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CaM-kinase kinase beta Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamideKi29700.0 [1]
K252aKi1.8 [1]
N-(2-Guanidinoethyl)-5-isoquinolinesulfonamideKi13000.0 [1]
2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidIC507.94 [1]
Lavendustin cIC50200.0 [1]
(2S,3S)-3-((7-(Benzylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-5-yl)amino)butane-1,2,4-triolIC502450.0 [1]
4-(5-Phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidIC50199.53 [1]
STO-609 acetateIC5010.0 [1]
4-[5-(3-Methylsulfonylphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]benzoic acidIC50125.89 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
Methyl 4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoateIC501258.93 [1]
2-Isobutyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidIC5025.12 [1]
2-Ethyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidIC5019.95 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
4-[[4-Benzyl-6-[(6-ethyl-1,3-benzothiazol-2-yl)amino]pyrimidin-2-yl]amino]cyclohexan-1-olIC50199.53 [1]
N'-Benzyl-N'-[2-[benzyl-[(3-methoxyphenyl)methyl]amino]ethyl]-N,N-dimethylethane-1,2-diamineIC5040400.0 [1]
Chembl4126920IC50398.11 [1]
4-[[4-Cyclopentyloxy-5-(2-methyl-1,3-benzoxazol-6-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-N-methylbenzamideIC50680.0 [1]
Nintedanib impurity EKi15.0 [1]
Melk-IN-1Ki31.0 [1]
2-Hydroxy-3-[N-[4-[methyl-[2-(4-methylpiperazin-1-yl)acetyl]amino]phenyl]-C-phenylcarbonimidoyl]-1H-indole-5-carboxylic acidKi85.0 [1]
5,5-Dimethyl-8-[[4-(2,2,2-trifluoroethylamino)furo[3,2-d]pyrimidin-2-yl]amino]-1H-4,1-benzoxazepin-2-oneIC501910.0 [1]
N-[4-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-N'-hydroxyoctanediamideIC5053.0 [1]
4-[2-[2-Methyl-5-(morpholin-4-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-2-propan-2-ylbenzonitrileIC5012.59 [1]
4-[2-[2-Methyl-4-(2-morpholin-4-ylethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC501.58 [1]
4-[2-[2-Methyl-5-(morpholin-4-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-2-propan-2-ylbenzamideIC5019.95 [1]
4-[2-[2-Methyl-5-(2-morpholin-4-ylethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5031.62 [1]
4-[2-[2-Methyl-3-(2-morpholin-4-ylethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5015.85 [1]
2-Cyclopentyl-4-[5-[2-(trifluoromethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC501995.26 [1]
2-Cyclopentyl-4-(1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidIC5031.62 [1]
4-[2-[2-Methyl-4-(2-morpholin-4-ylethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzonitrileIC50251.19 [1]
4-[2-[3-(Methanesulfonamido)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5012.59 [1]
4-[2-[2-Methyl-3-(morpholin-4-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5012.59 [1]
3-[4-(4-Carbamoylphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-N-[3-(dimethylamino)propyl]benzamideIC5012.59 [1]
4-[2-(2-Methoxyanilino)pyrimidin-4-yl]-2-propan-2-ylbenzamideIC501584.89 [1]
2-Cyclopentyl-4-[5-[2-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC503981.07 [1]
4-[2-(2-Fluoro-5-phenylanilino)pyrimidin-4-yl]benzamideIC5019.95 [1]
4-[2-(2-Methoxyanilino)pyrimidin-4-yl]benzoic acidIC501584.89 [1]
4-[2-(3-Phenylanilino)pyrimidin-4-yl]benzamideIC5025.12 [1]
2-Cyclopentyl-4-[5-(2-hydroxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC50125.89 [1]
4-[2-(2-Methoxyanilino)pyrimidin-4-yl]benzamideIC501258.93 [1]
4-[2-[2-Methyl-5-(morpholin-4-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzonitrileIC50398.11 [1]
4-[5-[2-(Cyanomethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl]-2-cyclopentylbenzamideIC502511.89 [1]
2-Cyclopentyl-4-[5-(2-propan-2-yloxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC501584.89 [1]
2-Cyclopentyl-4-[2-(2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC502.0 [1]
4-[5-Fluoro-2-(2-methoxyanilino)pyrimidin-4-yl]-2-propan-2-ylbenzoic acidIC507.94 [1]
4-[2-(2-Methoxyanilino)pyrimidin-4-yl]-2-propan-2-ylbenzoic acidIC502.0 [1]
4-[2-[4-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5025.12 [1]
2-Cyclopentyl-4-[5-[2-(dimethylamino)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC503981.07 [1]
4-(6-Cyano-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-propan-2-ylbenzoic acidIC50794.33 [1]
4-[5-Chloro-2-(2-methoxyanilino)pyrimidin-4-yl]-2-propan-2-ylbenzamideIC501584.89 [1]
4-[2-[2-Methyl-4-(morpholin-4-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5025.12 [1]
4-(6-Cyano-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-cyclopentylbenzamideIC505.0 [1]
4-[2-[4-(Methanesulfonamido)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5012.59 [1]
2-Cyclopentyl-4-[5-(2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC50199.53 [1]
4-(6-Cyano-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidIC505.0 [1]
4-[2-[2-Methyl-4-(2-morpholin-4-ylethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-2-propan-2-ylbenzamideIC507.94 [1]
5-Phenyl-3-[4-(tetrazol-1-yl)phenyl]-1H-pyrrolo[2,3-b]pyridineIC50398.11 [1]
4-(1H-Pyrrolo[2,3-b]pyridin-3-yl)benzoic acidIC501995.26 [1]
4-[2-[4-[3-(Dimethylamino)propylcarbamoyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5012.59 [1]
4-[2-(3-Phenylanilino)pyrimidin-4-yl]benzoic acidIC50100.0 [1]
4-(6-Carbamoyl-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-cyclopentylbenzoic acidIC505.0 [1]
4-(6-Cyano-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-propan-2-ylbenzamideIC505.0 [1]
4-[2-[2-Methyl-4-(2-morpholin-4-ylethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-2-propan-2-ylbenzonitrileIC506.31 [1]
4-[2-(2-Methoxy-5-phenylanilino)pyrimidin-4-yl]benzamideIC50251.19 [1]
4-[2-(2-Methyl-5-phenylanilino)pyrimidin-4-yl]benzamideIC50501.19 [1]
4-[2-[2-Methyl-5-(morpholin-4-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5015.85 [1]
4-[5-Fluoro-2-(2-methoxyanilino)pyrimidin-4-yl]-2-propan-2-ylbenzamideIC50316.23 [1]
4-[5-(2-Phenoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC50100.0 [1]
4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5031.62 [1]
4-(6-Cyano-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-cyclopentylbenzoic acidIC5015.85 [1]
4-[5-(3-Methylsulfonylphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC50199.53 [1]
2-Cyclopentyl-4-(6-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidIC50630.96 [1]
4-[2-(2-Methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamideIC5019.95 [1]
2-Cyclopentyl-4-[5-(2-phenoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamideIC501584.89 [1]
Chembl4126272IC5050.12 [1]
Chembl4127245IC503.98 [1]
Chembl4128483IC5050.12 [1]
Items per page: 1 - 10 of 78
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References

This online tool may be cited as follows

MLA

"Quest Database™ CaM-kinase kinase beta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/cam-kinase-kinase-beta-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ CaM-kinase kinase beta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cam-kinase-kinase-beta-inhibitors-ic50-ki.
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