Calcium release-activated calcium channel protein 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Miconazole	IC50	27000.0 [1], 100000.0 [2]
	Mibefradil	IC50	52100.0 [1], 100000.0 [2]
	Econazole	IC50	17000.0 [1], 94000.0 [2]
	N-[4-(2,5-Dimethoxyphenyl)phenyl]-3-fluoro-N-methylpyridine-4-carboxamide	IC50	26.0 [1], 1300.0 [2]
	1-[2-(4-Methoxyphenyl)-2-[4-(4-methoxyphenyl)butoxy]ethyl]imidazole	IC50	42000.0 [1], 67000.0 [2]
	3,5-Dichloro-2-(2-pyridin-3-yloxyethoxy)benzaldehyde	IC50	100000.0 [1]
	CRAC Channel Inhibitor, BTP2	IC50	2800.0 [1]
	2-(4-Methoxyphenoxy)-1-[4-(4-phenylcyclohexyl)piperazin-1-yl]ethanone	IC50	75000.0 [1]
	4-Chloro-4'-[3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl]benzanilide	IC50	57000.0 [1]
	1-[5-Hydroxy-3-(3-nitrophenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	89000.0 [1]
	2-(4-Chlorophenyl)-1-[5-hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanone	IC50	47000.0 [1]
	2-(3-Chlorophenyl)-1-[5-hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanone	IC50	75000.0 [1]
	1-[5-Hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(4-methoxyphenyl)ethanone	IC50	33000.0 [1]
	1-[5-Hydroxy-5-(trifluoromethyl)-3-[3-(trifluoromethyl)phenyl]-4H-pyrazol-1-yl]-2-phenylethanone	IC50	29000.0 [1]
	1-[3-(2,5-Dichlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	54000.0 [1]
	2-(3-Chlorophenyl)-1-[5-hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanone	IC50	79000.0 [1]
	1-[5-Hydroxy-3-(trifluoromethyl)-5-[2-(trifluoromethyl)phenyl]-4H-pyrazol-1-yl]-2-phenylethanone	IC50	49000.0 [1]
	1-[5-Hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(3-methylphenyl)ethanone	IC50	45000.0 [1]
	2-(2-Chlorophenyl)-1-[5-hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanone	IC50	42000.0 [1]
	1-[5-Hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(3-methylphenyl)ethanone	IC50	42000.0 [1]
	1-[3-(2-Bromophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	30000.0 [1]
	2-(2-Chlorophenyl)-1-[5-hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanone	IC50	40000.0 [1]
	1-[3-(3-Chlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	48000.0 [1]
	1-[5-Hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(3-methoxyphenyl)ethanone	IC50	32000.0 [1]
	1-[3-(2,3-Difluorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	55000.0 [1]
	2-(4-Chlorophenyl)-1-[5-hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanone	IC50	60000.0 [1]
	1-[3-(2-Chlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	33000.0 [1]
	1-[5-Hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	36000.0 [1]
	1-[5-Hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenoxyethanone	IC50	105000.0 [1]
	1-[5-Hydroxy-3-(5,6,7,8-tetrahydronaphthalen-2-yl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	89000.0 [1]
	1-[5-Hydroxy-3-(4-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(2-methylphenyl)ethanone	IC50	55000.0 [1]
	1-[3-(2,4-Dichlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanone	IC50	58000.0 [1]
	1-[5-Hydroxy-3-(4-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(3-methylphenyl)ethanone	IC50	42000.0 [1]
	Chembl4128571	IC50	47000.0 [1]
	N-[6-(Benzimidazol-1-yl)pyridin-3-yl]-3-(dimethylamino)benzamide	IC50	48000.0 [1]
	2-(2-Chloro-6-fluorophenyl)-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1H-pyrrolo[2,3-b]pyridine	IC50	100.0 [1]
	2-(2-Chloro-6-fluorophenyl)-5-(6-methoxy-4-methylpyridin-3-yl)-1H-pyrrolo[2,3-b]pyridine	IC50	104.0 [1]
	2-(2-Chloro-6-fluorophenyl)-5-(4,6-dimethoxypyridin-3-yl)-1H-pyrrolo[2,3-b]pyridine	IC50	440.0 [1]
	(E)-1-[2-[2-(4-Butan-2-ylphenoxy)ethoxy]-3,5-dichlorophenyl]-N-(1,2,4-triazol-4-yl)methanimine	IC50	69900.0 [1]
	N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-2H-benzotriazole-5-carboxamide	IC50	182.5 [1]
	2-(Benzimidazol-1-yl)-N-[4-(3,5-dicyclopropylpyrazol-1-yl)phenyl]acetamide	IC50	383.1 [1]
	2-(Benzotriazol-1-yl)-N-[4-(3,5-dicyclopropylpyrazol-1-yl)phenyl]acetamide	IC50	51.31 [1]
	N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-2-quinolin-6-ylacetamide	IC50	146.7 [1]
	2-(Benzotriazol-1-yl)-N-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]acetamide	IC50	39.17 [1]
	2-(Benzotriazol-2-yl)-N-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]acetamide	IC50	139.0 [1]
	N-[4-(3,5-Dicyclopropylpyrazol-1-yl)-3-fluorophenyl]-2-quinolin-6-ylacetamide	IC50	263.2 [1]
	N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]quinoline-6-carboxamide	IC50	86.12 [1]
	2-(Benzotriazol-1-yl)-N-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]acetamide	IC50	160.5 [1]
	N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]quinoxaline-6-carboxamide	IC50	53.36 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 49 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Calcium release-activated calcium channel protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/calcium-release-activated-calcium-channel-protein-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Calcium release-activated calcium channel protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/calcium-release-activated-calcium-channel-protein-1-inhibitors-ic50-ki.
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