Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| PF-670462 free base | IC50 | 8.0 [1], 29.0 [2], 32.0 [3], 80.0 [4], 130.0 [5] | |
| 3-[(3-Chlorophenoxy)methyl]-1-(Tetrahydro-2h-Pyran-4-Yl)-1h-Pyrazolo[3,4-D]pyrimidin-4-Amine | IC50 | 32.0 [1] | |
| Bischof-5 | IC50 | 199.0 [1] | |
| N-(2,2-Difluoro-5H-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-[[2-(trifluoromethoxy)benzoyl]amino]-1,3-thiazole-4-carboxamide | IC50 | 190.0 [1], 210.0 [2] | |
| N-(2,2-Difluoro-5H-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-3-methoxybenzamide | IC50 | 160.0 [1], 520.0 [2] | |
MLA | "Quest Database™ Casein kinase I epsilon Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Jan. 2026, https://www.aatbio.com/data-sets/casein-kinase-i-epsilon-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2026, January 20). Quest Database™ Casein kinase I epsilon Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/casein-kinase-i-epsilon-inhibitors-ic50-ki. | |
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