 | 2-(Biphenyl-3-Yl)-5-Hydroxy-3-Methylpyrimidin-4(3h)-One | IC50 | 170.0 [1], 5000.0 [2] |
 | 5-(4-Methylbenzene-1-sulfonyl)quinolin-8-ol | IC50 | 19.95 [1], 501.19 [2] |
 | 8-Hydroxyquinoline | IC50 | 1584.89 [1], 3162.28 [2] |
 | Tolcapone | IC50 | 1.0 [1], 127.0 [2] |
 | 1-(Biphenyl-3-Yl)-3-Hydroxypyridin-4(1h)-One | IC50 | 47.0 [1], 1100.0 [2] |
 | 5-Hydroxy-2-[hydroxy(phenyl)methyl]-1-(3-phenylphenyl)pyridin-4-one | IC50 | 88.0 [1], 1300.0 [2] |
 | 5-Hydroxy-2-(1-hydroxybutyl)-1-(3-phenylphenyl)pyridin-4-one | IC50 | 57.0 [1], 1000.0 [2] |
 | 5-Hydroxy-2-(1-hydroxy-2-methylpropyl)-1-(3-phenylphenyl)pyridin-4-one | IC50 | 180.0 [1], 1900.0 [2] |
 | 2-(2-Aminoethyl)-5-hydroxy-1-(3-phenylphenyl)pyridin-4-one | IC50 | 13000.0 [1], 24000.0 [2] |
 | 5-Cyclopentylsulfonyl-7-fluoroquinolin-8-ol | IC50 | 2.0 [1], 2511.89 [2] |
 | 7-Fluoro-5-(4-fluorophenyl)sulfonylquinolin-8-ol | IC50 | 3.98 [1], 1584.89 [2] |
 | 7-Chloro-5-(4-fluorophenyl)sulfonylquinolin-8-ol | IC50 | 199.53 [1], 10000.0 [2] |
 | 7-Chloro-5-pyrrolidin-1-ylsulfonylquinolin-8-ol | IC50 | 10.0 [1], 3162.28 [2] |
 | 7-Chloro-5-cyclopentylsulfonylquinolin-8-ol | IC50 | 19.95 [1], 7943.28 [2] |
 | 7-Fluoro-5-[4-(trifluoromethyl)phenyl]sulfonylquinolin-8-ol | IC50 | 79.43 [1], 6309.57 [2] |
 | CID 122440031 | IC50 | 7.94 [1], 1995.26 [2] |
 | 5-Cyclopentylsulfonylquinolin-8-ol | IC50 | 6.31 [1], 501.19 [2] |
 | 7-Chloro-5-(4-methylphenyl)sulfonylquinolin-8-ol | IC50 | 316.23 [1], 10000.0 [2] |
 | 5-Cyclopentylsulfonyl-7-(trifluoromethyl)quinolin-8-ol | IC50 | 10000.0 [1] |
 | 5-Ethylsulfonylquinolin-8-ol | IC50 | 50.12 [1], 1584.89 [2] |
 | 7-Fluoranyl-5-(4-methylphenyl)sulfonyl-quinolin-8-ol | IC50 | 6.31 [1], 501.19 [2] |
 | 5-[4-(Trifluoromethyl)phenyl]sulfonylquinolin-8-ol | IC50 | 63.1 [1], 1258.93 [2] |
 | 7-Bromo-5-(4-methylphenyl)sulfonylquinolin-8-ol | IC50 | 1258.93 [1], 10000.0 [2] |
 | 7-Methyl-5-pyrrolidin-1-ylsulfonylquinolin-8-ol | IC50 | 19.95 [1], 3162.28 [2] |
 | 7-Fluoro-5-pyrrolidin-1-ylsulfonylquinolin-8-ol | IC50 | 3.98 [1], 1584.89 [2] |
 | 5-(4-Methylphenyl)sulfonyl-7-(trifluoromethyl)quinolin-8-ol | IC50 | 10000.0 [1] |
 | 5-(2-Benzylpyrrolidin-1-yl)sulfonylquinolin-8-ol | IC50 | 2.0 [1], 1995.26 [2] |
 | 3-Hydroxy-1-(2-phenylpyridin-4-yl)pyridin-4-one | IC50 | 456.0 [1], 2325.0 [2] |
 | 3-Hydroxy-1-(4-pyridin-2-yl-1,3-thiazol-2-yl)pyridin-4-one | IC50 | 5000.0 [1] |
 | 3-Hydroxy-1-isoquinolin-1-ylpyridin-4-one | IC50 | 962.0 [1], 1268.0 [2] |
 | 3-Hydroxy-1-(2-methylimidazo[1,2-b]pyridazin-6-yl)pyridin-4-one | IC50 | 1667.0 [1], 5000.0 [2] |
 | 5-Hydroxy-2-(1-hydroxyethyl)-1-(3-phenylphenyl)pyridin-4-one | IC50 | 99.0 [1], 940.0 [2] |
 | 3-Hydroxy-1-(6-phenylpyridin-2-yl)pyridin-4-one | IC50 | 128.0 [1], 2584.0 [2] |
 | 1-Biphenyl-3-yl-5-hydroxy-2-methylpyridin-4(1H)-one | IC50 | 53.0 [1], 2100.0 [2] |
 | 1-(Biphenyl-3-yl)-5-hydroxy-2-phenylpyridin-4(1H)-one | IC50 | 87.0 [1], 2500.0 [2] |
 | 3-Hydroxy-1-(4-phenylpyridin-2-yl)pyridin-4-one | IC50 | 40.0 [1], 3020.0 [2] |
 | 3-Hydroxy-1-(2-phenylpyrimidin-4-yl)pyridin-4(1H)-one | IC50 | 706.0 [1], 2054.0 [2] |
 | 5-Hydroxy-1-(3-phenylphenyl)-2-propan-2-ylpyridin-4-one | IC50 | 410.0 [1], 1500.0 [2] |
 | 3-Hydroxy-1-(3-phenylpyridin-2-yl)pyridin-4-one | IC50 | 5000.0 [1] |
 | 1-(3-Fluoro-4-phenylpyridin-2-yl)-3-hydroxypyridin-4-one | IC50 | 55.0 [1], 946.0 [2] |
 | 5'-Deoxy-5'-methylthioadenosine | Ki | 5400000.0 [1] |
 | Entacapone | IC50 | 386.0 [1] |
 | 8-Hydroxyquinoline-5-sulfonic acid | IC50 | 6309.57 [1] |
 | Opicapone | Ki | 10.0 [1] |
 | Hydroxy methylphenylpyridinone | IC50 | 18000.0 [1] |
 | 2,4-Dimethyl-5-(1H-Pyrazol-3-Yl)-1,3-Thiazole | Ki | 7943.28 [1] |
 | [(2S,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-dimethylsulfanium;iodide | Ki | 6000000.0 [1] |
 | 9-Hydroxy-6H-pyrido[2,1-c][1,4]benzothiazin-8-one | IC50 | 400.0 [1] |
 | 5-Hydroxy-2-thiophen-2-yl-1H-pyrimidin-6-one | IC50 | 860.0 [1] |
 | 5-Hydroxy-2-(hydroxymethyl)-1-(2-methoxyethyl)pyridin-4-one | IC50 | 10000.0 [1] |
 | 5-Hydroxy-2-(hydroxymethyl)-1-(3-phenylpropyl)pyridin-4-one | IC50 | 4500.0 [1] |
 | 1-(2,4-Dimethylphenyl)-5-hydroxy-2-(hydroxymethyl)pyridin-4-one | IC50 | 5800.0 [1] |
 | 1-(3,5-Dimethylphenyl)-3-hydroxy-2-methylpyridin-4-one | IC50 | 5500.0 [1] |
 | 1-(4-Butylphenyl)-5-hydroxy-2-(hydroxymethyl)pyridin-4-one | IC50 | 160.0 [1] |
 | 5-Hydroxy-2-(hydroxymethyl)-1-(4-phenylphenyl)pyridin-4-one | IC50 | 140.0 [1] |
 | 5-Hydroxy-2-(hydroxymethyl)-1-(3-phenylphenyl)pyridin-4-one | IC50 | 140.0 [1] |
 | 5-[3-(4-Fluorophenyl)pyrrolidin-1-yl]sulfonylquinolin-8-ol | IC50 | 3.16 [1] |
 | 5-Hydroxy-2-(hydroxymethyl)-1-phenylpyridin-4(1H)-one | IC50 | 3400.0 [1] |
 | 3-Hydroxy-1-(4-pyridin-2-ylpyridin-2-yl)pyridin-4-one | IC50 | 826.0 [1] |
 | 3-Hydroxy-1-(4-pyridin-4-ylpyridin-2-yl)pyridin-4-one | IC50 | 672.0 [1] |
 | 3-Hydroxy-1-(4-pyridin-3-ylpyridin-2-yl)pyridin-4-one | IC50 | 574.0 [1] |
 | 1-[4-(1-Benzylpyrazol-4-yl)pyridin-2-yl]-3-hydroxypyridin-4-one | IC50 | 49.5 [1] |
 | (5E)-5-[(3,4-Dihydroxy-5-nitrophenyl)methylidene]-3-ethyl-1,3-thiazolidine-2,4-dione | IC50 | 179.0 [1] |
 | 2-N,2-N,3-N,3-N-Tetraethyl-6,7-dihydroxy-5-nitronaphthalene-2,3-dicarboxamide | IC50 | 54.0 [1] |
 | (2S)-N-[3-[2-[2-[3-[5-[(3As,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]propoxy]ethoxy]ethoxy]propyl]-2-[(4-azidobenzoyl)amino]-N'-[6-[[4-(3,4-dihydroxy-5-nitrobenzoyl)phenyl]methyl-methylamino]-6-oxohexyl]butanediamide | IC50 | 648.0 [1] |
 | 5-Hydroxy-2-(hydroxymethyl)-1-(4-methylphenyl)pyridin-4-one | IC50 | 1700.0 [1] |
 | 3-Hydroxy-5-(4-methoxyphenyl)-1-methyl-6-pyridin-4-ylpyridin-2-one | IC50 | 2100.0 [1] |
 | 6-(4-Methylphenyl)sulfonylquinolin-8-ol | IC50 | 1584.89 [1] |
 | (8-Hydroxyquinolin-5-yl)-pyrrolidin-1-ylmethanone | IC50 | 10000.0 [1] |
 | 5-(4-Methylphenyl)quinolin-8-ol | IC50 | 251.19 [1] |
 | (8-Hydroxyquinolin-5-yl)-(4-methylphenyl)methanone | IC50 | 3981.07 [1] |
 | 8-Methoxy-5-pyrrolidin-1-ylsulfonylquinoline | IC50 | 10000.0 [1] |
 | 3-Chloro-5,6-dihydroxy-7-nitro-1-benzothiophene-2-carboxylic acid | Ki | 1.0 [1] |
 | 2'-Methyl-1H,2'H-3,3'-bipyrazole | Ki | 25118.86 [1] |
 | (3-Amino-3-carboxypropyl)-[2-(2-methoxyphenyl)ethyl]-methylsulfanium;iodide | Ki | 5800000.0 [1] |
 | [(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-methyl-(2-phenylethyl)sulfanium;iodide | Ki | 800000.0 [1] |
 | [(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[2-(2-methoxyphenyl)ethyl]-methylsulfanium;iodide | Ki | 800000.0 [1] |
 | [(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[2-[5-[2-[benzyl(methyl)amino]-1-hydroxyethyl]-2-methoxyphenyl]ethyl]-methylsulfanium;iodide | Ki | 500000.0 [1] |
 | Isobutyryloxymethyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 17.0 [1] |
 | (2-Oxo-1,3-dioxol-4-yl)methyl 3-chloro-5,6-dihydroxy-7-nitro-1-benzothiophene-2-carboxylate | Ki | 1.6 [1] |
 | Methyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 2.2 [1] |
 | Propyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 9.2 [1] |
 | Butyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 1.3 [1] |
 | Isopropyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 1.1 [1] |
 | Benzyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 10.2 [1] |
 | 1-(Isobutyryloxy)ethyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 17.0 [1] |
 | Butyryloxymethyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 10.6 [1] |
 | 1-(Butyryloxy)ethyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate | Ki | 16.6 [1] |
 | (2-Amino-3-methylbutanoyl)oxymethyl 3-chloro-5,6-dihydroxy-7-nitro-1-benzothiophene-2-carboxylate | Ki | 6.0 [1] |
 | 3-[2-Methyl-4-(Trifluoromethyl)-1,3-Thiazol-5-Yl]-1H-1,2,4-Triazole | Ki | 251188.64 [1] |
 | [1-(Biphenyl-3-yl)-5-hydroxy-4-oxo-1,4-dihydropyridin-3-yl]boronic acid | IC50 | 200.0 [1] |
 | 1-[4-(3,4-Dichlorophenyl)pyridin-2-yl]-3-hydroxypyridin-4-one | IC50 | 35.0 [1] |
 | 1-(3,5-Dimethylphenyl)-5-hydroxy-2-(hydroxymethyl)pyridin-4-one | IC50 | 680.0 [1] |
 | 1-[4-(2-Tert-butyl-1,3-thiazol-4-yl)pyridin-2-yl]-3-hydroxypyridin-4-one | IC50 | 101.0 [1] |
 | 3-Hydroxy-1-phenylpyridin-4-one | IC50 | 2400.0 [1] |
 | 1',3'-Dimethyl-1H,1'H-3,4'-bipyrazole | Ki | 15848.93 [1] |
 | 3-Hydroxy-1-[4-[6-(trifluoromethyl)pyridin-2-yl]pyridin-2-yl]pyridin-4-one | IC50 | 84.0 [1] |
 | 5-Hydroxy-2-[3-(2-phenylethynyl)phenyl]-1H-pyrimidin-6-one | IC50 | 590.0 [1] |
 | 5-Hydroxy-2-(4-trifluoromethyl-phenyl)-3H-pyrimidin-4-one | IC50 | 210.0 [1] |
 | 5-Hydroxy-2-[3-(4-methoxyphenoxy)phenyl]-3-methylpyrimidin-4(3H)-one | IC50 | 93.0 [1] |
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