 | Toxoflavin | IC50 | 10000.0 [1], 30000.0 [2], 34000.0 [3], 340000.0 [4] |
| Toxoflavin | Ki | 3650.0 [1], 3800.0 [2], 5820.0 [3] |
 | Cercosporin | IC50 | 10000.0 [1], 41000.0 [2], 130000.0 [3], 150000.0 [4] |
| Cercosporin | Ki | 5900.0 [1], 35560.0 [2] |
 | 4-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanoic acid | IC50 | 15000.0 [1], 170000.0 [2], 340000.0 [3] |
| 4-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanoic acid | Ki | 1000.0 [1], 17000.0 [2], 59000.0 [3] |
 | N-(4-Amino-1,2,5-oxadiazol-3-yl)-2-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetamide | IC50 | 31000.0 [1], 550000.0 [2], 630000.0 [3] |
| N-(4-Amino-1,2,5-oxadiazol-3-yl)-2-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetamide | Ki | 2700.0 [1], 31000.0 [2], 88000.0 [3] |
 | 8-[2-(2H-Tetrazol-5-yl)ethyl]-13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaene | IC50 | 76000.0 [1], 770000.0 [2], 850000.0 [3] |
| 8-[2-(2H-Tetrazol-5-yl)ethyl]-13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaene | Ki | 18000.0 [1], 53000.0 [2], 180000.0 [3] |
 | 4-Amino-N-(13-oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-ylimino)-1,2,5-oxadiazole-3-carboxamide | IC50 | 30000.0 [1], 52000.0 [2], 60000.0 [3] |
| 4-Amino-N-(13-oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-ylimino)-1,2,5-oxadiazole-3-carboxamide | Ki | 1200.0 [1], 20000.0 [2], 36000.0 [3] |
 | [(2R)-1-[3,10-Dihydroxy-12-[(2R)-2-(4-hydroxyphenoxy)carbonyloxypropyl]-2,6,7,11-tetramethoxy-4,9-dioxoperylen-1-yl]propan-2-yl] benzoate | IC50 | 10000.0 [1], 38000.0 [2], 77000.0 [3], 110000.0 [4] |
| [(2R)-1-[3,10-Dihydroxy-12-[(2R)-2-(4-hydroxyphenoxy)carbonyloxypropyl]-2,6,7,11-tetramethoxy-4,9-dioxoperylen-1-yl]propan-2-yl] benzoate | Ki | 17780.0 [1] |
 | 1-Hydroxy-5-[2-(2H-tetrazol-5-yl)ethyl]indazole | IC50 | 13000.0 [1], 300000.0 [2], 350000.0 [3] |
| 1-Hydroxy-5-[2-(2H-tetrazol-5-yl)ethyl]indazole | Ki | 3140.0 [1], 3800.0 [2] |
 | (4S)-4-[[(2S)-3-Carboxy-2-[[(2S)-2-[[2-(5-chloro-1H-indol-2-yl)acetyl]amino]-3-naphthalen-2-ylpropanoyl]amino]propanoyl]amino]-5-methoxy-5-oxopentanoic acid | IC50 | 6300.0 [1], 210000.0 [2], 680000.0 [3] |
| (4S)-4-[[(2S)-3-Carboxy-2-[[(2S)-2-[[2-(5-chloro-1H-indol-2-yl)acetyl]amino]-3-naphthalen-2-ylpropanoyl]amino]propanoyl]amino]-5-methoxy-5-oxopentanoic acid | Ki | 1300.0 [1], 1360.0 [2] |
 | 2-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetic acid | IC50 | 25000.0 [1], 280000.0 [2], 450000.0 [3] |
| 2-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetic acid | Ki | 4100.0 [1] |
 | 3-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)propanoic acid | IC50 | 48000.0 [1], 580000.0 [2], 790000.0 [3] |
| 3-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)propanoic acid | Ki | 3300.0 [1] |
 | 2-[[2-(4-Ethylphenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]-N-(2-phenylethyl)acetamide | Ki | 195470.0 [1], 364710.0 [2], 370000.0 [3] |
 | (5Z)-5-{[2,5-Dimethyl-1-(3-pyridinyl)-1H-pyrrol-3-yl]methylene}-3-phenyl-1,3-thiazolidine-2,4-dione | Ki | 40670.0 [1], 53510.0 [2], 54000.0 [3] |
 | 2-Phenoxybenzamide | Ki | 24390.0 [1], 180990.0 [2] |
 | Ethyl 4-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanoate | Ki | 52000.0 [1], 120000.0 [2] |
 | 4-[5-(3,4-Dimethoxy-benzylidene)-4-oxo-2-thioxo-thiazolidin-3-yl]-butyric acid | Ki | 46810.0 [1], 80340.0 [2] |
 | 2,3-Bis(4-chlorophenyl)quinoxaline-6-carboxylic acid | Ki | 8800.0 [1], 13000.0 [2] |
 | 5-[4-(4-Chlorophenoxy)phenyl]-3-isoxazolecarboxylic acid | Ki | 21000.0 [1], 77000.0 [2] |
 | Ethyl 2-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetate | Ki | 63000.0 [1], 150000.0 [2] |
 | Methyl 3-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)propanoate | Ki | 100000.0 [1] |
 | 2-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetonitrile | Ki | 130000.0 [1], 240000.0 [2] |
 | 3-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)propanenitrile | Ki | 39000.0 [1], 47000.0 [2] |
 | 4-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanenitrile | Ki | 120000.0 [1], 160000.0 [2] |
 | 8-[3-(2H-Tetrazol-5-yl)propyl]-13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaene | Ki | 51000.0 [1], 74000.0 [2] |
 | 2,3-DI(1,3-Benzodioxol-5-YL)-7-hydroxy-6-quinoxalinecarboxylic acid | Ki | 8700.0 [1], 12000.0 [2] |
 | 5H-[1,2,5]Oxadiazolo[3',4':5,6]pyrazino[2,3-b]indole | Ki | 120000.0 [1], 280000.0 [2] |
 | 3-[2-(1-Hydroxyindazol-5-yl)ethyl]-2H-1,2,4-oxadiazole-5-thione | Ki | 7240.0 [1], 70370.0 [2] |
 | 3-[(1-Hydroxybenzotriazol-5-yl)methyl]-2H-1,2,4-oxadiazole-5-thione | Ki | 42020.0 [1], 105900.0 [2] |
 | 1-Hydroxy-5-[2-(2H-tetrazol-5-yl)ethyl]benzotriazole | Ki | 3830.0 [1], 7600.0 [2] |
 | (4-Amino-1,2,5-oxadiazol-3-yl)(pyrrolidin-1-yl)methanone | Ki | 1700000.0 [1] |
 | 3-Butanoyl-1,8-dihydroxy-2-methylphenanthrene-9,10-dione | IC50 | 10000.0 [1] |
 | N-[(E)-(5-Methylfuran-2-yl)methylideneamino]-2-phenoxybenzamide | Ki | 1800.0 [1] |
 | 9H-Indeno[1,2-b][1,2,5]oxadiazolo[3,4-E]pyrazin-9-one | Ki | 310000.0 [1] |
 | 13-Oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-yliminothiourea | Ki | 240000.0 [1] |
 | CID 1416323 | Ki | 80000.0 [1] |
 | 4-Amino-1,2,5-oxadiazole-3-carboxamide | Ki | 2000000.0 [1] |
 | 1-[12-[2-(2,4-Dihydroxy-6-methylbenzoyl)oxypropyl]-3,10-dihydroxy-2,6,7,11-tetramethoxy-4,9-dioxoperylen-1-yl]propan-2-yl 2,4-dihydroxy-6-methylbenzoate | IC50 | 10000.0 [1] |
 | 13-Oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-yldiazene | Ki | 230000.0 [1] |
 | 2-Hydroxy-5-({3-[(phenylsulfonyl)amino]quinoxalin-2-yl}amino)benzoic acid | Ki | 13000.0 [1] |
 | 4-Amino-N-isobutyl-1,2,5-oxadiazole-3-carboxamide | Ki | 2000000.0 [1] |
 | 4-Amino-N-benzyl-1,2,5-oxadiazole-3-carboxamide | Ki | 1700000.0 [1] |
 | 2-[(3S,6S,9S,12S,16Z,21S)-12-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-5-amino-5-oxopentanoyl]amino]-21-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-12,21-dimethyl-6-(2-methylpropyl)-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclohenicos-16-en-3-yl]acetic acid | IC50 | 5000.0 [1] |
 | 2-[(3S,6S,9S,12S,16Z,21S)-12-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]-21-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-12,21-dimethyl-6-(2-methylpropyl)-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclohenicos-16-en-3-yl]acetic acid | IC50 | 5000.0 [1] |
 | Methyl (6R,6aS,14aR)-1,6,8,14a-tetrahydroxy-11-[[(2R,3S,4S,5S,6R)-4-hydroxy-3,5-dimethoxy-6-methyloxan-2-yl]amino]-6a-methoxy-3-methyl-7,9,12,14-tetraoxo-5,6-dihydrobenzo[a]tetracene-2-carboxylate | IC50 | 10000.0 [1] |
 | 1-Hydroxy-5-[2-(2H-tetrazol-1-ium-1-yl)ethyl]benzotriazole | Ki | 54200.0 [1] |
 | 1-Hydroxy-5-(2H-tetrazol-1-ium-1-ylmethoxymethyl)indazole | Ki | 13550.0 [1] |
 | 3-[(1-Hydroxybenzotriazol-5-yl)methyl]-4H-1,2,4-oxadiazol-5-one | Ki | 125100.0 [1] |
 | 3-[2-(1-Hydroxybenzotriazol-5-yl)ethyl]-4H-1,2,4-oxadiazol-5-one | Ki | 551250.0 [1] |
 | 3-[2-(1-Hydroxyindazol-5-yl)ethyl]-4H-1,2,4-oxadiazol-5-one | Ki | 97700.0 [1] |
 | 1-Hydroxy-5-(2H-tetrazol-5-ylmethyl)benzotriazole | Ki | 94400.0 [1] |
 | 1-Hydroxy-5-(2H-tetrazol-5-ylmethoxymethyl)benzotriazole | Ki | 155100.0 [1] |
 | 3-[2-(1-Hydroxybenzotriazol-5-yl)ethyl]-2H-1,2,4-oxadiazole-5-thione | Ki | 24360.0 [1] |
 | 1-Hydroxy-5-(2H-tetrazol-5-ylmethoxy)benzotriazole | Ki | 50400.0 [1] |
 | 5-[2-(2H-Tetrazol-5-yl)ethyl]-1H-indazole | Ki | 179930.0 [1] |
 | 1-Hydroxy-N-(2H-tetrazol-5-ylmethyl)indazol-5-amine | Ki | 3380.0 [1] |
 | 3-Bromo-5-fluoro-N-(1-hydroxyindazol-5-yl)-N-(2H-tetrazol-5-ylmethyl)benzamide | Ki | 28740.0 [1] |
 | 3-Chloro-N-(1-hydroxyindazol-5-yl)-N-(2H-tetrazol-5-ylmethyl)benzamide | Ki | 33140.0 [1] |
 | N-(1-Hydroxyindazol-5-yl)-N-(2H-tetrazol-5-ylmethyl)pyridine-3-carboxamide | Ki | 179930.0 [1] |
 | N-(1-Hydroxyindazol-5-yl)-3,5-dimethyl-N-(2H-tetrazol-5-ylmethyl)-1,2-oxazole-4-carboxamide | Ki | 16570.0 [1] |
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