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Casein kinase I delta Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
PF-670462 free baseIC5013.0 [1]
3-[(2,4,6-Trimethoxyphenyl)methylidene]-1H-indol-2-oneIC501000.0 [1], 2570.0 [2]
3-[(3-Chlorophenoxy)methyl]-1-(Tetrahydro-2h-Pyran-4-Yl)-1h-Pyrazolo[3,4-D]pyrimidin-4-AmineIC5032.0 [1], 711.0 [2]
4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazoleIC50120.0 [1], 124.0 [2]
CK1 InhibitorIC50300.0 [1]
Bischof-5IC5022.0 [1], 42.0 [2]
[(4-{2-[(3-Hydroxyphenyl)amino]-1h-Benzimidazol-1-Yl}-1,3,5-Triazin-2-Yl)amino]acetonitrileIC5016000.0 [1], 40000.0 [2]
4-[1-Methyl-3-(4-fluorophenyl)-1H-pyrazole-4-yl]pyridineIC5048.1 [1], 545.0 [2]
3-[4-[3-(4-Fluorophenyl)-1-methylpyrazol-4-yl]pyridin-2-yl]morpholineIC506.6 [1], 90.0 [2]
9-[3-(4-Fluorophenyl)-1-Methyl-1h-Pyrazol-4-Yl]-2,3,4,5-Tetrahydropyrido[2,3-F][1,4]oxazepineIC506.0 [1], 42.1 [2]
1-{4-[3-(4-Fluorophenyl)-1-Methyl-1h-Pyrazol-4-Yl]pyridin-2-Yl}-N-MethylmethanamineIC5012.9 [1], 63.8 [2]
4-[1-Methyl-3-(4-fluorophenyl)-1H-pyrazole-4-yl]pyridine-2-methanolIC5014.2 [1], 237.0 [2]
HarmineIC501500.0 [1]
4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridyl)-1H-imidazoleIC50188.0 [1]
1-Tert-butyl-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC5041.0 [1]
1,4-DihydroxyanthraquinoneIC5040000.0 [1]
N3-(4-Fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,4-diamineIC50510.0 [1]
HymenialdisineIC5035.0 [1]
3-[(2,4,6-Trimethoxy-phenyl)-methylene]-indolin-2-oneIC501000.0 [1]
1-(Tert-Butyl)-3-(p-tolyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC50170.0 [1]
(3Z)-3-[(2,4,6-Trimethoxyphenyl)methylidene]-1H-indol-2-oneIC50700.0 [1]
1,4-DiaminoanthraquinoneIC50330.0 [1]
CID 46209401IC5010000.0 [1]
1-Amino-4-hydroxyanthraquinoneIC50660.0 [1]
1-(Tert-Butyl)-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC50150.0 [1]
JNK Inhibitor VIIIKi7800.0 [1]
N-(1,3-Benzothiazol-2-yl)-2-phenylacetamideIC50330.0 [1]
CID 59604787IC5010000.0 [1]
N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-9-(3-fluorophenyl)-2-morpholin-4-ylpurin-6-amineIC5044.0 [1]
Hymenialdisine Analogue 1IC501352.0 [1]
4-(Pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-oneIC5010000.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamideKi7800.0 [1]
4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamideKi7800.0 [1]
4-[3-(4-Fluorophenyl)-5-isopropylisoxazol-4-yl]pyridineIC50230.0 [1]
7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrileKi7826.0 [1]
1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
Khk-IN-1IC5040000.0 [1]
5-(4-Chlorophenyl)-N-(4-piperazin-1-ylphenyl)furan-2-carboxamideIC5030000.0 [1]
2,2-Dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-1-[(1R)-1-phenylethyl]-3H-quinazolin-4-oneIC501000.0 [1]
7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamideKi10000.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamideKi7800.0 [1]
N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi7800.0 [1]
N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi7800.0 [1]
N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamideKi7800.0 [1]
3-Methyl-N-[6-methylsulfanyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amineIC501900.0 [1]
3-[[[5-[1-(4-Methoxyphenyl)-1H-benzimidazol-6-yl]-1,3,4-oxadiazol-2-yl]thio]methyl]benzonitrileIC5010000.0 [1]
2-(4-Fluorophenyl)-3-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]imidazo[1,2-a]pyrimidin-7-amineIC50100000.0 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amineIC50530.0 [1]
3-[(1R)-1-[(2S,6R)-2,6-Dimethylmorpholin-4-yl]ethyl]-N-[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amineIC5010.0 [1]
N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamideIC50740.0 [1]
N-(1,3-Benzothiazol-2-yl)-3,3-diphenylpropanamideIC502500.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
4-(Cyclopentylamino)-2-[(2-methoxyphenyl)methylamino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamideIC5030000.0 [1]
2-[2-[(4-Fluoro-2-methylphenoxy)methyl]-5-methoxypyridin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneIC5059.0 [1]
4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamideIC5030000.0 [1]
4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideIC5030000.0 [1]
CID 71553154IC50110.0 [1]
CID 76072859IC5084.0 [1]
4-[2-[1-(2-Diethoxyphosphorylethyl)triazol-4-yl]-5-(4-fluorophenyl)-3-methylimidazol-4-yl]pyridineIC503100.0 [1]
4-[4-[4-(4-Fluorophenyl)-1-methyl-5-pyridin-4-ylimidazol-2-yl]triazol-1-yl]benzoic acidIC501600.0 [1]
2-[4-[4-(4-Fluorophenyl)-1-methyl-5-pyridin-4-ylimidazol-2-yl]triazol-1-yl]ethanolIC50240.0 [1]
4-[5-(4-Fluorophenyl)-3-methyl-2-(2H-triazol-4-yl)imidazol-4-yl]pyridineIC50202.0 [1]
3-[4-[4-(4-Fluorophenyl)-1-methyl-5-pyridin-4-ylimidazol-2-yl]triazol-1-yl]benzoic acidIC5089.0 [1]
2-[(2,2-Diphenylacetyl)amino]-benzothiazoleIC501960.0 [1]
CID 90643548IC50104.0 [1]
N-[6-(Methylsulfonyl)benzothiazol-2-yl]-2-(2-thienyl)acetamideIC502690.0 [1]
N-Methyl-4-(2-(piperidin-4-yl)-5-(3-(trifluoromethyl)phenyl)-1H-imidazol-4-yl)pyrimidin-2-amineIC501400.0 [1]
(2R,3R,4R,5S,6R)-3-[4-[4-(4-Fluorophenyl)-1-methyl-5-pyridin-4-ylimidazol-2-yl]triazol-1-yl]-6-(hydroxymethyl)oxane-2,4,5-triolIC50439.0 [1]
7-Ethynyl-2-(4-fluorophenyl)-3-(2-methylsulfanylpyrimidin-4-yl)imidazo[1,2-a]pyrimidineIC50100000.0 [1]
7-[1-(2-Diethoxyphosphorylethyl)triazol-4-yl]-2-(4-fluorophenyl)-3-(2-methylsulfanylpyrimidin-4-yl)imidazo[1,2-a]pyrimidineIC5021400.0 [1]
4-[2-(4-Ethynylphenyl)-5-(4-fluorophenyl)-1H-imidazol-4-yl]-1H-pyridin-2-oneIC5019900.0 [1]
4-[5-(4-Fluorophenyl)-2-[4-[1-(2-hydroxyethyl)triazol-4-yl]phenyl]-1H-imidazol-4-yl]-1H-pyridin-2-oneIC5017900.0 [1]
Ethyl 2-[4-[4-[5-(4-fluorophenyl)-4-(2-oxo-1H-pyridin-4-yl)-1H-imidazol-2-yl]phenyl]triazol-1-yl]acetateIC5024500.0 [1]
4-[2-[4-[1-(2-Diethoxyphosphorylethyl)triazol-4-yl]phenyl]-5-(4-fluorophenyl)-1H-imidazol-4-yl]-1H-pyridin-2-oneIC5044300.0 [1]
4-[5-(4-Fluorophenyl)-2-piperidin-4-yl-1H-imidazol-4-yl]-1H-pyridin-2-oneIC5012000.0 [1]
4-[2-(4-Ethynylphenyl)-4-(4-fluorophenyl)-1H-imidazol-5-yl]-2-methylsulfanylpyrimidineIC5066300.0 [1]
N-[2-(1,3-Benzothiazol-2-ylamino)-2-oxoethyl]benzamideIC507290.0 [1]
4-[4-[3-[4-[(Propan-2-ylamino)methyl]anilino]-1H-pyrazol-5-yl]phenyl]benzene-1,3-diolIC506340.0 [1]
N-(6-Ethoxy-1,3-benzothiazol-2-yl)-2,2-diphenylacetamideIC502820.0 [1]
3-Amino-1-methyl-6-[4-(4-methylpiperazin-1-yl)phenyl]-5H-pyrazolo[4,3-c]pyridin-4-oneIC5039000.0 [1]
4-[5-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-1H-imidazol-4-yl]-1H-pyridin-2-oneIC5019700.0 [1]
Sodium;5-[5-(4-fluorophenyl)-4-(2-oxo-1H-pyridin-4-yl)-1H-imidazol-2-yl]-2-hydroxybenzoateIC5021200.0 [1]
4-[4-(4-Fluorophenyl)-5-(2-methylsulfanylpyrimidin-4-yl)-1H-imidazol-2-yl]phenolIC505960.0 [1]
N-(1,3-Benzothiazol-2-yl)-3-(3-chlorophenyl)propanamideIC503580.0 [1]
N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-2-(4-methylpiperazin-1-yl)-9-pyridin-3-ylpurin-6-amineIC50700.0 [1]
N-[(6-Methoxy-1H-benzimidazol-2-yl)methyl]-2-piperazin-1-yl-9-pyridin-3-ylpurin-6-amineIC50625.0 [1]
N-[(6-Methoxy-1H-benzimidazol-2-yl)methyl]-2-morpholin-4-yl-9-pyridin-3-ylpurin-6-amineIC50520.0 [1]
6-N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-9-(3-fluorophenyl)-2-N-(3-morpholin-4-ylpropyl)purine-2,6-diamineIC50915.0 [1]
6-N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-9-(3-fluorophenyl)purine-2,6-diamineIC5055.0 [1]
N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-9-(4-fluorophenyl)-2-morpholin-4-ylpurin-6-amineIC50535.0 [1]
9-(3-Fluorophenyl)-2-morpholin-4-yl-N-[(5-phenyl-1H-imidazol-2-yl)methyl]purin-6-amineIC50215.0 [1]
9-(3-Fluorophenyl)-N-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]methyl]-2-morpholin-4-ylpurin-6-amineIC5050.0 [1]
N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-2-(1,1-dioxo-1,4-thiazinan-4-yl)-9-(3-fluorophenyl)purin-6-amineIC50175.0 [1]
N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-9-(2,4-difluorophenyl)-2-morpholin-4-ylpurin-6-amineIC50525.0 [1]
N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-2-(4-methylpiperazin-1-yl)-9-(2-methylpyridin-4-yl)purin-6-amineIC50295.0 [1]
6-N-[(4,5-Difluoro-1H-benzimidazol-2-yl)methyl]-9-(3-fluorophenyl)-2-N-(2-morpholin-4-ylethyl)purine-2,6-diamineIC50830.0 [1]
N-(1H-Benzimidazol-2-ylmethyl)-2-morpholin-4-yl-9-pyridin-3-ylpurin-6-amineIC501155.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Casein kinase I delta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/casein-kinase-i-delta-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Casein kinase I delta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/casein-kinase-i-delta-inhibitors-ic50-ki.
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