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Caspase-1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Ac-Yvad-choIC508.4 [1], 17.0 [2], 2000.0 [3], 68000.0 [4]
Ac-Yvad-choKi0.76 [1], 6.0 [2]
PralnacasanIC502.0 [1], 3.6 [2], 420.0 [3]
(S)-5-(2-Phenoxymethyl-pyrrolidine-1-sulfonyl)-1H-indole-2,3-dioneIC5010000.0 [1], 500000.0 [2]
(S)-5-(2-Phenoxymethyl-pyrrolidine-1-sulfonyl)-1H-indole-2,3-dioneKi17000.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseCaspase-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.10 Dec2025https://www.aatbio.com/data-sets/caspase-1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 10). Quest DatabaseCaspase-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/caspase-1-inhibitors-ic50-ki.
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