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Casein kinase I alpha Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
3-[(2,4,6-Trimethoxyphenyl)methylidene]-1H-indol-2-oneIC501000.0 [1], 1240.0 [2]
StaurosporineIC504188.0 [1]
GefitinibIC5050000.0 [1]
SorafenibIC50250.0 [1]
SunitinibIC501.0 [1]
DasatinibIC501.0 [1]
N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamideKi38300.0 [1]
SeliciclibIC504000.0 [1]
DoramapimodIC5030000.0 [1]
1,4-DihydroxyanthraquinoneIC5040000.0 [1]
N-(2-Aminoethyl)-5-chloroisoquinoline-8-sulfonamideIC5010000.0 [1]
CK1 InhibitorIC50300.0 [1]
2-((3,5-Difluoro-4-hydroxyphenyl)amino)-8-isopentyl-5,7-dimethyl-7,8-dihydropteridin-6(5H)-oneIC50450.0 [1]
(3Z)-3-[(2,4,6-Trimethoxyphenyl)methylidene]-1H-indol-2-oneIC5011000.0 [1]
1,4-DiaminoanthraquinoneIC504000.0 [1]
N-(2-Aminoethyl)-5-chloronaphthalene-1-sulfonamideKi80000.0 [1]
1-Amino-4-hydroxyanthraquinoneIC504000.0 [1]
(2S,3S)-3-((7-(Benzylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-5-yl)amino)butane-1,2,4-triolIC501040.0 [1]
2-(3-Hydroxy-4-methoxystyryl)-8-hydroxyquinoline-7-carboxylic acidIC5010000.0 [1]
Cep-11981IC5048.0 [1]
(R)-2-((9-Isopropyl-6-((3-(pyridin-2-yl)phenyl)amino)-9H-purin-2-yl)amino)butan-1-olIC5014.0 [1]
CID 44814409IC5010000.0 [1]
7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrileKi6916.0 [1]
1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
2-(2,4-Dihydroxybenzylcarbamoyl)-8-hydroxyquinoline-7-carboxylic acidIC5010000.0 [1]
1-[5-Amino-4-(3,4-dichlorophenyl)-3-methylpyrazol-1-yl]ethanoneIC50100000.0 [1]
3-{[(1R)-1-Phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dioneIC50250.0 [1]
N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamideIC50872.0 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC509120.11 [1]
1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaIC5030000.0 [1]
7,8-Dichloro-9-methyl-1-oxospiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileIC50330.0 [1]
2-[(2S)-2-(4-Fluorophenyl)morpholin-4-yl]-3-methyl-6-pyrimidin-4-ylpyrimidin-4-oneIC501500.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-oneIC5010000.0 [1]
1-[3-[(3-Amino-2H-pyrazolo[3,4-d]pyrimidin-6-yl)amino]phenyl]-3-(3-chloro-4-fluorophenyl)ureaIC5078.0 [1]
2-[2-[(4-Fluoro-2-methylphenoxy)methyl]-5-methoxypyridin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC50442.0 [1]
CID 76072859IC50694.0 [1]
CID 90643548IC50545.0 [1]
N-Methyl-4-(2-(piperidin-4-yl)-5-(3-(trifluoromethyl)phenyl)-1H-imidazol-4-yl)pyrimidin-2-amineIC501100.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
3-[5-Chloro-4-[(2,4-difluorophenyl)methoxy]-6-oxopyrimidin-1-yl]-N-(2-hydroxyethyl)-4-methylbenzamideIC5010000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
2-[3-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
5,5-Dimethyl-8-[[4-(2,2,2-trifluoroethylamino)furo[3,2-d]pyrimidin-2-yl]amino]-1H-4,1-benzoxazepin-2-oneIC5010000.0 [1]
2-Amino-7-methyl-4-[(4-methylphenyl)methylamino]-9H-pyrimido[4,5-b]indol-6-olIC50100000.0 [1]
(2E)-2-[(3,4-Dihydroxyphenyl)methylidene]-1-benzofuran-3-oneIC5078800.0 [1]
4-(4-(4-Fluorophenyl)-2-(4-methylcyclohexyl)-1H-imidazol-5-yl)pyridineIC501300.0 [1]
(R)-2-((9-Isopropyl-6-((3-(pyridin-2-yl)phenyl)-amino)-9H-purin-2-yl)amino)butan-1-olIC5014.0 [1]
(1S,2R,3R)-3-[[9-Propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]cyclohexane-1,2-diolIC50600.0 [1]
(2R)-3-[[9-Propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]propane-1,2-diolIC50180.0 [1]
N-[(4-Methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridin-4-amineKi1000000.0 [1]
4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diolKi1000000.0 [1]
2-[(4-{[3-(Trifluoromethyl)pyridin-2-Yl]oxy}phenyl)amino]-1h-Benzimidazole-6-CarbonitrileIC5012100.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC5010000.0 [1]
2-[2-[(3,4-Difluorophenoxy)methyl]-5-methoxypyridin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC50251.0 [1]
2-N-(1H-Indazol-6-yl)-4-N-(2,2,2-trifluoroethyl)furo[3,2-d]pyrimidine-2,4-diamineIC505220.0 [1]
N~4~-Cyclopropyl-N~2~-(3-Methyl-1h-Indazol-6-Yl)furo[3,2-D]pyrimidine-2,4-DiamineIC507540.0 [1]
2-N-(3-Chloro-4-morpholin-4-ylphenyl)-4-N-(2,2,2-trifluoroethyl)furo[3,2-d]pyrimidine-2,4-diamineIC5010000.0 [1]
(2S)-4-[[9-Propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]butane-1,2-diolIC50660.0 [1]
1-[4-[(3-Amino-2H-pyrazolo[3,4-d]pyrimidin-6-yl)amino]phenyl]-3-[(1R)-1-phenylethyl]ureaIC5010000.0 [1]
2-[(4-Tert-Butylphenyl)amino]-1h-Benzimidazole-6-CarbonitrileIC507580.0 [1]
1-[4-[(3-Amino-2H-pyrazolo[3,4-d]pyrimidin-6-yl)amino]phenyl]-3-(3-chloro-4-fluorophenyl)ureaIC5010000.0 [1]
2-(4-Phenoxyanilino)-3H-benzimidazole-5-carbonitrileIC508820.0 [1]
2-(4-Phenylanilino)-3H-benzimidazole-5-carbonitrileIC505490.0 [1]
1-[3-[(3-Amino-2H-pyrazolo[3,4-d]pyrimidin-6-yl)amino]phenyl]-3-[(1R)-1-phenylethyl]ureaIC502470.0 [1]
2-[4-(2-Fluoropyridin-3-yl)anilino]-3H-benzimidazole-5-carbonitrileIC504670.0 [1]
2-(4-Methylanilino)-3H-benzimidazole-5-carbonitrileIC5019700.0 [1]
2-[4-(2-Hydroxypropan-2-yl)anilino]-3H-benzimidazole-5-carbonitrileIC509180.0 [1]
1-[3-[(3-Amino-2H-pyrazolo[3,4-d]pyrimidin-6-yl)amino]phenyl]-3-(5-tert-butyl-1H-pyrazol-3-yl)ureaIC50142.0 [1]
2-[4-(1-Methylpyrazol-4-yl)anilino]-3H-benzimidazole-5-carbonitrileIC503540.0 [1]
(3R,5S)-5-(Hydroxymethyl)-1-[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]pyrrolidin-3-olIC50390.0 [1]
[(2R)-2-Hydroxy-3-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]propyl] (2S)-2-amino-3-methylbutanoate;hydrochlorideIC50150.0 [1]
2-[2-[2-(4-Fluorophenyl)ethyl]-5-methoxypyridin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC50736.0 [1]
2-[5-Methoxy-2-(Quinolin-3-Yl)pyrimidin-4-Yl]-1,5,6,7-Tetrahydro-4h-Pyrrolo[3,2-C]pyridin-4-OneIC509.0 [1]
2-[2-[(E)-2-(4-Fluorophenyl)ethenyl]-5-methoxypyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC5033.0 [1]
2-[2-[(4-Fluorophenoxy)methyl]-5-methoxypyridin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC50174.0 [1]
2-[2-[(4,5-Difluoro-2-methylphenoxy)methyl]-5-methoxypyridin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC50383.0 [1]
2-[2-[2-(4-Fluorophenyl)ethyl]-5-methoxypyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC50568.0 [1]
2-[2-[(4-Fluorophenyl)methoxy]-5-methoxypyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC5095.0 [1]
2-(2-Anilino-5-methoxypyrimidin-4-yl)-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC5054.0 [1]
2-(5-Methoxy-2-phenoxypyrimidin-4-yl)-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC5018500.0 [1]
2-[2-(Benzylamino)-5-methoxypyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC5019.0 [1]
2-[2-[(4-Fluorophenoxy)methyl]-5-methoxypyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC50146.0 [1]
2-[2-[(2,4-Difluorophenoxy)methyl]-5-methoxypyridin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC50225.0 [1]
1-[(3-Hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea;methanesulfonic acidIC50469800.0 [1]
Items per page: 1 - 10 of 85
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References

This online tool may be cited as follows

MLA

"Quest Database™ Casein kinase I alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/casein-kinase-i-alpha-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Casein kinase I alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/casein-kinase-i-alpha-inhibitors-ic50-ki.
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