Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Tert-butyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate | IC50 | 39.1 [1], 56.7 [2], 69.0 [3], 81.0 [4] | |
| Tert-butyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate | Ki | 6.6 [1], 8.9 [2] | |
| Molibresib | IC50 | 42.4 [1], 160.0 [2], 390.0 [3], 400.0 [4] | |
| Molibresib | Ki | 30.3 [1], 53.9 [2] | |
| Birabresib | IC50 | 21.0 [1], 38.5 [2], 92.0 [3] | |
MLA | "Quest Database™ Bromodomain-containing protein 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 13 Dec. 2025, https://www.aatbio.com/data-sets/bromodomain-containing-protein-3-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 13). Quest Database™ Bromodomain-containing protein 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bromodomain-containing-protein-3-inhibitors-ic50-ki. | |
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