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C-C chemokine receptor type 8 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(5R)-3-[1-(1H-Indol-2-ylmethyl)piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-oneIC5019.95 [1], 100.0 [2], 501.19 [3]
(4-Chlorophenyl)-[9-[(2-phenoxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]methanoneIC5081.28 [1]
3-[2-(2-Methoxyphenoxy)benzyl]-9-(1-oxidoisonicotinoyl)-3,9-diazaspiro[5.5]undecaneIC50114.82 [1]
[9-[[3-(2-Methoxyphenoxy)phenyl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-(1-oxidopyridin-1-ium-4-yl)methanoneIC5032.36 [1], 33.11 [2]
[9-[(3-Phenoxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-pyrimidin-4-ylmethanoneIC5027.54 [1]
[9-[(3-Phenoxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-pyridin-4-ylmethanoneIC5017.38 [1], 18.2 [2]
(4-Chlorophenyl)-[9-[(3-phenoxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]methanoneIC5019.05 [1]
[9-[[2-(2-Methoxyphenoxy)phenyl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-pyridin-4-ylmethanoneIC5011.48 [1], 12.02 [2]
(4-Chlorophenyl)-[9-[[2-(2-methoxyphenoxy)phenyl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]methanoneIC5034.67 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamideIC500.3 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamideKi0.3 [1]
1-Ethyl-N-[1-[[3-(2-methoxyphenoxy)phenyl]methyl]piperidin-4-yl]-4-phenylpiperidine-4-carboxamideIC5056.0 [1]
1-Ethyl-N-[1-[[3-(2-methoxyphenoxy)phenyl]methyl]piperidin-4-yl]-4-phenylpiperidine-4-carboxamideKi11.0 [1]
N-[1-[[3-(2-Chlorophenoxy)phenyl]methyl]piperidin-4-yl]-1-ethyl-4-phenylpiperidine-4-carboxamideIC5043.0 [1]
N-[1-[[3-(2-Chlorophenoxy)phenyl]methyl]piperidin-4-yl]-1-ethyl-4-phenylpiperidine-4-carboxamideKi15.0 [1]
N-[1-[[3-(2-Methoxyphenoxy)phenyl]methyl]piperidin-4-yl]-4-phenylpiperidine-4-carboxamideIC5011.0 [1]
N-[1-[[3-(2-Methoxyphenoxy)phenyl]methyl]piperidin-4-yl]-4-phenylpiperidine-4-carboxamideKi62.0 [1]
N-{1-[3-(2-Methoxy-phenoxy)-benzyl]-piperidin-4-yl}-2-phenyl-acetamideIC5055.0 [1]
N-{1-[3-(2-Methoxy-phenoxy)-benzyl]-piperidin-4-yl}-2-phenyl-acetamideKi250.0 [1]
2-[3-[[1-[[3-(2-Chlorophenoxy)phenyl]methyl]piperidin-4-yl]carbamoyl]-3-phenylpyrrolidin-1-yl]-2-methylpropanoic acidIC501.0 [1]
2-[3-[[1-[[3-(2-Chlorophenoxy)phenyl]methyl]piperidin-4-yl]carbamoyl]-3-phenylpyrrolidin-1-yl]-2-methylpropanoic acidKi6.0 [1]
N-[1-[[3-(2-Chlorophenoxy)phenyl]methyl]piperidin-4-yl]-3-phenylpyrrolidine-3-carboxamideIC5022.0 [1]
N-[1-[[3-(2-Chlorophenoxy)phenyl]methyl]piperidin-4-yl]-3-phenylpyrrolidine-3-carboxamideKi27.0 [1]
2-[4-[[1-[[3-(2-Chlorophenoxy)phenyl]methyl]piperidin-4-yl]carbamoyl]-4-phenylpiperidin-1-yl]-2-methylpropanoic acidIC504.0 [1]
2-[4-[[1-[[3-(2-Chlorophenoxy)phenyl]methyl]piperidin-4-yl]carbamoyl]-4-phenylpiperidin-1-yl]-2-methylpropanoic acidKi9.0 [1]
N-[4-(4-Methoxy-phenylsulfamoyl)-naphthalen-1-yl]-benzamideIC50150.0 [1]
N-[4-(4-Methoxy-phenylsulfamoyl)-naphthalen-1-yl]-benzamideKi42.6 [1]
CID 46861584IC5010000.0 [1]
Ethyl 1-(3-phenoxybenzyl)-4-piperidinecarboxylateKi2600.0 [1]
(2S)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-2-(2-piperidin-1-ylethylamino)-2-thiophen-3-ylacetamideIC501000.0 [1]
3-[1-[(3,4-Dimethylphenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-oneIC5039.81 [1]
5-(6-Methoxyquinolin-4-yl)-3-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]-1,3-oxazolidin-2-oneIC501258.93 [1]
2-Methyl-N-{4-[({1-[(2S)-pyrrolidin-2-ylcarbonyl]piperidin-4-yl}amino)sulfonyl]-1-naphthyl}benzamideKi1.0 [1]
1-[4-Chloro-2-hydroxy-3-[(3S)-3-methyloxolan-3-yl]sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]ureaIC5010000.0 [1]
N-{4-[1-(2-Amino-acetyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamideKi4.1 [1]
3-[1-[(4-Bromophenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-oneIC5050.12 [1]
3-[1-[(4-Chlorophenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-oneIC50630.96 [1]
4-(4-Benzoylamino-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl esterKi0.17 [1]
4-(4-o-Tolylcarbamoyl-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl esterKi5.21 [1]
3-(1-Hexylpiperidin-4-yl)-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-oneIC50501.19 [1]
5-(6-Methoxyquinolin-4-yl)-3-[1-[(1-methylindol-2-yl)methyl]piperidin-4-yl]-1,3-oxazolidin-2-oneIC503162.28 [1]
3-[1-(1-Benzothiophen-2-ylmethyl)piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-oneIC50794.33 [1]
5-(6-Methoxyquinolin-4-yl)-3-[1-(3-phenylpropyl)piperidin-4-yl]-1,3-oxazolidin-2-oneIC50251.19 [1]
3-[1-(1H-Indol-2-ylmethyl)piperidin-4-yl]-5-(6-methoxy-1,5-naphthyridin-4-yl)-1,3-oxazolidin-2-oneIC5031.62 [1]
3-[1-[(3,4-Dichlorophenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-oneIC50125.89 [1]
N-[4-(Morpholin-4-ylsulfonyl)naphthyl]benzamideKi7745.0 [1]
N-[4-(4-Methyl-piperazine-1-sulfonyl)-naphthalen-1-yl]benzamideKi30000.0 [1]
N-[4-(Piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-benzamideKi578.0 [1]
N-{4-[(Benzylamino)sulfonyl]-1-naphthyl}benzamideKi233.1 [1]
4-(4-Cyclohexylcarbamoyl-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl esterKi9.5 [1]
N-{4-[(Pyridin-4-ylmethyl)-sulfamoyl]-naphthalen-1-yl}-benzamideKi3277.0 [1]
N-(4-Cyclohexylsulfamoyl-naphthalen-1-yl)-benzamideKi4.4 [1]
N-[1-(3-Phenoxy-benzyl)-piperidin-4-yl]-2-phenyl-acetamideKi1400.0 [1]
N-Ethyl-1-[(3-phenoxyphenyl)methyl]piperidine-4-carboxamideKi9100.0 [1]
1-(4-Chlorophenyl)-N-[1-[[3-(2-methoxyphenoxy)phenyl]methyl]piperidin-4-yl]cyclohexane-1-carboxamideKi250.0 [1]
1-[[3-(2-Chlorophenoxy)phenyl]methyl]-4-[(1-ethyl-4-phenylpiperidine-4-carbonyl)amino]piperidine-4-carboxylic acidKi23.0 [1]
N-[1-(3-Phenoxy-benzyl)-piperidin-4-yl]-propionamideKi9200.0 [1]
1-[[3-(2-Methoxyphenoxy)phenyl]methyl]-4-[(4-phenylpiperidine-4-carbonyl)amino]piperidine-4-carboxylic acidKi60.0 [1]
N-Methyl-4-[[4-[(2-methylbenzoyl)amino]naphthalen-1-yl]sulfonylamino]piperidine-1-carboxamideKi0.7 [1]
N-(4-Phenylsulfamoyl-naphthalen-1-yl)-benzamideKi1760.0 [1]
[9-[[3-(2-Methoxyphenoxy)phenyl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-(1-oxidopyridin-1-ium-2-yl)methanoneIC5026.92 [1]
(1-Oxidopyridin-1-ium-4-yl)-[9-[(3-phenoxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]methanoneIC50165.96 [1]
[9-[[2-(2-Methoxyphenoxy)phenyl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-(1-oxidopyridin-1-ium-2-yl)methanoneIC5079.43 [1]
3-[9-[[2-(2-Methoxyphenoxy)phenyl]methyl]-3,9-diazaspiro[5.5]undecane-3-carbonyl]-1H-pyridin-2-oneIC5054.95 [1]
(5-Aminopyridin-2-yl)-[9-[(2,2-dimethyl-3H-1-benzofuran-7-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]methanoneIC502.63 [1]
[9-[(2-Methyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-pyridin-4-ylmethanoneIC50128.82 [1]
[9-(2,3-Dihydro-1-benzofuran-7-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-pyridin-4-ylmethanoneIC501479.11 [1]
[9-[(2,2-Dimethyl-3H-1-benzofuran-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-pyridin-4-ylmethanoneIC5030.9 [1]
(5-Aminopyridin-2-yl)-[9-[(2,2-dimethyl-3H-1-benzofuran-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]methanoneIC508.13 [1]
(2-Aminopyridin-4-yl)-[9-[(2,2-dimethyl-1,3-benzodioxol-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]methanoneIC506.61 [1]
N-[4-(Methyl-phenyl-sulfamoyl)-naphthalen-1-yl]-benzamideKi44000.0 [1]
4-(4-Benzoylamino-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid tert-butyl esterKi15.2 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]methyl}-1-naphthyl)-2-methylbenzamideIC503300.0 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-4-methylbenzamideIC509.5 [1]
N-[4-(1-Butyryl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-2-fluoro-benzamideIC5019.2 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-4-fluorobenzamideIC5059.5 [1]
4-Butyl-N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)benzamideIC5015.3 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-4-pentylbenzamideIC5036.1 [1]
4-(Benzyloxy)-N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)benzamideIC5024.6 [1]
N-[4-[(1-Butanoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]-1-benzothiophene-2-carboxamideIC5023.6 [1]
N-[4-[(1-Butanoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]-5-methyl-2-(trifluoromethyl)furan-3-carboxamideIC5046.9 [1]
N-[4-[(1-Butanoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]-2-chloro-6-methylpyridine-4-carboxamideIC5043.9 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-pyrazine-2-carboxamideIC501004.0 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-pyridine-2-carboxamideIC5041.7 [1]
Ethyl 4-({[4-(Isonicotinoylamino)-1-naphthyl]sulfonyl}amino)-piperidine-1-carboxylateIC50100.0 [1]
N-[4-[(1-Butanoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]cyclobutanecarboxamideIC5057.9 [1]
N-[4-[(1-Butanoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]cyclohexanecarboxamideIC506.1 [1]
N-[4-[(1-Butanoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]-1-methylpiperidine-4-carboxamideIC501900.0 [1]
N-(4-{[(1-Butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-ethylbutanamideIC50638.5 [1]
N-[4-[(1-Butanoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]-3,3-dimethylbutanamideIC50612.5 [1]
4-[4-(2-Methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid ethyl esterKi1.6 [1]
Ethyl 4-(1-hydroxynaphthalene-4-sulfonamido)piperidine-1-carboxylateKi5000.0 [1]
Ethyl 4-({[4-(benzoyloxy)-1-naphthyl]sulfonyl}amino)-piperidine-1-carboxylateKi16.4 [1]
2-Methyl-N-[4-(1-propionyl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-benzamideKi2.5 [1]
N-(4-{[(1-Acetylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamideKi6.7 [1]
N-[4-(1-Cyclopentanecarbonyl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-2-methyl-benzamideKi9.1 [1]
N-{4-[1-(2-Methoxy-acetyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamideKi15.8 [1]
N-{4-[1-(3-Amino-propionyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamideKi11.3 [1]
N-[4-[[1-(5-Aminopentanoyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamideKi199.0 [1]
N-[4-[[1-(Azetidine-3-carbonyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamideKi1.5 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ C-C chemokine receptor type 8 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/c-c-chemokine-receptor-type-8-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ C-C chemokine receptor type 8 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/c-c-chemokine-receptor-type-8-inhibitors-ic50-ki.
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