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Bromodomain-containing protein 3 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Tert-butyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetateIC5039.1 [1], 56.7 [2], 69.0 [3], 81.0 [4]
Tert-butyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetateKi6.6 [1], 8.9 [2]
MolibresibIC5042.4 [1], 160.0 [2], 390.0 [3], 400.0 [4]
MolibresibKi30.3 [1], 53.9 [2]
BirabresibIC5021.0 [1], 38.5 [2], 92.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseBromodomain-containing protein 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Dec2025https://www.aatbio.com/data-sets/bromodomain-containing-protein-3-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 13). Quest DatabaseBromodomain-containing protein 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bromodomain-containing-protein-3-inhibitors-ic50-ki.
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