 | 4-[4-(Pyridin-3-ylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | IC50 | 155.0 [1], 2560.0 [2] |
| 4-[4-(Pyridin-3-ylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 59.0 [1] |
 | CID 104934 | Ki | 210.0 [1] |
 | Grassystatin A | IC50 | 5000.0 [1] |
 | N-[3-[1-[[(3S)-2-Hydroxy-5-oxooxolan-3-yl]carbamoyl]cyclopropyl]-2,4-dioxo-1-propan-2-ylpyrimidin-5-yl]-2-methyl-4-(naphthalen-2-ylamino)benzamide | IC50 | 2980.0 [1] |
 | Inhibitor 62b | Ki | 32000.0 [1] |
 | 4-[4-[[3,5-Bis(trifluoromethyl)phenyl]methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 48.0 [1] |
 | 4-[4-[(2-Nitrophenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 24.0 [1] |
 | 4-(4-Benzylpiperazin-1-yl)-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 41.0 [1] |
 | 4-[4-[(3,5-Dimethoxyphenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 34.0 [1] |
 | 4-[4-(2-Phenylethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 16.0 [1] |
 | 4-[4-[(3-Methoxyphenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 111.0 [1] |
 | 4-[4-(Pyridin-4-ylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 34.0 [1] |
 | 2,4-Dipyrrolidin-1-yl-6-[4-[[4-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]pyrimidine | Ki | 135.0 [1] |
 | 4-[4-(Cyclohexylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 59.0 [1] |
 | [4-[[4-(2,6-Dipyrrolidin-1-ylpyrimidin-4-yl)piperazin-1-yl]methyl]phenyl]-phenylmethanone | Ki | 28.0 [1] |
 | 4-[4-[(4-Nitrophenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine | Ki | 99.0 [1] |
 | 4-(Piperazin-1-yl)-2,6-di(pyrrolidin-1-yl)pyrimidine | Ki | 47.0 [1] |
 | 5-[[5-[[(2S)-1-Carboxy-4-(2-chlorophenyl)sulfanyl-3-oxobutan-2-yl]carbamoyl]pyridin-2-yl]methylsulfamoyl]-2-hydroxybenzoic acid | Ki | 11000.0 [1] |
 | 4-(Cyclopentylamino)-6-(3,5-difluorophenylamino)-1,3,5-triazine-2-carbonitrile | IC50 | 13489.63 [1] |
 | 3-[2-[5-Tert-butyl-3-[(4-methyl-1,2,5-oxadiazol-3-yl)methylamino]-2-oxopyrazin-1-yl]butanoylamino]-5-[hexyl(methyl)amino]-4-oxopentanoic acid;hydrochloride | IC50 | 0.2 [1] |
 | Inhibitor 47c | Ki | 98000.0 [1] |
 | (3S)-3-[4-(3-Carboxy-4-hydroxyphenylsulfonylaminomethyl)benzoylamino]-4-oxobutanoic acid | Ki | 12000.0 [1] |
 | CID 5327304 | Ki | 22000.0 [1] |
 | Inhibitor 64b | Ki | 23000.0 [1] |
 | Inhibitor 66a | Ki | 24000.0 [1] |
 | Inhibitor 66b | Ki | 63000.0 [1] |
 | Inhibitor 69b | Ki | 36000.0 [1] |
 | (E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-6-ethoxy-6-oxohex-4-enoic acid | IC50 | 100000.0 [1] |
 | (E,3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3,3-dimethylbutanoyl]azetidine-2-carbonyl]amino]-5-methylsulfonylpent-4-enoic acid | IC50 | 35200.0 [1] |
 | (E,3S)-3-[[(2S,3S)-2-[[(2S)-5-Amino-2-[[(2S)-3-(1H-indol-3-yl)-2-(phenylmethoxycarbonylamino)propanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]-5-methylsulfonylpent-4-enoic acid | IC50 | 750.0 [1] |
 | (E,3S)-3-[[(2S,3S)-2-[[(2S)-5-Amino-2-[[(2S)-3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]-5-methylsulfonylpent-4-enoic acid | IC50 | 19500.0 [1] |
 | (E,3S)-3-[[(2S)-1-[(2R)-2-[(4-Amino-3-chlorobenzoyl)amino]-3,3-dimethylbutanoyl]pyrrolidine-2-carbonyl]amino]-5-methylsulfonylpent-4-enoic acid | IC50 | 560.0 [1] |
 | 3-[[4-(2,6-Dipyrrolidin-1-ylpyrimidin-4-yl)piperazin-1-yl]methyl]-2,5,7,8-tetramethyl-3,4-dihydro-2H-chromen-6-ol | Ki | 81.0 [1] |
 | 3-[2-[5-Tert-butyl-3-[(4-methyl-1,2,5-oxadiazol-3-yl)methylamino]-2-oxopyrazin-1-yl]butanoylamino]-5-[methyl(pentyl)amino]-4-oxopentanoic acid | IC50 | 0.81 [1] |
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