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Cathepsin H Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
LeupeptinKi9200.0 [1]
Gallinamide AIC5030000.0 [1]
(S)-2-Amino-N-((S)-2-biphenyl-4-yl-1-cyano-ethyl)-butyramideIC5010000.0 [1]
(S)-2-Amino-N-((S)-2-biphenyl-4-yl-1-cyano-ethyl)-butyramideKi3700.0 [1]
2-Methyl-5-nitroquinoline-8-olKi89000.0 [1]
N-(1-Cyanocyclopropyl)-8-hydroxy-5-nitroquinoline-7-carboxamideKi329000.0 [1]
7-(Cyanomethylaminomethyl)-5-nitro-8-quinolinolKi129000.0 [1]
5-Nitro-8-(4-methylpiperidino)quinolineKi221000.0 [1]
PepstatinIC50100000.0 [1]
e-64IC50190.0 [1]
CID 11199915IC50100000.0 [1]
OdanacatibIC5010.0 [1]
(2S)-1-[(2S,3S)-3-Methyl-2-[[(2S,3S)-3-(propylcarbamoyl)oxirane-2-carbonyl]amino]pentanoyl]pyrrolidine-2-carboxylic acidIC50100000.0 [1]
CID 118253852IC5020000.0 [1]
N-[(2S)-1-[[(E,3S)-1-(Benzenesulfonyl)-5-phenylpent-1-en-3-yl]amino]-4-methyl-1-oxopentan-2-yl]morpholine-4-carboxamideKi1400.0 [1]
Grassystatin AIC5010000.0 [1]
(S)-Tert-butyl 1-oxohexan-2-ylcarbamateIC5013000.0 [1]
Cruzain-IN-1IC50125.89 [1]
9-(3,5-Difluorophenyl)-6-(ethylamino)-2-purinecarbonitrileIC50645.65 [1]
(S)-2-Amino-N-((S,E)-5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)pentanamideKi137.0 [1]
Pyrrolidine, 1-(4-nitro-1-naphthalenyl)-Ki251000.0 [1]
(2S)-1-Phenylpropan-2-yl [(2S)-1-oxohexan-2-yl]carbamateIC5040.0 [1]
3-Acetyl-8-bromo-5-chloro-2-(4-chlorophenylamino)quinolin-4(1H)-oneIC50100000.0 [1]
[(3S)-4,4-Dimethyl-2-oxooxolan-3-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC50500.0 [1]
(1R)-2-Methyl-1-(phenylmethyl)propyl[(1S)-1-formylpentyl]carbamateIC5018.0 [1]
1-(Phenylmethyl)cyclopentyl[(1S)-1-formylpentyl]carbamateIC5013000.0 [1]
(1-Benzylcyclobutyl)methyl N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC505000.0 [1]
[1-(3-Phenylpropyl)cyclobutyl]methyl N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC502000.0 [1]
[1-(2-Phenylethyl)cyclobutyl]methyl N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC502000.0 [1]
Benzyl N-[(2S)-1-[[(2S)-4-fluoro-3-oxo-1-phenylbutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamateIC50100000.0 [1]
(2R)-2-[[(1S)-1-(4-Bromophenyl)-2,2,2-trifluoroethyl]amino]-N-(1-cyanocyclopropyl)-3-methylsulfonylpropanamideIC5050000.0 [1]
(2S)-1-Cyclohexylpropan-2-yl 1-cyanopyrrolidine-2-carboxylateIC50580.0 [1]
[(2S)-1-Cyclohexylpropan-2-yl] N-[(3S)-1-cyanopyrrolidin-3-yl]carbamateIC508300.0 [1]
(2-Methyl-2-phenylpropyl) N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC505000.0 [1]
(2,2-Dimethyl-3-phenylpropyl) N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC505000.0 [1]
(1-Benzylcyclopentyl) N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5012000.0 [1]
[1-(4-Fluorobenzyl)cyclobutyl]methyl (1S)-1-[oxo(1H-pyrazol-5-ylamino)acetyl]pentylcarbamateIC50500.0 [1]
Gly-Phe-DMKIC5029000.0 [1]
P2,P3 Ketoamide derivativeIC505000.0 [1]
[1-[(4-Fluorophenyl)methyl]cyclobutyl]methyl N-[(3S)-7-(morpholine-4-carbonylamino)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC505000.0 [1]
(1-Benzylcyclopentyl)methyl N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC505000.0 [1]
(3S)-1-Diazo-3-[(aminoacetyl)amino]-4-(4-iodophenyl)-2-butanoneIC509800.0 [1]
1-(2-Benzyloxycarbonylamino-propionyl)-aziridine-2,3-dicarboxylic acid diethyl esterKi160000.0 [1]
Ethyl (2R,3R)-3-[[(2S)-4-methyl-1-oxo-1-phenylmethoxypentan-2-yl]carbamoyl]-1-[(2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-phenylpropanoyl]aziridine-2-carboxylateKi137000.0 [1]
1-((S)-2-Tert-Butoxycarbonylamino-3-phenyl-propionyl)-aziridine-2,3-dicarboxylic acid diethyl esterKi210000.0 [1]
Ethyl (2S,3S)-3-[[(2S)-4-methyl-1-oxo-1-phenylmethoxypentan-2-yl]carbamoyl]-1-[(2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-phenylpropanoyl]aziridine-2-carboxylateKi93000.0 [1]
[(3S)-4,4-Dimethyl-2-oxopyrrolidin-3-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5013000.0 [1]
[(2S)-1-Phenylpropan-2-yl] N-[(1E,2S)-1-(morpholine-4-carbonylhydrazinylidene)hexan-2-yl]carbamateIC50230.0 [1]
(3R,4R)-4-(2,3-Dimethylphenoxy)piperidin-3-olIC50100000.0 [1]
N-(Cyanomethyl)-8-hydroxy-5-nitroquinoline-7-carboxamideKi462000.0 [1]
(4S)-4-[[(2S)-2-[[(2S)-1-[(2S)-2-[[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-Acetamidoacetyl)amino]-5-carbamimidamidopentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-4-methylsulfanylbutanoyl]amino]carbamoylamino]propanoyl]pyrrolidine-2-carbonyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-5-[[(2R)-1-[[(2R)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-5-oxopentanoic acidKi7000.0 [1]
N-[[1-(1,3-Benzoxazol-2-yl)piperidin-4-yl]methyl]-8-hydroxy-5-nitroquinoline-7-carboxamideKi108000.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[[(2S)-1-[(2S)-1-[(2S)-2-[(4-Aminobenzoyl)amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]amino]carbamoylamino]-3-phenylpropanoyl]amino]-3-hydroxypropanoyl]-N-[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxy-3-nitrophenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamideKi1300.0 [1]
(4S,5R)-4-(2,3-Dimethylphenoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC502653.0 [1]
2-Bromo-4-nitronaphthalen-1-amineKi354000.0 [1]
cis-(S)-2-Amino-N-((1R,2R)-1-cyano-2-phenylcyclopropyl)-3-(thiophen-2-yl)propanamideIC5050000.0 [1]
(4S,5S)-4-(2,3-Dimethylphenoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC5030000.0 [1]
(4S,5R)-4-Phenoxy-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC506591.0 [1]
(4S,5R)-4-Phenylmethoxy-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC5010000.0 [1]
(4S,5R)-4-(2-Methylpropoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC5010000.0 [1]
(4S,5S)-4-Bromo-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC50100000.0 [1]
6-[[4-(4-Acetylpiperazin-1-yl)phenoxy]methyl]-7-[2-(4,4-difluorocyclohexyl)ethyl]pyrrolo[2,3-d]pyrimidine-2-carbonitrileKi10000.0 [1]
3-Acetyl-5,8-dichloro-2-(2,4-dichlorophenylamino)quinolin-4(1H)-oneIC50100000.0 [1]
3-((S)-1-Benzyloxycarbonyl-3-methyl-butylcarbamoyl)-aziridine-2-carboxylic acid ethyl esterKi260000.0 [1]
(2S)-1-Cyclohexylpropan-2-yl 1-cyanoazetidine-2-carboxylateIC5040.0 [1]
(1S)-2-Cyclohexyl-1-methylethyl 2-cyano-2-isopropylhydrazinecarboxylateKi0.46 [1]
(1S)-2-Cyclohexyl-1-methylethyl 2-cyano-2-methylhydrazinecarboxylateKi1.4 [1]
(Cyano-methyl-amino)-acetic acid (S)-2-cyclohexyl-1-methyl-ethyl esterKi13000.0 [1]
[(1S)-1,2,3,4-Tetrahydronaphthalen-1-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC502000.0 [1]
2-Adamantyl N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC505000.0 [1]
[(1S)-2,3-Dihydro-1H-inden-1-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5013000.0 [1]
(1,3,3-Trimethyl-2-bicyclo[2.2.1]heptanyl) N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5013000.0 [1]
[(3R,5R)-3,5-Dimethylcyclohexyl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5013000.0 [1]
[(3S,5R)-3,5-Dimethylcyclohexyl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5013000.0 [1]
2-Bicyclo[2.2.1]heptanyl N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5013000.0 [1]
{(S)-1-[(Morpholine-4-carbonyl)-hydrazonomethyl]-pentyl}-carbamic acid tert-butyl esterIC5013000.0 [1]
Tert-butyl N-[(1E,2S)-1-(2,3-dihydroindole-1-carbonylhydrazinylidene)hexan-2-yl]carbamateIC5013000.0 [1]
[(2R)-3-Methyl-1-phenylbutan-2-yl] N-[(1E,2S)-1-(morpholine-4-carbonylhydrazinylidene)hexan-2-yl]carbamateIC50190.0 [1]
(1-Benzylcyclopentyl) N-[(1E,2S)-1-(2,3-dihydroindole-1-carbonylhydrazinylidene)hexan-2-yl]carbamateIC5013000.0 [1]
(4S,5R)-4-Phenoxy-6-oxa-1-azabicyclo[3.2.1]octane-7-thioneIC50100000.0 [1]
5-((2,3-Dimethylphenoxy)methyl)-3-methyloxazolidin-2-oneIC50100000.0 [1]
4-(3-Chlorophenylamino)-6-(cyclopentylamino)-1,3,5-triazine-2-carbonitrileIC5014454.4 [1]
4-(Cyclopentylamino)-6-(3,5-difluorophenylamino)-1,3,5-triazine-2-carbonitrileIC5016218.1 [1]
3-Acetyl-5,8-dibromo-2-(4-bromophenylamino)quinolin-4(1H)-oneIC5091760.0 [1]
3-Acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-methylquinolin-4(1H)-oneIC5066520.0 [1]
3-Acetyl-8-chloro-2-(4-chlorophenylamino)-6-nitroquinolin-4(1H)-oneIC50145.0 [1]
3-Acetyl-2-(4-tert-butylphenylamino)-8-chloro-6-nitroquinolin-4(1H)-oneIC50100000.0 [1]
3-Acetyl-6-chloro-2-(2-chloro-4-methylanilino)-8-nitro-1H-quinolin-4-oneIC50100000.0 [1]
3-Acetyl-6-chloro-2-(2,4-dichloroanilino)-8-nitro-1H-quinolin-4-oneIC5032570.0 [1]
2-Amino-N-[(1R,2R)-1-cyano-2-phenylcyclopropyl]-3-(3-fluorothiophen-2-yl)propanamide;2,2,2-trifluoroacetic acidIC5050000.0 [1]
(2R)-2-Amino-N-[(1S,2S)-1-cyano-2-phenylcyclopropyl]-3-thiophen-2-ylpropanamide;2,2,2-trifluoroacetic acidIC5050000.0 [1]
(2S)-2-Amino-N-[(1R,2R)-1-cyano-2-phenylcyclopropyl]-3-thiophen-2-ylpropanamide;2,2,2-trifluoroacetic acidIC5050000.0 [1]
(3S,4R)-4-(2,3-Dimethylphenoxy)piperidin-3-olIC50100000.0 [1]
N-[(2R)-3-Benzylsulfonyl-1-oxo-1-[[(2S)-1-[4-(trifluoromethoxy)anilino]propan-2-yl]amino]propan-2-yl]morpholine-4-carboxamideKi30000.0 [1]
Items per page: 1 - 10 of 94
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cathepsin H Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/cathepsin-h-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Cathepsin H Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cathepsin-h-inhibitors-ic50-ki.
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