Canalicular multispecific organic anion transporter 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Cyclosporin A	IC50	13600.0 [1], 14500.0 [2], 20000.0 [3], 25600.0 [4]
	Cyclosporin A	Ki	4700.0 [1], 8110.0 [2], 21000.0 [3]
	Verlukast	IC50	1000.0 [1], 4000.0 [2], 10000.0 [3], 133000.0 [4]
	Verlukast	Ki	13100.0 [1], 26400.0 [2]
	Sodium	IC50	133000.0 [1]
	Calcium	IC50	133000.0 [1]
	Etoposide	IC50	133000.0 [1]
	Etoposide	Ki	756000.0 [1]
	Verapamil	IC50	133000.0 [1], 200000.0 [2]
	Reserpine	IC50	68400.0 [1]
	Reserpine	Ki	295000.0 [1]
	Simvastatin	IC50	25000.0 [1], 133000.0 [2]
	Probenecid	IC50	133000.0 [1]
	Probenecid	Ki	42200.0 [1]
	Dolutegravir	IC50	90000.0 [1], 100000.0 [2]
	(5S,6R,7E,9E,11Z,14Z)-6-[(2S)-2-[[(4S)-4-Amino-4-carboxybutanoyl]amino]-3-(carboxymethylamino)-3-oxopropyl]sulfanyl-5-hydroxyicosa-7,9,11,14-tetraenoic acid	IC50	150.0 [1], 3300.0 [2]
	Potassium	IC50	133000.0 [1]
	Testosterone	IC50	133000.0 [1]
	Aspirin	IC50	133000.0 [1]
	5-Fluorouracil	IC50	133000.0 [1]
	Doxorubicin	IC50	133000.0 [1]
	Dexamethasone	IC50	133000.0 [1]
	Cyclophosphamide	IC50	133000.0 [1]
	Prednisolone	IC50	133000.0 [1]
	Methotrexate	IC50	133000.0 [1]
	Propranolol	IC50	133000.0 [1]
	Caffeine	IC50	133000.0 [1]
	Warfarin	IC50	133000.0 [1]
	Paclitaxel	IC50	133000.0 [1]
	Acetaminophen	IC50	133000.0 [1]
	Indomethacin	IC50	235000.0 [1]
	Melatonin	IC50	133000.0 [1]
	Cyclosporine	IC50	3100.0 [1]
	Methylprednisolone	IC50	133000.0 [1]
	Lidocaine	IC50	133000.0 [1]
	Nicotine	IC50	133000.0 [1]
	Ciprofloxacin	IC50	133000.0 [1]
	Isoniazid	IC50	133000.0 [1]
	Theophylline	IC50	133000.0 [1]
	Vincristine	Ki	802000.0 [1]
	Tretinoin	IC50	133000.0 [1]
	Vincristine sulfate	IC50	133000.0 [1]
	Metformin	IC50	133000.0 [1]
	Tetracycline	IC50	133000.0 [1]
	Imatinib	IC50	133000.0 [1]
	Tamoxifen	IC50	133000.0 [1]
	Gemcitabine	IC50	133000.0 [1]
	Cytarabine	IC50	133000.0 [1]
	Rifampicin	IC50	53000.0 [1]
	Camptothecin	IC50	133000.0 [1]
	Naloxone	IC50	133000.0 [1]
	Somatostatin	IC50	133000.0 [1]
	Carbamazepine	IC50	133000.0 [1]
	Chlorpromazine	IC50	133000.0 [1]
	Quercetin	IC50	133000.0 [1]
	Levodopa	IC50	133000.0 [1]
	Haloperidol	IC50	133000.0 [1]
	Tacrolimus	IC50	40300.0 [1]
	Amoxicillin	IC50	133000.0 [1]
	Nifedipine	IC50	133000.0 [1]
	Fluoxetine	IC50	133000.0 [1]
	Furosemide	IC50	133000.0 [1]
	Chloroquine	IC50	133000.0 [1]
	Azathioprine	IC50	133000.0 [1]
	Salbutamol	IC50	133000.0 [1]
	Calcitriol	IC50	133000.0 [1]
	Colchicine	IC50	133000.0 [1]
	Erythromycin	IC50	133000.0 [1]
	Clozapine	IC50	133000.0 [1]
	Omeprazole	IC50	133000.0 [1]
	Fluconazole	IC50	133000.0 [1]
	Acyclovir	IC50	133000.0 [1]
	Metronidazole	IC50	133000.0 [1]
	Vinblastine	IC50	21000.0 [1]
	Ketamine	IC50	133000.0 [1]
	Carbon tetrachloride	IC50	133000.0 [1]
	Vincaleukoblastine	IC50	133000.0 [1]
	Risperidone	IC50	133000.0 [1]
	Hydroxyurea	IC50	133000.0 [1]
	Ribavirin	IC50	133000.0 [1]
	Amiodarone	IC50	133000.0 [1]
	Ethinyl estradiol	IC50	133000.0 [1]
	Argipressin	IC50	133000.0 [1]
	Bupivacaine hydrochloride	IC50	133000.0 [1]
	Olanzapine	IC50	133000.0 [1]
	Zidovudine	IC50	133000.0 [1]
	Apomorphine	IC50	133000.0 [1]
	Clarithromycin	IC50	133000.0 [1]
	Staurosporine	IC50	133000.0 [1]
	Docetaxel	IC50	133000.0 [1]
	Allopurinol	IC50	133000.0 [1]
	Ofloxacin	IC50	133000.0 [1]
	Imipramine	IC50	133000.0 [1]
	Dipyridamole	IC50	133000.0 [1]
	Ticlopidine hydrochloride	IC50	133000.0 [1]
	Captopril	IC50	133000.0 [1]
	Quinine	IC50	133000.0 [1]
	Ganciclovir	IC50	133000.0 [1]
	Leucovorin	IC50	133000.0 [1]
	Doxycycline hydrochloride	IC50	133000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Canalicular multispecific organic anion transporter 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/canalicular-multispecific-organic-anion-transporter-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Canalicular multispecific organic anion transporter 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/canalicular-multispecific-organic-anion-transporter-1-inhibitors-ic50-ki.
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