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C-C chemokine receptor type 4 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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N-Cycloheptyl-6,7-dimethoxy-2-(4-pyrrolidine-1-ylpiperidine-1-yl)quinazolin-4-amineIC50200.0 [1]
N-[5-Bromo-3-[[3-[2-(dimethylamino)ethoxy]-4-methoxyphenyl]methoxy]pyrazin-2-yl]-4-methylbenzenesulfonamideIC503.89 [1]
N-[5-Bromo-3-[[3-[2-(dimethylamino)ethoxy]-4-methoxyphenyl]methoxy]pyrazin-2-yl]-4-methylbenzenesulfonamideKi3.16 [1]
[4-[4-[(2,4-Dichlorophenyl)methylamino]pyrimidin-2-yl]piperazin-1-yl]-[(2R)-piperidin-2-yl]methanoneIC507.94 [1], 10.0 [2], 50.0 [3], 380.0 [4]
[4-[4-[(2,4-Dichlorophenyl)methylamino]pyrimidin-2-yl]piperazin-1-yl]-[(2R)-piperidin-2-yl]methanoneKi2.51 [1]
[4-[4-[(2,4-Dichlorophenyl)methylamino]pyrido[2,3-d]pyrimidin-2-yl]piperazin-1-yl]-[(2R)-piperidin-2-yl]methanoneIC505.5 [1]
[4-[4-[(2,4-Dichlorophenyl)methylamino]pyrido[2,3-d]pyrimidin-2-yl]piperazin-1-yl]-[(2R)-piperidin-2-yl]methanoneKi0.79 [1]
CID 25141301IC5024.0 [1], 110.0 [2], 150.0 [3]
SporanoxIC50200.0 [1], 501.19 [2], 7943.28 [3], 12589.25 [4]
CCR4 AntagonistIC5018.0 [1], 73.0 [2], 140.0 [3]
2,3-Dichloro-N-(3-methoxypyrazin-2-yl)benzenesulfonamideIC5015.85 [1], 31.62 [2], 501.19 [3]
CID 23585443IC502.51 [1], 3.98 [2], 158.49 [3], 316.23 [4]
QuercetinIC5010000.0 [1], 31622.78 [2]
CID 46861584IC5014.79 [1], 39.81 [2]
CID 46861584Ki10.0 [1]
N-[[3-[[3-[(5-Chlorothiophen-2-yl)sulfonylamino]-4-methoxyindazol-1-yl]methyl]phenyl]methyl]acetamideIC5031.62 [1]
N-[[3-[[3-[(5-Chlorothiophen-2-yl)sulfonylamino]-4-methoxyindazol-1-yl]methyl]phenyl]methyl]acetamideKi12.59 [1]
4-((Bis(cyclohexylmethyl)amino)methyl)-N-(naphthalen-1-yl)thiazol-2-amineIC5018.0 [1], 31.0 [2], 530.0 [3]
(2S)-1-(5-Chloronaphthalen-2-yl)sulfonyl-N-methyl-N-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-2-carboxamideKi100.0 [1], 150.0 [2], 500.0 [3]
[4-[4-[(2,4-Dichlorophenyl)methylamino]pyrido[2,3-d]pyrimidin-2-yl]piperazin-1-yl]-[(2S)-piperidin-2-yl]methanoneIC503.0 [1], 7.0 [2], 20.0 [3]
4-Methyl-N-(naphthalen-1-yl)thiazol-2-amineIC501700.0 [1], 3000.0 [2], 6400.0 [3]
3-(4-Hydroxy-2,6-diiodophenyl)-3-(4-hydroxy-3,5-diiodophenyl)-2-benzofuran-1-oneIC501600.0 [1], 3981.07 [2], 10000.0 [3]
N4-(2,4-Dichlorobenzyl)-N2-(4-(diethylamino)pentyl)pyrimidine-2,4-diamineIC50280.0 [1], 800.0 [2], 5000.0 [3]
N-(5-Bromo-3-methoxypyrazin-2-yl)-5-chlorothiophene-2-sulfonamideIC5063.1 [1], 199.53 [2]
2,3-Dichloro-N-(4-methoxy-1-methylindazol-3-yl)benzenesulfonamideIC50602.56 [1]
[1-[1-[4-(4-Chloroanilino)-6,7-dimethoxyquinazolin-2-yl]piperidin-4-yl]piperidin-3-yl]methanolIC5019.0 [1], 23.0 [2]
N-[(3-Chloro-2-methylphenyl)methyl]-2-[(2R,5R)-2-(2,4-dichlorophenyl)-4-oxo-3-[2-oxo-2-(3-piperidin-1-ylpropylamino)ethyl]-1,3-thiazolidin-5-yl]acetamideIC50140.0 [1]
4-N-[(2,4-Dichlorophenyl)methyl]-2-N-[5-(diethylamino)pentan-2-yl]pyrimidine-2,4-diamineIC50270.0 [1], 5000.0 [2]
N-[(2,4-Dichlorophenyl)methyl]-2-[2-(pyrrolidin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-8-yl]pyrimidin-4-amineIC507.94 [1]
N-[(2,4-Dichlorophenyl)methyl]-2-[2-(pyrrolidin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-8-yl]pyrimidin-4-amineKi1.58 [1]
N-[(2,4-Difluorophenyl)methyl]-2-[2-(pyrrolidin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-8-yl]pyrimidin-4-amineIC507.94 [1]
N-[(2,4-Difluorophenyl)methyl]-2-[2-(pyrrolidin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-8-yl]pyrimidin-4-amineKi3.16 [1]
N-[(2,4-Dichlorophenyl)methyl]-N-methyl-2-[2-(pyrrolidin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-8-yl]pyrimidin-4-amineIC507.94 [1]
N-[(2,4-Dichlorophenyl)methyl]-N-methyl-2-[2-(pyrrolidin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-8-yl]pyrimidin-4-amineKi1.0 [1]
[1-[1-[4-(Cycloheptylamino)-6,7-dimethoxyquinazolin-2-yl]piperidin-4-yl]piperidin-3-yl]methanolIC5030.0 [1], 100.0 [2]
N-Cycloheptyl-2-[4-(dimethylamino)piperidine-1-yl]-6,7-dimethoxyquinazolin-4-amineIC50260.0 [1], 730.0 [2]
N-Cycloheptyl-2-(4-isopropylpiperazine-1-yl)-6,7-dimethoxyquinazolin-4-amineIC50220.0 [1], 660.0 [2]
N-Cyclohexyl-6,7-dimethoxy-2-(4-pyrrolidin-1-ylpiperidin-1-yl)quinazolin-4-amineIC50480.0 [1], 1900.0 [2]
N-Cyclooctyl-6,7-dimethoxy-2-(4-pyrrolidin-1-ylpiperidin-1-yl)quinazolin-4-amineIC50200.0 [1], 1200.0 [2]
CID 44562155IC5025.0 [1], 69.0 [2]
CID 44562156IC50220.0 [1], 510.0 [2]
CID 44562189IC5031.0 [1], 320.0 [2]
3-[[1-[4-(4-Chloroanilino)-6,7-dimethoxyquinazolin-2-yl]piperidin-4-yl]-methylamino]propan-1-olIC5043.0 [1], 280.0 [2]
4-[[1-[4-(4-Chloroanilino)-6,7-dimethoxyquinazolin-2-yl]piperidin-4-yl]-methylamino]butan-1-olIC5061.0 [1], 360.0 [2]
1-[1-[4-(4-Chloroanilino)-6,7-dimethoxyquinazolin-2-yl]piperidin-4-yl]piperidin-3-olIC5048.0 [1], 85.0 [2]
N-(4-Chlorophenyl)-6,7-dimethoxy-2-[4-(3-methoxypiperidin-1-yl)piperidin-1-yl]quinazolin-4-amineIC50100.0 [1], 510.0 [2]
N-(4-Chlorophenyl)-6,7-dimethoxy-2-[4-[3-(methoxymethyl)piperidin-1-yl]piperidin-1-yl]quinazolin-4-amineIC5052.0 [1], 64.0 [2]
[4-[1-[4-(4-Chloroanilino)-6,7-dimethoxyquinazolin-2-yl]piperidin-4-yl]morpholin-2-yl]methanolIC50100.0 [1], 620.0 [2]
[1-[1-[4-[(4-Chlorophenyl)methylamino]-6,7-dimethoxyquinazolin-2-yl]piperidin-4-yl]piperidin-3-yl]methanolIC5087.0 [1], 450.0 [2]
3-[[3-[(5-Chlorothiophen-2-yl)sulfonylamino]-4-methoxyindazol-1-yl]methyl]-N,N-dimethylbenzamideIC50416.87 [1]
3-[[3-[(5-Chlorothiophen-2-yl)sulfonylamino]-4-methoxyindazol-1-yl]methyl]-N,N-dimethylbenzamideKi1258.93 [1]
5-Chloro-N-[1-[(3,4-dimethoxyphenyl)methyl]-4-methoxyindazol-3-yl]thiophene-2-sulfonamideIC5022.91 [1]
5-Chloro-N-[1-[(3,4-dimethoxyphenyl)methyl]-4-methoxyindazol-3-yl]thiophene-2-sulfonamideKi19.95 [1]
3-{[3-{[(5-Chloro-2-thienyl)sulfonyl]amino}-4-(methyloxy)-1H-indazol-1-yl]methyl}-N-methylbenzamideIC5079.43 [1]
3-{[3-{[(5-Chloro-2-thienyl)sulfonyl]amino}-4-(methyloxy)-1H-indazol-1-yl]methyl}-N-methylbenzamideKi316.23 [1]
N-[1-[[3-(Aminomethyl)phenyl]methyl]-4-methoxyindazol-3-yl]-5-chlorothiophene-2-sulfonamideIC5091.2 [1]
N-[1-[[3-(Aminomethyl)phenyl]methyl]-4-methoxyindazol-3-yl]-5-chlorothiophene-2-sulfonamideKi100.0 [1]
5-Chloro-N-[4-methoxy-1-[(3-methoxyphenyl)methyl]indazol-3-yl]thiophene-2-sulfonamideIC50158.49 [1]
5-Chloro-N-[4-methoxy-1-[(3-methoxyphenyl)methyl]indazol-3-yl]thiophene-2-sulfonamideKi125.89 [1]
3-{[3-{[(5-Chloro-2-thienyl)sulfonyl]amino}-4-(methyloxy)-1H-indazol-1-yl]methyl}benzamideIC5054.95 [1]
3-{[3-{[(5-Chloro-2-thienyl)sulfonyl]amino}-4-(methyloxy)-1H-indazol-1-yl]methyl}benzamideKi39.81 [1]
N-[[3-[[3-[(5-Chlorothiophen-2-yl)sulfonylamino]-4-methoxyindazol-1-yl]methyl]phenyl]methyl]-2-hydroxyacetamideIC5027.54 [1]
N-[[3-[[3-[(5-Chlorothiophen-2-yl)sulfonylamino]-4-methoxyindazol-1-yl]methyl]phenyl]methyl]-2-hydroxyacetamideKi15.85 [1]
N-[[3-[[3-[(5-Chlorothiophen-2-yl)sulfonylamino]-4-methoxyindazol-1-yl]methyl]phenyl]methyl]-2-hydroxypropanamideIC5012.59 [1]
N-[[3-[[3-[(5-Chlorothiophen-2-yl)sulfonylamino]-4-methoxyindazol-1-yl]methyl]phenyl]methyl]-2-hydroxypropanamideKi7.94 [1]
5-Chloro-N-[1-[[2-(hydroxymethyl)phenyl]methyl]-4-methoxyindazol-3-yl]thiophene-2-sulfonamideIC50323.59 [1]
5-Chloro-N-[1-[[2-(hydroxymethyl)phenyl]methyl]-4-methoxyindazol-3-yl]thiophene-2-sulfonamideKi251.19 [1]
5-Chloro-N-[1-[[3-(hydroxymethyl)phenyl]methyl]-4-methoxyindazol-3-yl]thiophene-2-sulfonamideIC5032.36 [1]
5-Chloro-N-[1-[[3-(hydroxymethyl)phenyl]methyl]-4-methoxyindazol-3-yl]thiophene-2-sulfonamideKi39.81 [1]
N-(1-Benzyl-4-methoxyindazol-3-yl)-5-chlorothiophene-2-sulfonamideIC50389.05 [1]
N-(1-Benzyl-4-methoxyindazol-3-yl)-5-chlorothiophene-2-sulfonamideKi251.19 [1]
5-Chloro-N-[1-[[4-(hydroxymethyl)phenyl]methyl]-4-methoxyindazol-3-yl]thiophene-2-sulfonamideIC5047.86 [1]
5-Chloro-N-[1-[[4-(hydroxymethyl)phenyl]methyl]-4-methoxyindazol-3-yl]thiophene-2-sulfonamideKi50.12 [1]
AmiodaroneKi11405.0 [1]
DisulfiramKi4397.0 [1]
ClotrimazoleIC501600.0 [1]
(S)-N1-((1H-Benzo[d]imidazol-2-yl)methyl)-N1-(5,6,7,8-tetrahydroquinolin-8-yl)butane-1,4-diamineIC5010000.0 [1]
CenicrivirocIC501100.0 [1]
TAK-779 cationIC5010000.0 [1]
N-[(2S)-2-(3-Chlorophenyl)-4-(1-oxospiro[2H-1-benzothiophene-3,4'-piperidine]-1'-yl)butyl]-N-methylbenzenesulfonamideIC5010000.0 [1]
5,7-Dihydroxy-4-methyl-3-(4-methylpiperazin-1-yl)-2H-chromen-2-oneIC5021.2 [1]
Benzyl N-ethyl-N-[1-[4-[(4R)-4-(1H-indol-3-ylmethyl)-2,5-dioxoimidazolidin-1-yl]-3-phenylbutyl]piperidin-4-yl]carbamateIC501000.0 [1]
Benzyl N-[1-[4-[(4R)-4-(1H-indol-3-ylmethyl)-2,5-dioxoimidazolidin-1-yl]-3-phenylbutyl]piperidin-4-yl]-N-prop-2-enylcarbamateIC501000.0 [1]
Benzyl N-[1-[4-[(4R)-4-(1H-indol-3-ylmethyl)-2,5-dioxoimidazolidin-1-yl]-3-methyl-3-phenylbutyl]piperidin-4-yl]-N-prop-2-enylcarbamateIC501000.0 [1]
J-113863 Cation, trans-IC5010000.0 [1]
1-(1,3-Dimethyl-1H-pyrazolo[3,4-b]pyridine-5-carbonyl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)ureaIC5010000.0 [1]
(2S)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-2-(2-piperidin-1-ylethylamino)-2-thiophen-3-ylacetamideIC502000.0 [1]
Isothiourea-1aIC503000.0 [1]
5-Butyl-9-[1-(4,6-dimethylpyrimidine-5-carbonyl)-4-methylpiperidin-4-yl]-3-[(4-ethoxycyclohexyl)methyl]-3,9-diazaspiro[5.5]undecan-4-oneIC5050000.0 [1]
PharmaGSID_48521IC5050000.0 [1]
5,7-Dihydroxy-4-methyl-3-(piperazin-1-yl)-2H-chromen-2-oneIC504360.0 [1]
5,7-Dihydroxy-4-methyl-3-[4-[(E)-3-phenylprop-2-enoyl]piperazin-1-yl]chromen-2-oneIC501570.0 [1]
5,7-Dihydroxy-4-methyl-3-(4-prop-2-enoylpiperazin-1-yl)chromen-2-oneIC504240.0 [1]
3-[4-(2-Chloroacetyl)piperazin-1-yl]-5,7-dihydroxy-4-methylchromen-2-oneIC508580.0 [1]
3-(4-Benzoylpiperazin-1-yl)-5,7-dihydroxy-4-methylchromen-2-oneIC504360.0 [1]
3-[4-(Benzenesulfonyl)piperazin-1-yl]-5,7-dihydroxy-4-methylchromen-2-oneIC506040.0 [1]
N-[4-[4-(5,7-Dihydroxy-4-methyl-2-oxochromen-3-yl)piperazin-1-yl]sulfonylphenyl]acetamideIC502560.0 [1]
4-(5,7-Dihydroxy-4-methyl-2-oxochromen-3-yl)-N-(4-propan-2-ylphenyl)piperazine-1-carboxamideIC501320.0 [1]
4-(5,7-Dihydroxy-4-methyl-2-oxochromen-3-yl)-N-heptylpiperazine-1-carboxamideIC50539.0 [1]
4-(5,7-Dihydroxy-4-methyl-2-oxochromen-3-yl)-N-(2-phenoxyphenyl)piperazine-1-carboxamideIC506000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ C-C chemokine receptor type 4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/c-c-chemokine-receptor-type-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ C-C chemokine receptor type 4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/c-c-chemokine-receptor-type-4-inhibitors-ic50-ki.
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