Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| 4-Amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide | IC50 | 12.59 [1] | |
| N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamide | IC50 | 0.4 [1], 1.0 [2], 1.26 [3], 10.0 [4], 25.12 [5], 3162.28 [6] | |
| 4-Amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-4-(2-nitroimidazol-1-yl)-1-oxobutan-2-yl]benzenesulfonamide | IC50 | 53.0 [1], 251.19 [2], 690.0 [3], 794.33 [4] | |
| 4-Amino-3,5-dichloro-N-[(2S)-1-(4-methylpiperidin-1-yl)-1-oxo-4-phenylbutan-2-yl]benzenesulfonamide | IC50 | 10000.0 [1] | |
| N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-6-sulfonamide | IC50 | 7.94 [1], 15.85 [2] | |
MLA | "Quest Database™ C-C chemokine receptor type 10 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 7 Feb. 2026, https://www.aatbio.com/data-sets/c-c-chemokine-receptor-type-10-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2026, February 7). Quest Database™ C-C chemokine receptor type 10 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/c-c-chemokine-receptor-type-10-inhibitors-ic50-ki. | |
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