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Cannabinoid CB1 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
RimonabantIC506.0 [1]
RimonabantKi0.43 [1], 1.6 [2], 5.4 [3]
Win 55212-2IC5016.0 [1], 17.0 [2]
Win 55212-2Ki3802.0 [1]
5-(1,1-Dimethylheptyl)-2-[5-hydroxy-2-(3-hydroxypropyl)cyclohexyl]phenolIC500.13 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseCannabinoid CB1 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/cannabinoid-cb1-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseCannabinoid CB1 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cannabinoid-cb1-receptor-inhibitors-ic50-ki.
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