], 760.0 [2]
CID 91827373IC5046.0 [1], 619.0 [2]
4-Cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50200.0 [1]
3-Cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50270.0 [1]
2-Cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC501700.0 [1]
N-(1-Methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC501400.0 [1]
4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50100000.0 [1]
N-(1,3-Dimethyl-2-oxoquinolin-6-yl)-2-methoxybenzenesulfonamideIC50130.0 [1]
2-(1,3,6-Trimethyl-2-Oxidanylidene-Benzimidazol-5-Yl)benzo[de]isoquinoline-1,3-DioneIC5094.0 [1], 740.0 [2]
2-(6-Methoxy-1,3-dimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC50115.0 [1], 1500.0 [2]
6-(4-Hydroxypiperidin-1-yl)-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5066.0 [1], 2120.0 [2]
6-(4-Methylpiperazin-1-yl)-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5093.0 [1], 1240.0 [2]
6-Piperidin-1-yl-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5095.0 [1], 10000.0 [2]
6-[Methyl(2-pyrrolidin-1-ylethyl)amino]-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5084.0 [1], 941.0 [2]
6-Morpholin-4-yl-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5061.0 [1], 613.0 [2]
6-[4-(Cyclopropylmethyl)piperazin-1-yl]-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5080.0 [1], 863.0 [2]
6-[4-[2-(Dimethylamino)ethyl]piperazin-1-yl]-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5074.0 [1], 420.0 [2]
6-Chloro-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5037.0 [1], 675.0 [2]
6-(4-Methoxypiperidin-1-yl)-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5053.0 [1], 915.0 [2]
6-Pyrrolidin-1-yl-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC50126.0 [1], 10000.0 [2]
4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic AcidIC5019952.62 [1]
CID 40642506IC501110.0 [1]
N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-5,6,7,8-tetrahydro-2-naphthalenesulfonamideIC502050.0 [1]
CID 15990224IC507943.28 [1]
CID 35397514IC501200.0 [1]
N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamideIC507943.28 [1]
N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-N-ethyl-2-methoxybenzamideIC5050118.72 [1]
N-[6-(4-Methoxyphenoxy)-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1h-Benzimidazol-5-Yl]benzenesulfonamideIC502770.0 [1]
3,4-Dimethoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzenesulfonamideIC501750.0 [1]
N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamideIC501000.0 [1]
1-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-3-methyl-2,5,6,7-tetrahydropyrrolo[3,4-c]pyridin-4-oneIC501000.0 [1]
4-Cyano-N-methyl-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC506700.0 [1]
4-Cyano-2-methoxy-N-(7-methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5080.0 [1]
3-Chloro-4-cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50450.0 [1]
4-Cyano-N-(8-fluoro-1,3-dimethyl-2-oxoquinolin-6-yl)-2-methoxybenzenesulfonamideIC50510.0 [1]
3,4-Dichloro-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50230.0 [1]
4-Cyano-N-(7-methoxy-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50520.0 [1]
N-(7-Methoxy-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50380.0 [1]
N-(4-Cyanophenyl)-1-methyl-2-oxoquinoline-6-sulfonamideIC50150.0 [1]
4-Cyano-N-(7-methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50100.0 [1]
N-(7-Methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50190.0 [1]
4-Cyano-N-(7-Methoxy-1,4-Dimethyl-2-Oxo-1,2-Dihydroquinolin-6-Yl)benzene-1-SulfonamideIC501800.0 [1]
4-Cyano-N-(1,4-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50150.0 [1]
8-[[(3R,4R)-3-[(1,1-Dioxothian-4-yl)methoxy]-1-methylpiperidin-4-yl]amino]-3-methyl-5-(5-methylpyridin-3-yl)-1H-1,7-naphthyridin-2-oneKi398.11 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,2-dimethyl-3,4-dihydrochromene-6-sulfonamideIC502460.0 [1]
(2S)-N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,3-dimethoxy-2,3-dimethyl-1,4-benzodioxine-6-sulfonamideIC5010000.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-3,4-dihydro-2H-chromene-6-sulfonamideIC501600.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-2-methylbenzenesulfonamideIC501700.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3-methoxybenzenesulfonamideIC501990.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-5,6,7,8-tetrahydronaphthalene-2-sulfonamideIC502670.0 [1]
5-Bromo-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC50124.0 [1]
6-(Propylamino)-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC50121.0 [1]
2-[1,3-Dimethyl-6-(4-methylpiperazin-1-yl)-2-oxobenzimidazol-5-yl]benzo[de]isoquinoline-1,3-dioneIC50366.0 [1]
2-(6-Bromo-1,3-dimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC50153.0 [1]
6-Bromo-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5051.0 [1]
5-Hydroxy-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC50102.0 [1]
1,3-Dioxo-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-5-carbonitrileIC50248.0 [1]
5-Nitro-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5082.0 [1]
6-(4-Hydroxybutyl)-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5070.0 [1]
5-Amino-2-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5063.0 [1]
4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)-2-methoxybenzenesulfonamideIC504400.0 [1]
4-Cyano-2-methoxy-N-(1-methyl-2-oxo-3-propan-2-ylquinolin-6-yl)benzenesulfonamideIC503300.0 [1]
2-[6-(Dimethylamino)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzo[de]isoquinoline-1,3-dioneIC50100.0 [1]
1-Methyl-2-oxo-N-phenylquinoline-6-sulfonamideIC507800.0 [1]
4-Cyano-N-(1-methyl-2-oxo-3-propan-2-ylquinolin-6-yl)benzenesulfonamideIC5014000.0 [1]
N-(1,3-Dimethyl-2-oxo-7-pyrrolidin-1-ylquinolin-6-yl)-2-methoxybenzamideIC502600.0 [1]
2-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC50450.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-3-fluoro-4-methylbenzenesulfonamideIC506140.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-4-propan-2-ylbenzenesulfonamideIC504300.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,3-dihydro-1H-indene-5-sulfonamideIC501710.0 [1]
4-Chloro-N-(1,3-dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)benzenesulfonamideIC503470.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3,4-dimethoxybenzenesulfonamideIC501210.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3,4-dimethylbenzenesulfonamideIC505160.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-4-methoxybenzenesulfonamideIC501330.0 [1]
N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-2-methylbenzenesulfonamideIC502380.0 [1]
N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-4-propoxybenzenesulfonamideIC5010000.0 [1]
4-Chloro-N-(1,3-dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-2-methylbenzenesulfonamideIC502390.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-5-fluoro-2-methylbenzenesulfonamideIC502420.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3-fluoro-4-methylbenzenesulfonamideIC503690.0 [1]
N-[6-(4-Methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]-4-methylbenzenesulfonamideIC5010000.0 [1]
4-Methoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzenesulfonamideIC503580.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxy-2,3-dihydro-1H-benzimidazol-5-yl)-4-methylbenzenesulfonamideIC502920.0 [1]
Items per page: 1 - 10 of 84
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References

This online tool may be cited as follows

MLA

"Quest Database™ Bromodomain-containing protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/bromodomain-containing-protein-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Bromodomain-containing protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bromodomain-containing-protein-1-inhibitors-ic50-ki.
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