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Bromodomain testis-specific protein Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Tert-butyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetateIC50103.0 [1], 183.0 [2], 217.0 [3]
4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic AcidIC5050.12 [1], 31622.78 [2]
BET Inhibitor C3IC502300.0 [1], 5200.0 [2]
BET Inhibitor C3Ki450.0 [1]
BI-2536IC50260.0 [1], 1400.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseBromodomain testis-specific protein Inhibitors (IC50, Ki)." AAT Bioquest, Inc.14 Dec2025https://www.aatbio.com/data-sets/bromodomain-testis-specific-protein-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 14). Quest DatabaseBromodomain testis-specific protein Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bromodomain-testis-specific-protein-inhibitors-ic50-ki.
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