Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Tert-butyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate | IC50 | 77.0 [1] | |
| Tert-butyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate | Ki | 12.0 [1], 14.9 [2] | |
| Molibresib | IC50 | 120.0 [1] | |
| Molibresib | Ki | 23.0 [1], 32.3 [2], 38.8 [3], 46.4 [4] | |
| Apabetalone | IC50 | 1985.0 [1] | |
MLA | "Quest Database™ Bromodomain-containing protein 4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 13 Dec. 2025, https://www.aatbio.com/data-sets/bromodomain-containing-protein-4-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 13). Quest Database™ Bromodomain-containing protein 4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bromodomain-containing-protein-4-inhibitors-ic50-ki. | |
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