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Carboxypeptidase B2 isoform A Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
(2s)-5-Amino-2-[(1-Propyl-1h-Imidazol-4-Yl)methyl]pentanoic AcidIC50450.0 [1], 5000.0 [2]
(2s)-5-Amino-2-[(1-Propyl-1h-Imidazol-4-Yl)methyl]pentanoic AcidKi10.0 [1], 16.0 [2]
3-Pyridinepropanoic acid, 6-amino-alpha-1H-imidazol-5-yl-IC5035.0 [1], 80.0 [2], 1500.0 [3], 31000.0 [4]
(5r)-5-(3-Aminopropyl)-1-Propyl-4,5,6,7-Tetrahydro-1h-Benzimidazole-5-Carboxylic AcidIC508.0 [1], 76.0 [2], 1000.0 [3]
2-Mercaptomethyl-5-guanidinopentanoic acidIC508.0 [1]
2-Mercaptomethyl-5-guanidinopentanoic acidKi4.0 [1]
3-(6-Aminopyridin-3-yl)-2-[1-(3-methylbutyl)imidazol-4-yl]propanoic acidIC504.0 [1], 5.0 [2]
(2S)-2-(2-Aminoethylamino)-3-(1-propylimidazol-4-yl)propanoic acidKi84.0 [1], 150.0 [2]
(2S)-6-Amino-2-[[(2R)-3-cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]hexanoic acidIC503.0 [1], 7.0 [2]
(2S)-6-Amino-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]hexanoic acid;hydrochlorideIC5051.0 [1], 123.0 [2]
2-[(6-Amino-5-chloropyridin-3-yl)methyl]-3-propanoylselanylpropanoic acidIC501.5 [1], 370000.0 [2]
2-(2-Aminoethylamino)-3-(1-propylimidazol-4-yl)propanoic acidIC50620.0 [1], 8000.0 [2]
Ethyl 7-amino-2-(propanoylselanylmethyl)heptanoateIC5030.0 [1], 1400.0 [2]
2-(Propanoylselenomethyl)-7-aminoheptanoic acidIC501.1 [1], 760.0 [2]
2-[(4-Phenylbutyrylseleno)methyl]-7-aminoheptanoic acidIC504.1 [1], 1600.0 [2]
2-[(3-Phenylpropionylseleno)methyl]-7-aminoheptanoic acidIC505.3 [1], 2000.0 [2]
Ethyl 2-[(6-aminopyridin-3-yl)methyl]-3-propanoylselanylpropanoateIC50890.0 [1], 180000.0 [2]
Ethyl 2-[(6-amino-5-chloropyridin-3-yl)methyl]-3-propanoylselanylpropanoateIC502600.0 [1], 3800000.0 [2]
7-Amino-2-[[(7-amino-2-carboxyheptyl)diselanyl]methyl]heptanoic acidIC502.0 [1], 3800000.0 [2]
3-(6-Aminopyridin-3-yl)-2-[[[3-(6-aminopyridin-3-yl)-2-carboxypropyl]diselanyl]methyl]propanoic acidIC500.0 [1], 200.0 [2]
3-(6-Amino-5-chloropyridin-3-yl)-2-[[[3-(6-amino-5-chloropyridin-3-yl)-2-carboxypropyl]diselanyl]methyl]propanoic acidIC500.03 [1], 3300.0 [2]
(2S,3R)-2-[(6-Aminopyridin-3-yl)methyl]-3-sulfanylbutanoic acidIC5087.0 [1], 400.0 [2]
(5R)-5-(3-Aminopropyl)-1-cyclohexyl-6,7-dihydro-4H-benzimidazole-5-carboxylic acidIC5080.0 [1], 117.0 [2]
(5R)-5-(3-Aminopropyl)-1-[(3-phenylphenyl)methyl]-6,7-dihydro-4H-benzimidazole-5-carboxylic acidIC50106.0 [1], 2500.0 [2]
5-(3-Aminopropyl)-1-[2-(4-cyclohexylcyclohexyl)ethyl]-6,7-dihydro-4H-benzimidazole-5-carboxylic acidIC50124.0 [1], 16000.0 [2]
5-(3-Aminopropyl)-1-phenyl-6,7-dihydro-4H-benzimidazole-5-carboxylic acidIC50585.0 [1], 7100.0 [2]
7-(3-Aminopropyl)-3-ethyl-6,8-dihydro-5H-imidazo[1,2-a]pyridine-7-carboxylic acidIC502270.0 [1], 100000.0 [2]
(7R)-7-(3-Aminopropyl)-3-phenyl-6,8-dihydro-5H-imidazo[1,2-a]pyridine-7-carboxylic acidIC5066.0 [1], 1300.0 [2]
5-Amino-2-[[1-(4-methylcyclohexyl)imidazol-4-yl]methyl]pentanoic acidIC508.3 [1], 9.3 [2]
5-Amino-2-[[1-(4-hydroxycyclohexyl)imidazol-4-yl]methyl]pentanoic acidIC5019.0 [1], 26.0 [2]
(5R)-5-(3-Aminopropyl)-1-(3-methylbutyl)-6,7-dihydro-4H-benzimidazole-5-carboxylic acidIC5041.0 [1], 100.0 [2]
(7R)-7-(3-Aminopropyl)-3-[3-(2,4-dichlorophenyl)phenyl]-6,8-dihydro-5H-imidazo[1,2-a]pyridine-7-carboxylic acidIC5041.0 [1], 3200.0 [2]
2-Benzylsuccinic acidIC501600.0 [1]
Anabaenopeptin FIC501.5 [1]
Anabaenopeptin BIC501.5 [1]
Oscillamide YIC50400.0 [1]
(2S)-7-Amino-2-[[hydroxy-[(1R)-2-methyl-1-(3-phenylpropanoylamino)propyl]phosphoryl]methyl]heptanoic acidIC505.5 [1]
alpha-Benzyl-1H-imidazole-4-acetic acidIC50100000.0 [1]
5-Amino-2-[(1-propylimidazol-4-yl)methyl]pentanoic acidKi46.0 [1]
(2S)-2-(2-Aminoethoxy)-3-(1-phenylimidazol-4-yl)propanoic AcidKi3.5 [1]
6-Amino-2-(1H-imidazol-4-yl)-hexanoic acidIC50590.0 [1]
(S)-2-((R)-1-Aminopropan-2-yloxy)-3-(1-phenyl-1H-imidazol-4-yl)propanoic acidKi7.5 [1]
3-Mercapto-2-(piperidin-4-yl)propanoic acidIC5037.0 [1]
2-(1-Carbamimidoylpiperidin-4-yl)-3-mercaptopropanoic acidIC501070.0 [1]
2-(Mercaptomethyl)-3-(piperidin-4-yl)propanoic acidIC50139.0 [1]
3-Mercapto-2-(piperidin-3-yl)propanoic acidIC5068.0 [1]
2-(3-Aminophenyl)-3-mercaptopropanoic acidIC50785.0 [1]
2-(1-Carbamimidoylpiperidin-3-yl)-3-mercaptopropanoic acidIC5045.0 [1]
2-[3-(Diaminomethylideneamino)phenyl]-3-sulfanylpropanoic acidIC503.0 [1]
2-(2-Chloro-5-guanidinophenyl)-3-mercaptopropanoic acidIC5011.0 [1]
2-(1-(1-Iminoethyl)piperidin-4-yl)-3-mercaptopropanoic acidIC505300.0 [1]
2-(1-(2-Aminoacetyl)piperidin-4-yl)-3-mercaptopropanoic acidIC507350.0 [1]
(2S)-2-[(2R)-1-Aminopropan-2-yl]oxy-3-(1-pyridin-2-ylimidazol-4-yl)propanoic acidKi5.8 [1]
(S)-2-(2-Aminoethylamino)-3-(1-isobutyl-1H-imidazol-4-yl)propanoic acidKi100.0 [1]
(2S)-2-[(2-Aminoethyl)amino]-3-(1H-imidazol-4-yl)propanoic acidKi344.0 [1]
(S)-2-(2-Aminoethylamino)-3-(1-butyl-1H-imidazol-4-yl)propanoic acidKi70.0 [1]
(2S)-6-Amino-2-[[(3S,6S,9S,12S,15R)-3-benzyl-9-[2-(4-hydroxyphenyl)ethyl]-6,7-dimethyl-2,5,8,11,14-pentaoxo-12-propan-2-yl-1,4,7,10,13-pentazacyclononadec-15-yl]carbamoylamino]hexanoic acidIC501.9 [1]
(2S)-6-Amino-2-[[(2R)-1-oxo-3-phenyl-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]hexanoic acidIC5015.0 [1]
(2S)-6-Amino-2-[[(2R)-4-methyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]pentan-2-yl]carbamoylamino]hexanoic acidIC5057.0 [1]
(2S)-6-Amino-2-[[(2R)-3-methyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]butan-2-yl]carbamoylamino]hexanoic acidIC50460.0 [1]
(2S)-6-Amino-2-[[(1R)-1-cyclohexyl-2-oxo-2-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]ethyl]carbamoylamino]hexanoic acidIC501000.0 [1]
(2S)-6-Amino-2-[[2-oxo-2-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]ethyl]carbamoylamino]hexanoic acidIC503700.0 [1]
(2S)-6-Amino-2-[[2-methyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]hexanoic acidIC506100.0 [1]
(2S)-6-Amino-2-[[(2R)-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]pentan-2-yl]carbamoylamino]hexanoic acidIC5015.0 [1]
(2S)-6-Amino-2-[[(2R)-3-cyclopropyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]hexanoic acidIC507.0 [1]
(2S)-6-Amino-2-[[(2R)-3-cyclobutyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]hexanoic acidIC509.0 [1]
(2S)-6-Amino-2-[[3-cyclopentyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]hexanoic acidIC504.0 [1]
(2S)-5-Amino-2-[[(2R)-3-cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]pentanoic acidIC5018.0 [1]
(2R)-3-(2-Aminoethylsulfonyl)-2-[[(2R)-3-cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]propanoic acidIC5038.0 [1]
(2R)-3-(2-Aminoethylsulfanyl)-2-[[(2R)-3-cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]propanoic acidIC504.0 [1]
(2S)-2-[[(2R)-3-Cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]-5-(diaminomethylideneamino)pentanoic acidIC504.0 [1]
(2S)-2-[[(2R)-3-Cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]-4-(diaminomethylideneamino)oxybutanoic acidIC50100.0 [1]
(2S)-3-(6-Aminopyridin-3-yl)-2-[[(2R)-3-cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]propanoic acidIC501.0 [1]
(2R)-3-(6-Aminopyridin-3-yl)-2-[[(2R)-3-cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]propanoic acidIC50250.0 [1]
(2S)-6-Amino-2-[[(2R)-3-cyclohexyl-1-oxo-1-[(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]propan-2-yl]carbamoylamino]hexanamideIC50750.0 [1]
(2R)-2-[[(2S)-1-Amino-3-(6-aminopyridin-3-yl)-1-oxopropan-2-yl]carbamoylamino]-3-cyclohexyl-N-(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)propanamideIC50570.0 [1]
(2R)-2-[[(1S)-2-(6-Aminopyridin-3-yl)-1-cyanoethyl]carbamoylamino]-3-cyclohexyl-N-(4,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl)propanamideIC5054000.0 [1]
(2S)-6-Amino-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]hexanoic acidIC5012.0 [1]
(2S)-6-(Carbamoylamino)-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]hexanoic acidIC5030000.0 [1]
(2S)-6-Amino-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]-6-oxohexanoic acidIC5030000.0 [1]
(2S)-6-Amino-2-[[(2R)-1-(2-bicyclo[2.2.1]heptanylamino)-3-cyclohexyl-1-oxopropan-2-yl]sulfamoylamino]hexanoic acidIC5075000.0 [1]
(2S)-2-[[(2S)-3-Cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]-6-hydroxyhexanoic acidIC5030000.0 [1]
(2S)-6-Amino-2-[[(2S)-3-cyclohexyl-1-(cyclohexylamino)-1-oxopropan-2-yl]sulfamoylamino]hexanoic acidIC501700.0 [1]
(2S)-2-[[(2S)-3-Cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]-3-phenylpropanoic acidIC5024000.0 [1]
(2S)-2-[[(2S)-1-(1-Adamantylamino)-1-oxopropan-2-yl]sulfamoylamino]-6-aminohexanoic acidIC5030000.0 [1]
(2S)-6-Amino-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(2S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]carbamoylamino]hexanoic acidIC503.0 [1]
(2S)-2-[[(2S)-1-(1-Adamantylamino)-3-methyl-1-oxobutan-2-yl]sulfamoylamino]-6-aminohexanoic acidIC5030000.0 [1]
(2S)-2-[[(2S)-3-Cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]-3-piperidin-4-ylpropanoic acidIC50880.0 [1]
(2S)-3-(6-Aminopyridin-3-yl)-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]propanoic acidIC5026.0 [1]
(2S)-5-(1-Aminoethylideneamino)-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]pentanoic acidIC501500.0 [1]
(2S)-2-[[(2S)-1-(1-Adamantylamino)-4-methyl-1-oxopentan-2-yl]sulfamoylamino]-6-aminohexanoic acidIC5010000.0 [1]
(2S)-2-[[(2S)-3-Cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]-6-(dimethylamino)hexanoic acidIC5044000.0 [1]
(2S)-3-(4-Aminocyclohexyl)-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]propanoic acidIC5030000.0 [1]
(2S)-2-[[2-(1-Adamantylamino)-2-oxoethyl]sulfamoylamino]-6-aminohexanoic acidIC5030000.0 [1]
(2S)-6-Amino-2-[[(2S)-1-(2-bicyclo[2.2.1]heptanylamino)-3-cyclohexyl-1-oxopropan-2-yl]carbamoylamino]hexanoic acidIC5038.0 [1]
(2S)-6-Amino-2-[[(2S)-1-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-3-cyclohexyl-1-oxopropan-2-yl]sulfamoylamino]hexanoic acidIC50420.0 [1]
(2S)-2-[[(1S)-2-(1-Adamantylamino)-2-oxo-1-phenylethyl]sulfamoylamino]-6-aminohexanoic acidIC5030000.0 [1]
(2S)-2-[[(2S)-3-Cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]-3-(1H-imidazol-5-yl)propanoic acidIC504400.0 [1]
(2S)-6-Amino-2-[[(2S)-1-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-3-cyclohexyl-1-oxopropan-2-yl]sulfamoylamino]hexanoic acidIC50330.0 [1]
(2S)-6-Acetamido-2-[[(2S)-3-cyclohexyl-1-oxo-1-[[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propan-2-yl]sulfamoylamino]hexanoic acidIC5030000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Carboxypeptidase B2 isoform A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/carboxypeptidase-b2-isoform-a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Carboxypeptidase B2 isoform A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/carboxypeptidase-b2-isoform-a-inhibitors-ic50-ki.
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